BE891580A - Derives de piperazine 1,4-disubstitues et leur procede de preparation - Google Patents
Derives de piperazine 1,4-disubstitues et leur procede de preparationInfo
- Publication number
- BE891580A BE891580A BE0/206904A BE206904A BE891580A BE 891580 A BE891580 A BE 891580A BE 0/206904 A BE0/206904 A BE 0/206904A BE 206904 A BE206904 A BE 206904A BE 891580 A BE891580 A BE 891580A
- Authority
- BE
- Belgium
- Prior art keywords
- preparation process
- piperazine derivatives
- disubstituted piperazine
- disubstituted
- derivatives
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
- C07D263/52—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings condensed with carbocyclic rings or ring systems
- C07D263/54—Benzoxazoles; Hydrogenated benzoxazoles
- C07D263/56—Benzoxazoles; Hydrogenated benzoxazoles with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 2
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
- C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
- C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
- C07D235/06—Benzimidazoles; Hydrogenated benzimidazoles with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 2
- C07D235/14—Radicals substituted by nitrogen atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Life Sciences & Earth Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pain & Pain Management (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Pyridine Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP55182632A JPS57106663A (en) | 1980-12-23 | 1980-12-23 | 1,4-disubstituted piperazine derivative and its preparation |
Publications (1)
Publication Number | Publication Date |
---|---|
BE891580A true BE891580A (fr) | 1982-04-16 |
Family
ID=16121678
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BE0/206904A BE891580A (fr) | 1980-12-23 | 1981-12-22 | Derives de piperazine 1,4-disubstitues et leur procede de preparation |
Country Status (10)
Country | Link |
---|---|
JP (1) | JPS57106663A (xx) |
KR (1) | KR830007608A (xx) |
AU (1) | AU7877481A (xx) |
BE (1) | BE891580A (xx) |
DE (1) | DE3151123A1 (xx) |
FR (1) | FR2496661A1 (xx) |
GB (1) | GB2091255A (xx) |
IT (1) | IT1142620B (xx) |
SE (1) | SE8107680L (xx) |
ZA (1) | ZA818900B (xx) |
Cited By (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2000051614A1 (en) * | 1999-03-03 | 2000-09-08 | Merck & Co., Inc. | Inhibitors of prenyl-protein transferases |
Families Citing this family (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4835154A (en) * | 1987-06-01 | 1989-05-30 | Smithkline Beckman Corporation | 1-aralykyl-5-piperazinylmethyl-2-mercaptoimidazoles and 2-alkylthioimidazoles and their use as dopamine-βhydroxylase inhibitors |
US5149700A (en) * | 1990-05-30 | 1992-09-22 | American Home Products Corporation | Substituted arylsulfonamides and benzamides |
Family Cites Families (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2297045A1 (fr) * | 1975-01-10 | 1976-08-06 | Delalande Sa | Nouveaux (aroyl-2' eth-1' yl)-1 (acetamido-4'' piperazin-1'' yl methyl)-2 benzimidazoles a proprietes antisecretoire gastrique et antiulcereuse |
YU39992B (en) * | 1976-04-02 | 1985-06-30 | Janssen Pharmaceutica Nv | Process for obtaining new piperazine and piperidine derivatives |
-
1980
- 1980-12-23 JP JP55182632A patent/JPS57106663A/ja active Pending
-
1981
- 1981-12-21 SE SE8107680A patent/SE8107680L/xx not_active Application Discontinuation
- 1981-12-21 IT IT25742/81A patent/IT1142620B/it active
- 1981-12-22 AU AU78774/81A patent/AU7877481A/en not_active Abandoned
- 1981-12-22 BE BE0/206904A patent/BE891580A/fr not_active IP Right Cessation
- 1981-12-23 KR KR1019810005097A patent/KR830007608A/ko unknown
- 1981-12-23 GB GB8138720A patent/GB2091255A/en not_active Withdrawn
- 1981-12-23 FR FR8124075A patent/FR2496661A1/fr not_active Withdrawn
- 1981-12-23 DE DE19813151123 patent/DE3151123A1/de not_active Withdrawn
- 1981-12-23 ZA ZA818900A patent/ZA818900B/xx unknown
Cited By (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2000051614A1 (en) * | 1999-03-03 | 2000-09-08 | Merck & Co., Inc. | Inhibitors of prenyl-protein transferases |
Also Published As
Publication number | Publication date |
---|---|
JPS57106663A (en) | 1982-07-02 |
FR2496661A1 (fr) | 1982-06-25 |
DE3151123A1 (de) | 1982-08-12 |
KR830007608A (ko) | 1983-11-04 |
IT1142620B (it) | 1986-10-08 |
SE8107680L (sv) | 1982-06-24 |
ZA818900B (en) | 1982-12-29 |
GB2091255A (en) | 1982-07-28 |
IT8125742A0 (it) | 1981-12-21 |
AU7877481A (en) | 1982-07-01 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
RE | Patent lapsed |
Owner name: KYORIN PHARMACEUTICAL CO. LTD Effective date: 19911231 |