BE877567A - Nouveaux derives alcoxycarbonyl-3 benzodiazepines, leur procede de preparation et leur application en therapeutique - Google Patents
Nouveaux derives alcoxycarbonyl-3 benzodiazepines, leur procede de preparation et leur application en therapeutiqueInfo
- Publication number
- BE877567A BE877567A BE2/57941A BE2057941A BE877567A BE 877567 A BE877567 A BE 877567A BE 2/57941 A BE2/57941 A BE 2/57941A BE 2057941 A BE2057941 A BE 2057941A BE 877567 A BE877567 A BE 877567A
- Authority
- BE
- Belgium
- Prior art keywords
- alcoxycarbonyl
- new
- preparation process
- therapeutic application
- benzodiazepine derivatives
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D243/00—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
- C07D243/06—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4
- C07D243/10—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
- C07D243/14—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines
- C07D243/16—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals
- C07D243/18—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals substituted in position 2 by nitrogen, oxygen or sulfur atoms
- C07D243/24—Oxygen atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Engineering & Computer Science (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Biomedical Technology (AREA)
- Public Health (AREA)
- Pain & Pain Management (AREA)
- Anesthesiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GB95078 | 1978-01-10 |
Publications (1)
Publication Number | Publication Date |
---|---|
BE877567A true BE877567A (fr) | 1979-11-05 |
Family
ID=9713371
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BE2/57941A BE877567A (fr) | 1978-01-10 | 1979-07-09 | Nouveaux derives alcoxycarbonyl-3 benzodiazepines, leur procede de preparation et leur application en therapeutique |
Country Status (8)
Country | Link |
---|---|
JP (1) | JPS54151992A (ru) |
BE (1) | BE877567A (ru) |
CA (1) | CA1126730A (ru) |
CH (1) | CH637644A5 (ru) |
DE (1) | DE2900017A1 (ru) |
FR (1) | FR2414043A1 (ru) |
IT (1) | IT1118271B (ru) |
NL (1) | NL7900192A (ru) |
Families Citing this family (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US7160880B1 (en) | 1999-05-14 | 2007-01-09 | Cenes Limited | Short-acting benzodiazepines |
GB9911152D0 (en) * | 1999-05-14 | 1999-07-14 | Glaxo Group Ltd | Short-acting benzodiazepines |
KR20150081370A (ko) | 2006-07-10 | 2015-07-13 | 파이온 유케이 리미티드 | 속효형 벤조디아제핀 염 및 이의 중합체 형태 |
EP2450039A1 (en) | 2010-11-08 | 2012-05-09 | PAION UK Ltd. | Dosing regimen for sedation with CNS 7056 (Remimazolam) |
AR094963A1 (es) | 2013-03-04 | 2015-09-09 | Ono Pharmaceutical Co | Reacción de oxidación excelente en el índice de conversión |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3678043A (en) * | 1966-03-14 | 1972-07-18 | American Home Prod | 2,3-dihydro-2-oxo-1h-1,4-benzodiazepine-3-carboxylic acid esters and related compounds |
CH500997A (de) * | 1967-08-09 | 1970-12-31 | Hoffmann La Roche | Verfahren zur Herstellung von Benzodiazepin-Derivaten |
GB1538164A (en) * | 1976-05-05 | 1979-01-10 | Clin Midy | Benzodiazepine derivatives |
-
1979
- 1979-01-02 DE DE19792900017 patent/DE2900017A1/de not_active Withdrawn
- 1979-01-03 FR FR7900098A patent/FR2414043A1/fr active Granted
- 1979-01-08 JP JP32279A patent/JPS54151992A/ja active Pending
- 1979-01-09 IT IT67037/79A patent/IT1118271B/it active
- 1979-01-09 CH CH18779A patent/CH637644A5/fr not_active IP Right Cessation
- 1979-01-10 NL NL7900192A patent/NL7900192A/xx not_active Application Discontinuation
- 1979-01-10 CA CA319,406A patent/CA1126730A/fr not_active Expired
- 1979-07-09 BE BE2/57941A patent/BE877567A/xx not_active IP Right Cessation
Also Published As
Publication number | Publication date |
---|---|
JPS54151992A (en) | 1979-11-29 |
DE2900017A1 (de) | 1979-07-12 |
FR2414043B1 (ru) | 1982-03-26 |
CA1126730A (fr) | 1982-06-29 |
CH637644A5 (en) | 1983-08-15 |
FR2414043A1 (fr) | 1979-08-03 |
IT7967037A0 (it) | 1979-01-09 |
IT1118271B (it) | 1986-02-24 |
NL7900192A (nl) | 1979-07-12 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
RE | Patent lapsed |
Owner name: SANOFI Effective date: 19850731 |