BE877567A - Nouveaux derives alcoxycarbonyl-3 benzodiazepines, leur procede de preparation et leur application en therapeutique - Google Patents
Nouveaux derives alcoxycarbonyl-3 benzodiazepines, leur procede de preparation et leur application en therapeutiqueInfo
- Publication number
- BE877567A BE877567A BE2/57941A BE2057941A BE877567A BE 877567 A BE877567 A BE 877567A BE 2/57941 A BE2/57941 A BE 2/57941A BE 2057941 A BE2057941 A BE 2057941A BE 877567 A BE877567 A BE 877567A
- Authority
- BE
- Belgium
- Prior art keywords
- alcoxycarbonyl
- new
- preparation process
- therapeutic application
- benzodiazepine derivatives
- Prior art date
Links
- 229940053197 benzodiazepine derivative antiepileptics Drugs 0.000 title 1
- 150000001557 benzodiazepines Chemical class 0.000 title 1
- 238000002360 preparation method Methods 0.000 title 1
- 230000001225 therapeutic effect Effects 0.000 title 1
Classifications
- 
        - C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D243/00—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
- C07D243/06—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4
- C07D243/10—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
- C07D243/14—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines
- C07D243/16—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals
- C07D243/18—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals substituted in position 2 by nitrogen, oxygen or sulfur atoms
- C07D243/24—Oxygen atoms
 
- 
        - A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
 
- 
        - A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
 
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Pain & Pain Management (AREA)
- Anesthesiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title | 
|---|---|---|---|
| GB95078 | 1978-01-10 | 
Publications (1)
| Publication Number | Publication Date | 
|---|---|
| BE877567A true BE877567A (fr) | 1979-11-05 | 
Family
ID=9713371
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date | 
|---|---|---|---|
| BE2/57941A BE877567A (fr) | 1978-01-10 | 1979-07-09 | Nouveaux derives alcoxycarbonyl-3 benzodiazepines, leur procede de preparation et leur application en therapeutique | 
Country Status (8)
| Country | Link | 
|---|---|
| JP (1) | JPS54151992A (enrdf_load_html_response) | 
| BE (1) | BE877567A (enrdf_load_html_response) | 
| CA (1) | CA1126730A (enrdf_load_html_response) | 
| CH (1) | CH637644A5 (enrdf_load_html_response) | 
| DE (1) | DE2900017A1 (enrdf_load_html_response) | 
| FR (1) | FR2414043A1 (enrdf_load_html_response) | 
| IT (1) | IT1118271B (enrdf_load_html_response) | 
| NL (1) | NL7900192A (enrdf_load_html_response) | 
Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title | 
|---|---|---|---|---|
| US7160880B1 (en) | 1999-05-14 | 2007-01-09 | Cenes Limited | Short-acting benzodiazepines | 
| GB9911152D0 (en) * | 1999-05-14 | 1999-07-14 | Glaxo Group Ltd | Short-acting benzodiazepines | 
| SI2081921T1 (sl) | 2006-07-10 | 2011-01-31 | Paion Uk Ltd | Soli benzodiazepina s kratkotrajnim učinkom ter njihove polimorfne oblike | 
| EP2450039A1 (en) | 2010-11-08 | 2012-05-09 | PAION UK Ltd. | Dosing regimen for sedation with CNS 7056 (Remimazolam) | 
| AR094963A1 (es) | 2013-03-04 | 2015-09-09 | Ono Pharmaceutical Co | Reacción de oxidación excelente en el índice de conversión | 
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title | 
|---|---|---|---|---|
| US3678043A (en) * | 1966-03-14 | 1972-07-18 | American Home Prod | 2,3-dihydro-2-oxo-1h-1,4-benzodiazepine-3-carboxylic acid esters and related compounds | 
| CH500997A (de) * | 1967-08-09 | 1970-12-31 | Hoffmann La Roche | Verfahren zur Herstellung von Benzodiazepin-Derivaten | 
| GB1538164A (en) * | 1976-05-05 | 1979-01-10 | Clin Midy | Benzodiazepine derivatives | 
- 
        1979
        - 1979-01-02 DE DE19792900017 patent/DE2900017A1/de not_active Withdrawn
- 1979-01-03 FR FR7900098A patent/FR2414043A1/fr active Granted
- 1979-01-08 JP JP32279A patent/JPS54151992A/ja active Pending
- 1979-01-09 CH CH18779A patent/CH637644A5/fr not_active IP Right Cessation
- 1979-01-09 IT IT67037/79A patent/IT1118271B/it active
- 1979-01-10 CA CA319,406A patent/CA1126730A/fr not_active Expired
- 1979-01-10 NL NL7900192A patent/NL7900192A/xx not_active Application Discontinuation
- 1979-07-09 BE BE2/57941A patent/BE877567A/xx not_active IP Right Cessation
 
Also Published As
| Publication number | Publication date | 
|---|---|
| JPS54151992A (en) | 1979-11-29 | 
| FR2414043B1 (enrdf_load_html_response) | 1982-03-26 | 
| CH637644A5 (en) | 1983-08-15 | 
| DE2900017A1 (de) | 1979-07-12 | 
| FR2414043A1 (fr) | 1979-08-03 | 
| NL7900192A (nl) | 1979-07-12 | 
| IT1118271B (it) | 1986-02-24 | 
| CA1126730A (fr) | 1982-06-29 | 
| IT7967037A0 (it) | 1979-01-09 | 
Similar Documents
| Publication | Publication Date | Title | 
|---|---|---|
| BE892270A (fr) | Nouveaux derives aminomethyl-5 oxazolidiniques, leur procede de preparation et leur application en therapeutique | |
| BE890962R (fr) | Nouveaux derives du nor-tropane, leur procede de preparation et leur application en therapeutique | |
| BE892758A (fr) | Derives phenylcyclobutyliques, leur procede de preparation et leur application therapeutique | |
| FR2504920B1 (fr) | Derives phenylcyclobutyliques, leur procede de preparation et leur application therapeutique | |
| BE875174A (fr) | Nouveaux derives de carbostyrile, leur procede de preparation et leurs applications en therapeutique | |
| BE878723A (fr) | Derives de 4-anilinoquinazoline, leur procede de preparation et leur application en therapeutique | |
| BE881134A (fr) | Nouveaux derives du nor-tropane, leur procede de preparation et leur application en therapeutique | |
| BE865632A (fr) | Nouveaux derives de cephalosporine, leur procede de preparation et leur application en therapeutique | |
| FR2532648B1 (fr) | Derives de carbostyrile, leur procede de preparation et leur application en therapeutique | |
| LU76848A1 (fr) | Nouveaux hydroxymethyl-5 oxazolidinone-2, leur procede de preparation et leur application therapeutique | |
| BE854268A (fr) | Pyrrolidones, leur procede de preparation et leur application therapeutique | |
| FR2506306B1 (fr) | Nouveaux derives de l'amidinopiperidine, leur procede de preparation et leur application en therapeutique | |
| BE864312A (fr) | Nouveaux derives de la pyrrolidine, leur procede de preparation et leur application en therapeutique | |
| MA19331A1 (fr) | Derives de la thieno - pyridinone , leur procede de preparation et leur application therapeutique . | |
| BE883124A (fr) | Nouveaux derives de la 5h-furanone-2 et de la 3h-dihydro-furanone-2, leur procede de preparation et leur application en therapeutique | |
| FR2315925A1 (fr) | Nouveaux derives de 5-benzyle-2-oxazolidone, leur procede de preparation et leur application en therapeutique | |
| BE891526A (fr) | Nouveaux derives aminoalcoyl heterocycliques, leur procede de preparation et leur application en therapeutique | |
| BE883713A (fr) | Nouveau derives de carbostyrile, leur procede de preparation et leur application en therapeutique | |
| LU79606A1 (fr) | Derives de bisamidine,leur procede de preparation et leur application therapeutique | |
| BE877567A (fr) | Nouveaux derives alcoxycarbonyl-3 benzodiazepines, leur procede de preparation et leur application en therapeutique | |
| BE884620A (fr) | Nouveaux derives d'halovincamone, leur procede de preparation et medicaments les contenant | |
| FR2520739B1 (fr) | Nouveaux derives d'ester indoleacetique, leur procede de preparation et leur application en therapeutique | |
| FR2317930A1 (fr) | Nouveaux derives d'apovincaminol, leur procede de preparation et leur application | |
| FR2477142B1 (fr) | Nouveaux derives de la nitrosouree, leur procede de preparation et leur application en therapeutique | |
| FR2514768B1 (fr) | Derives de phosphoramide, leur procede de preparation et leur application en therapeutique | 
Legal Events
| Date | Code | Title | Description | 
|---|---|---|---|
| RE | Patent lapsed | Owner name: SANOFI Effective date: 19850731 |