BE891580A - Derives de piperazine 1,4-disubstitues et leur procede de preparation - Google Patents

Derives de piperazine 1,4-disubstitues et leur procede de preparation

Info

Publication number
BE891580A
BE891580A BE0/206904A BE206904A BE891580A BE 891580 A BE891580 A BE 891580A BE 0/206904 A BE0/206904 A BE 0/206904A BE 206904 A BE206904 A BE 206904A BE 891580 A BE891580 A BE 891580A
Authority
BE
Belgium
Prior art keywords
preparation process
piperazine derivatives
disubstituted piperazine
disubstituted
derivatives
Prior art date
Application number
BE0/206904A
Other languages
English (en)
French (fr)
Original Assignee
Kyorin Seiyaku Kk
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Kyorin Seiyaku Kk filed Critical Kyorin Seiyaku Kk
Publication of BE891580A publication Critical patent/BE891580A/fr

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D263/00Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
    • C07D263/52Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings condensed with carbocyclic rings or ring systems
    • C07D263/54Benzoxazoles; Hydrogenated benzoxazoles
    • C07D263/56Benzoxazoles; Hydrogenated benzoxazoles with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 2
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D235/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
    • C07D235/02Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
    • C07D235/04Benzimidazoles; Hydrogenated benzimidazoles
    • C07D235/06Benzimidazoles; Hydrogenated benzimidazoles with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 2
    • C07D235/14Radicals substituted by nitrogen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pain & Pain Management (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Pyridine Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
BE0/206904A 1980-12-23 1981-12-22 Derives de piperazine 1,4-disubstitues et leur procede de preparation BE891580A (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP55182632A JPS57106663A (en) 1980-12-23 1980-12-23 1,4-disubstituted piperazine derivative and its preparation

Publications (1)

Publication Number Publication Date
BE891580A true BE891580A (fr) 1982-04-16

Family

ID=16121678

Family Applications (1)

Application Number Title Priority Date Filing Date
BE0/206904A BE891580A (fr) 1980-12-23 1981-12-22 Derives de piperazine 1,4-disubstitues et leur procede de preparation

Country Status (10)

Country Link
JP (1) JPS57106663A (xx)
KR (1) KR830007608A (xx)
AU (1) AU7877481A (xx)
BE (1) BE891580A (xx)
DE (1) DE3151123A1 (xx)
FR (1) FR2496661A1 (xx)
GB (1) GB2091255A (xx)
IT (1) IT1142620B (xx)
SE (1) SE8107680L (xx)
ZA (1) ZA818900B (xx)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2000051614A1 (en) * 1999-03-03 2000-09-08 Merck & Co., Inc. Inhibitors of prenyl-protein transferases

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4835154A (en) * 1987-06-01 1989-05-30 Smithkline Beckman Corporation 1-aralykyl-5-piperazinylmethyl-2-mercaptoimidazoles and 2-alkylthioimidazoles and their use as dopamine-βhydroxylase inhibitors
US5149700A (en) * 1990-05-30 1992-09-22 American Home Products Corporation Substituted arylsulfonamides and benzamides

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2297045A1 (fr) * 1975-01-10 1976-08-06 Delalande Sa Nouveaux (aroyl-2' eth-1' yl)-1 (acetamido-4'' piperazin-1'' yl methyl)-2 benzimidazoles a proprietes antisecretoire gastrique et antiulcereuse
YU39992B (en) * 1976-04-02 1985-06-30 Janssen Pharmaceutica Nv Process for obtaining new piperazine and piperidine derivatives

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2000051614A1 (en) * 1999-03-03 2000-09-08 Merck & Co., Inc. Inhibitors of prenyl-protein transferases

Also Published As

Publication number Publication date
JPS57106663A (en) 1982-07-02
FR2496661A1 (fr) 1982-06-25
DE3151123A1 (de) 1982-08-12
KR830007608A (ko) 1983-11-04
IT1142620B (it) 1986-10-08
SE8107680L (sv) 1982-06-24
ZA818900B (en) 1982-12-29
GB2091255A (en) 1982-07-28
IT8125742A0 (it) 1981-12-21
AU7877481A (en) 1982-07-01

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Legal Events

Date Code Title Description
RE Patent lapsed

Owner name: KYORIN PHARMACEUTICAL CO. LTD

Effective date: 19911231