BE865851A - Dipyrido(4,3-b) (3,4-f) indoles, procede d'obtention, application therapeutique et compositions pharmaceutiques les contenant - Google Patents

Dipyrido(4,3-b) (3,4-f) indoles, procede d'obtention, application therapeutique et compositions pharmaceutiques les contenant

Info

Publication number
BE865851A
BE865851A BE186694A BE186694A BE865851A BE 865851 A BE865851 A BE 865851A BE 186694 A BE186694 A BE 186694A BE 186694 A BE186694 A BE 186694A BE 865851 A BE865851 A BE 865851A
Authority
BE
Belgium
Prior art keywords
dipyrido
indoles
obtaining
pharmaceutical compositions
compositions containing
Prior art date
Application number
BE186694A
Other languages
English (en)
Inventor
E Bisagni
C Ducrocq
C Rivalle
P Tambourin
F Wendling
J C Chermann
L Montagnier
Original Assignee
Anvar
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Anvar filed Critical Anvar
Publication of BE865851A publication Critical patent/BE865851A/fr
Priority to FR7908813A priority Critical patent/FR2422662A2/fr

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • A61P35/02Antineoplastic agents specific for leukemia
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C205/00Compounds containing nitro groups bound to a carbon skeleton
    • C07C205/44Compounds containing nitro groups bound to a carbon skeleton the carbon skeleton being further substituted by —CHO groups
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C205/00Compounds containing nitro groups bound to a carbon skeleton
    • C07C205/49Compounds containing nitro groups bound to a carbon skeleton the carbon skeleton being further substituted by carboxyl groups
    • C07C205/56Compounds containing nitro groups bound to a carbon skeleton the carbon skeleton being further substituted by carboxyl groups having nitro groups bound to carbon atoms of six-membered aromatic rings and carboxyl groups bound to acyclic carbon atoms of the carbon skeleton
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C247/00Compounds containing azido groups
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D217/00Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems
    • C07D217/22Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the nitrogen-containing ring
    • C07D217/24Oxygen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/12Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains three hetero rings
    • C07D487/14Ortho-condensed systems
BE186694A 1977-04-13 1978-04-10 Dipyrido(4,3-b) (3,4-f) indoles, procede d'obtention, application therapeutique et compositions pharmaceutiques les contenant BE865851A (fr)

Priority Applications (1)

Application Number Priority Date Filing Date Title
FR7908813A FR2422662A2 (fr) 1978-04-10 1979-04-06 Dipyrido (4,3-b) (3,4-f) indoles, procede d'obtention, application therapeutique et compositions pharmaceutiques les contenant

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR7711148A FR2387229A1 (fr) 1977-04-13 1977-04-13 Dipyrido (4,3-b) (3,4-f) indoles, procede d'obtention, application therapeutique et compositions pharmaceutiques les contenant

Publications (1)

Publication Number Publication Date
BE865851A true BE865851A (fr) 1978-10-10

Family

ID=9189361

Family Applications (1)

Application Number Title Priority Date Filing Date
BE186694A BE865851A (fr) 1977-04-13 1978-04-10 Dipyrido(4,3-b) (3,4-f) indoles, procede d'obtention, application therapeutique et compositions pharmaceutiques les contenant

Country Status (12)

Country Link
US (2) US4266060A (fr)
JP (1) JPS549299A (fr)
BE (1) BE865851A (fr)
CA (1) CA1117945A (fr)
CH (1) CH633796A5 (fr)
DE (1) DE2815724A1 (fr)
ES (1) ES468721A1 (fr)
FR (1) FR2387229A1 (fr)
GB (1) GB1603228A (fr)
IT (1) IT1095582B (fr)
LU (1) LU79422A1 (fr)
NL (1) NL184895C (fr)

Families Citing this family (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4334070A (en) * 1980-12-15 1982-06-08 Hoffmann-La Roche Inc. Cycloalka[4,5]pyrrolo[2,3-g]isoquinolines
DK158666C (da) * 1982-11-04 1990-11-19 Glaxo Group Ltd Analogifremgangsmaade til fremstilling af 5,14-dihydrobenz-oe5,6aa-isoindolooe2,1-baa-isoquinolin-8,13-dion
DE3576066D1 (de) * 1984-05-03 1990-03-29 Glaxo Group Ltd Isochinolinderivate.
JPH0642591B2 (ja) * 1984-11-30 1994-06-01 ミノルタカメラ株式会社 プリント配線基板の製造方法
NO872963L (no) * 1986-07-29 1988-02-01 Glaxo Group Ltd Isokinolinderivater.
DK616087A (da) * 1986-11-27 1988-05-28 Glaxo Group Ltd Isoquinolinderivater og farmaceutiske praeparater indeholdende dem
GB8800312D0 (en) * 1988-01-07 1988-02-10 Glaxo Group Ltd Process
FR2627493B1 (fr) * 1988-02-23 1991-10-31 Sanofi Sa Procede de preparation de derives d'isoquinoleine
FR2645861A1 (fr) * 1989-04-17 1990-10-19 Inst Nat Sante Rech Med Utilisation de dipyrido (4,3-b) (3,4-f) indoles pour la preparation de medicaments utiles pour le traitement du sida
US5281608A (en) * 1992-08-28 1994-01-25 American Home Products Corporation Substituted tetrahydropyrido[3',4':4,5]-pyrrolo[3,2-c]quinolines
FR2859474B1 (fr) * 2003-09-04 2006-01-13 Centre Nat Rech Scient Utilisation de composes derives d'indole pour la preparation d'un medicament utile pour le traitement de maladies genetiques resultant de l'alteration des processus d'epissage
AU2005206571B8 (en) * 2004-01-23 2010-09-02 Amgen Inc. Compounds and methods of use
KR101982461B1 (ko) 2009-06-12 2019-05-24 아비박스 조기 노화, 구체적으로 조로증을 치료하는데 유용한 화합물
EP2266972A1 (fr) * 2009-06-12 2010-12-29 Splicos Nouvelles molécules chimiques qui inhibent le mécanisme d'épissage pour le traitement de maladies résultant d'anomalies d'épissage
US10253020B2 (en) 2009-06-12 2019-04-09 Abivax Compounds for preventing, inhibiting, or treating cancer, AIDS and/or premature aging
EP2465502A1 (fr) 2010-12-15 2012-06-20 Société Splicos Composés utiles pour traiter le SIDA
EP2757161A1 (fr) 2013-01-17 2014-07-23 Splicos miRNA-124 comme biomarqueur de l'infection virale
EP3016656B1 (fr) 2013-07-05 2021-09-08 Abivax Composés bicycliques utiles pour le traitement de maladies causées par des rétrovirus
EP2974729A1 (fr) 2014-07-17 2016-01-20 Abivax Dérivés de quinoléine utilisés dans le traitement de maladies inflammatoires

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2248828B1 (fr) * 1973-10-29 1977-04-15 Anvar
US3933827A (en) * 1974-10-29 1976-01-20 Hoffmann-La Roche Inc. 9-Acyloxy-5,11-dimethyl-6H-pyrido[4,3-B]carbazoles

Also Published As

Publication number Publication date
DE2815724A1 (de) 1978-10-26
FR2387229A1 (fr) 1978-11-10
DE2815724C2 (fr) 1991-02-14
US4444776A (en) 1984-04-24
IT1095582B (it) 1985-08-10
JPS6225670B2 (fr) 1987-06-04
NL184895C (nl) 1989-12-01
JPS549299A (en) 1979-01-24
ES468721A1 (es) 1978-12-16
NL7803951A (nl) 1978-10-17
FR2387229B1 (fr) 1980-05-09
IT7822254A0 (it) 1978-04-12
CA1117945A (fr) 1982-02-09
CH633796A5 (fr) 1982-12-31
GB1603228A (en) 1981-11-18
NL184895B (nl) 1989-07-03
US4266060A (en) 1981-05-05
LU79422A1 (fr) 1979-11-07

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Legal Events

Date Code Title Description
RE Patent lapsed

Owner name: AGENCE NATIONALE DE VALORISATION DE LA RECHERCHE

Effective date: 19940430