BE872347A - Amides substitues de l- et dl-phenylglycine, leur procede de production et composition pharmaceutique les contenant - Google Patents

Amides substitues de l- et dl-phenylglycine, leur procede de production et composition pharmaceutique les contenant

Info

Publication number
BE872347A
BE872347A BE191995A BE191995A BE872347A BE 872347 A BE872347 A BE 872347A BE 191995 A BE191995 A BE 191995A BE 191995 A BE191995 A BE 191995A BE 872347 A BE872347 A BE 872347A
Authority
BE
Belgium
Prior art keywords
phenylglycin
amides
substitute
pharmaceutical composition
composition containing
Prior art date
Application number
BE191995A
Other languages
English (en)
French (fr)
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of BE872347A publication Critical patent/BE872347A/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K5/00Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06Dipeptides
    • C07K5/06008Dipeptides with the first amino acid being neutral
    • C07K5/06078Dipeptides with the first amino acid being neutral and aromatic or cycloaliphatic
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/08Vasodilators for multiple indications
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
BE191995A 1977-11-30 1978-11-28 Amides substitues de l- et dl-phenylglycine, leur procede de production et composition pharmaceutique les contenant BE872347A (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB4997577 1977-11-30

Publications (1)

Publication Number Publication Date
BE872347A true BE872347A (fr) 1979-05-28

Family

ID=10454182

Family Applications (1)

Application Number Title Priority Date Filing Date
BE191995A BE872347A (fr) 1977-11-30 1978-11-28 Amides substitues de l- et dl-phenylglycine, leur procede de production et composition pharmaceutique les contenant

Country Status (20)

Country Link
US (1) US4218474A (es)
JP (1) JPS5484546A (es)
AR (1) AR219957A1 (es)
AT (1) AT362770B (es)
AU (1) AU507028B2 (es)
BE (1) BE872347A (es)
CA (1) CA1101846A (es)
DE (1) DE2851435C2 (es)
DK (1) DK531178A (es)
ES (1) ES475514A1 (es)
FI (1) FI783638A (es)
FR (1) FR2410644A2 (es)
IE (1) IE47635B1 (es)
IL (1) IL56064A (es)
IT (1) IT1192590B (es)
LU (1) LU80596A1 (es)
NL (1) NL7811692A (es)
PH (1) PH14681A (es)
PT (1) PT68834A (es)
SE (1) SE7812268L (es)

Families Citing this family (21)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS58224427A (ja) * 1982-06-23 1983-12-26 Canon Electronics Inc 複合磁気ヘツド
JPS5921656A (ja) * 1982-07-28 1984-02-03 Takeda Chem Ind Ltd ポリペプチド誘導体
US4563352A (en) * 1982-10-04 1986-01-07 The Salk Institute For Biological Studies Human pancreatic GRF
US4595677A (en) * 1982-12-03 1986-06-17 Ciba-Geigy Corporation Substituted tetrapeptides
JPS59141547A (ja) * 1983-02-01 1984-08-14 Eisai Co Ltd 鎮痛作用を有する新規ペプタイドおよび製法
GB8322414D0 (en) * 1983-08-19 1983-09-21 Szelke M Renin inhibitors
AU598444B2 (en) * 1984-03-01 1990-06-28 Vernon Erk Method of prophylaxis or treatment of atherosclerosis
WO1985003874A1 (en) * 1984-03-01 1985-09-12 Vernon Erk Method of treating depression in vertebrates
AU598443B2 (en) * 1984-03-01 1990-06-28 Vernon Erk A method of treating hypoglycemia in vertebrates
EP0174957A4 (en) * 1984-03-01 1987-11-09 Vernon Erk METHOD FOR THE TREATMENT OF MEMORY DISORDERS IN ELDERLY PEOPLE.
EP0181342B1 (en) * 1984-03-01 1992-10-28 ERK, Vernon Method of treating hypertension in vertebrates
US4668663A (en) * 1984-03-27 1987-05-26 Merck & Co., Inc. Renin inhibitors containing homophe8
US4661473A (en) * 1984-03-27 1987-04-28 Merck & Co., Inc. Renin inhibitors containing peptide isosteres
US4659693A (en) * 1984-04-30 1987-04-21 Syntex (U.S.A.) Inc. N,N'-dialkyl substituted guanidino amino acyl residue substituted GRF-analog peptides
DE3527356A1 (de) * 1985-07-31 1987-02-05 Degussa Verfahren zur verbesserung der fruchtbarkeit von haustieren
US5252718A (en) * 1986-04-22 1993-10-12 The Salk Institute For Biological Studies Fibroblast growth factor antagonists
ATE122357T1 (de) * 1988-01-28 1995-05-15 Polygen Holding Corp Polypeptide mit hormonwachstumsbefreiender wirkung.
NL1010506C2 (nl) * 1998-11-06 2000-05-09 Dsm Nv Werkwijze voor de bereiding van bêta-lactam antibiotica.
KR100389644B1 (ko) * 2001-02-26 2003-06-27 한미약품 주식회사 4-히드록시페닐글리신 무수물 및 이의 제조방법
US7230097B2 (en) * 2003-03-10 2007-06-12 Lupin Ltd. Process for preparation of 7-[α-Amino (4-hydroxyphenyl) acetamido]-3-substituted-3-cephem-4-carboxylic acid
JP1610197S (es) 2017-09-25 2018-07-30

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2868818A (en) * 1953-12-15 1959-01-13 Merck & Co Inc Alpha methyl phenylalanines
US2833764A (en) * 1954-11-18 1958-05-06 American Cyanamid Co O-methyl-l-tyrosyl amides and their preparation
US3725470A (en) * 1969-05-14 1973-04-03 Hoffmann La Roche Amino acid derivatives
ES400897A1 (es) * 1972-03-18 1975-02-01 Beecham Group Ltd Un procedimiento para la preparacion de alfa-amino-p-hidro-xibencilpenicilina o de un ester de grafito.
DE2510634A1 (de) * 1975-03-12 1976-09-23 Boehringer Mannheim Gmbh L-3-(3,4-dihydroxy-phenyl)-2- methyl-alanin-peptide und verfahren zu deren herstellung
NL7514300A (nl) * 1975-12-09 1977-06-13 Stamicarbon Werkwijze voor de bereiding van optisch actief fenylglycineamide.
US4111981A (en) * 1975-12-15 1978-09-05 Smithkline Corporation Intermediates for preparing substituted phenylglycylcephalosporins
GB1547206A (en) * 1976-09-28 1979-06-06 Pfizer Ltd Pharmaceutical compositions
PH14064A (en) * 1977-05-06 1981-01-26 Pfizer Phenylgycine derivatives,pharmaceutical compositions and method of use

Also Published As

Publication number Publication date
IL56064A0 (en) 1979-01-31
IE47635B1 (en) 1984-05-16
FR2410644B2 (es) 1982-10-08
FR2410644A2 (fr) 1979-06-29
JPS5484546A (en) 1979-07-05
CA1101846A (en) 1981-05-26
AU4200878A (en) 1979-06-07
ATA850678A (de) 1980-11-15
ES475514A1 (es) 1979-04-01
LU80596A1 (fr) 1980-06-05
JPS5740139B2 (es) 1982-08-25
SE7812268L (sv) 1979-05-31
DK531178A (da) 1979-05-31
PT68834A (en) 1978-12-01
AR219957A1 (es) 1980-09-30
IT7830290A0 (it) 1978-11-28
IT1192590B (it) 1988-04-20
DE2851435A1 (de) 1979-06-13
IL56064A (en) 1982-01-31
DE2851435C2 (de) 1982-11-25
FI783638A (fi) 1979-05-31
AT362770B (de) 1981-06-10
AU507028B2 (en) 1980-01-31
IE782359L (en) 1979-05-30
NL7811692A (nl) 1979-06-01
US4218474A (en) 1980-08-19
PH14681A (en) 1981-11-10

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Legal Events

Date Code Title Description
RE Patent lapsed

Owner name: PFIZER CORP.

Effective date: 19861130