BE848696A - Derives de la 3,4-dihydro-quinazoline a activite antiallergique et procede pour leur preparation, - Google Patents

Derives de la 3,4-dihydro-quinazoline a activite antiallergique et procede pour leur preparation,

Info

Publication number
BE848696A
BE848696A BE172653A BE172653A BE848696A BE 848696 A BE848696 A BE 848696A BE 172653 A BE172653 A BE 172653A BE 172653 A BE172653 A BE 172653A BE 848696 A BE848696 A BE 848696A
Authority
BE
Belgium
Prior art keywords
quinazoline
dihydro
derivatives
preparation
antiallergic activity
Prior art date
Application number
BE172653A
Other languages
English (en)
French (fr)
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed filed Critical
Publication of BE848696A publication Critical patent/BE848696A/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72Quinazolines; Hydrogenated quinazolines
    • C07D239/86Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 4
    • C07D239/88Oxygen atoms
    • C07D239/91Oxygen atoms with aryl or aralkyl radicals attached in position 2 or 3
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/08Antiallergic agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72Quinazolines; Hydrogenated quinazolines
    • C07D239/86Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 4
    • C07D239/88Oxygen atoms
    • C07D239/90Oxygen atoms with acyclic radicals attached in position 2 or 3
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72Quinazolines; Hydrogenated quinazolines
    • C07D239/86Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 4
    • C07D239/93Sulfur atoms

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pulmonology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Immunology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
BE172653A 1975-12-05 1976-11-24 Derives de la 3,4-dihydro-quinazoline a activite antiallergique et procede pour leur preparation, BE848696A (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
IT29998/75A IT1050750B (it) 1975-12-05 1975-12-05 Derivati della 3.4 di idro chinazolina

Publications (1)

Publication Number Publication Date
BE848696A true BE848696A (fr) 1977-03-16

Family

ID=11228830

Family Applications (1)

Application Number Title Priority Date Filing Date
BE172653A BE848696A (fr) 1975-12-05 1976-11-24 Derives de la 3,4-dihydro-quinazoline a activite antiallergique et procede pour leur preparation,

Country Status (22)

Country Link
US (1) US4251531A (no)
JP (1) JPS5271485A (no)
AT (1) AT355029B (no)
AU (1) AU505660B2 (no)
BE (1) BE848696A (no)
CA (1) CA1084051A (no)
CH (2) CH626073A5 (no)
CS (1) CS194786B2 (no)
DE (1) DE2654215A1 (no)
DK (1) DK147855C (no)
FI (1) FI64359C (no)
FR (1) FR2333511A1 (no)
GB (1) GB1523081A (no)
HU (1) HU177817B (no)
IL (1) IL50849A (no)
IT (1) IT1050750B (no)
NL (1) NL7613450A (no)
NO (1) NO146095C (no)
NZ (1) NZ182778A (no)
SE (1) SE7613588L (no)
SU (1) SU786894A3 (no)
ZA (1) ZA766745B (no)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL69274A (en) * 1982-08-05 1986-08-31 Erba Farmitalia (substituted amino)derivatives of 3-benzylidene-pyrrolo(2,1-b)quinazolin-9-ones and 6-benzylidene-pyrido(2,1-b)quinazolin-11-ones,their preparation and pharmaceutical compositions containing them
JPS5925224U (ja) * 1982-08-10 1984-02-16 株式会社根来 かばん
US4666913A (en) * 1985-11-22 1987-05-19 William H. Rorer, Inc. Hydroxy and aminothiazolyl-benzodiazinone compounds, cardiotonic compositions including the same, and their uses
GB8827988D0 (en) * 1988-11-30 1989-01-05 Smith Kline French Lab Chemical compounds
US5430148A (en) * 1992-03-31 1995-07-04 Agouron Pharmaceuticals, Inc. Antiproliferative quinazolines
WO1999061406A2 (en) * 1998-05-22 1999-12-02 Abbott Laboratories Antiangiogenic drug to treat cancer, arthritis and retinopathy
US6632961B1 (en) 1998-05-22 2003-10-14 Abbott Laboratories Antiangiogenic drug to treat cancer, arthritis and retinopathy
CO5170498A1 (es) * 1999-05-28 2002-06-27 Abbott Lab Biaril sulfonamidas son utiles como inhibidores de proliferacion celular
US7893071B2 (en) * 2001-04-23 2011-02-22 University Of Virginia Patent Foundation Synthesis and evaluation of novel phthalimide mimics as anti-angiogenic
DE602004025803D1 (de) * 2003-06-06 2010-04-15 Arexis Ab Verwendung von kondensierten heterozyklischen verbindungen als scce-hemmern zur behandlung von hautzuständen
CN100518740C (zh) * 2003-06-06 2009-07-29 阿里克斯股份公司 杂环化合物作为scce抑制剂的制药用途
EP2050739B1 (en) * 2006-08-08 2016-07-06 ASKA Pharmaceutical Co., Ltd. Quinazoline derivative
DK2118074T3 (en) 2007-02-01 2014-03-10 Resverlogix Corp Compounds for the prevention and treatment of cardiovascular diseases
NZ755378A (en) 2009-03-18 2022-07-29 Resverlogix Corp Novel quinazolinones and related compounds for use as anti-inflammatory agents
US9757368B2 (en) 2009-04-22 2017-09-12 Resverlogix Corp. Anti-inflammatory agents
CA2977308A1 (en) 2015-03-13 2016-09-22 Resverlogix Corp. Compositions and therapeutic methods for the treatment of complement-associated diseases
GB201510254D0 (en) * 2015-06-12 2015-07-29 Syngenta Participations Ag Improvements in or relating to organic compounds
CA3105174A1 (en) * 2018-06-27 2020-01-02 Reborna Biosciences, Inc. Prophylactic or therapeutic agent for spinal muscular atrophy

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3696102A (en) * 1970-03-09 1972-10-03 Pfizer & Co C Process for the synthesis of substituted quinazolin-4-ones

Also Published As

Publication number Publication date
IL50849A (en) 1980-11-30
SU786894A3 (ru) 1980-12-07
GB1523081A (en) 1978-08-31
AT355029B (de) 1980-02-11
CS194786B2 (en) 1979-12-31
FR2333511A1 (fr) 1977-07-01
DE2654215A1 (de) 1977-06-16
NL7613450A (nl) 1977-06-07
DK147855B (da) 1984-12-24
ATA894376A (de) 1979-07-15
US4251531A (en) 1981-02-17
CH626075A5 (no) 1981-10-30
JPS5543464B2 (no) 1980-11-06
AU505660B2 (en) 1979-11-29
NZ182778A (en) 1978-07-28
DK147855C (da) 1985-06-10
SE7613588L (sv) 1977-06-06
NO764135L (no) 1977-06-07
ZA766745B (en) 1977-10-26
HU177817B (en) 1981-12-28
IT1050750B (it) 1981-03-20
FI64359C (fi) 1983-11-10
NO146095C (no) 1982-08-11
FI763391A (no) 1977-06-06
CA1084051A (en) 1980-08-19
IL50849A0 (en) 1977-01-31
DK546776A (da) 1977-06-06
FI64359B (fi) 1983-07-29
JPS5271485A (en) 1977-06-14
NO146095B (no) 1982-04-19
FR2333511B1 (no) 1979-03-02
CH626073A5 (no) 1981-10-30
AU1947276A (en) 1978-05-18

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Legal Events

Date Code Title Description
RE Patent lapsed

Owner name: CARLO ERBA S.P.A.

Effective date: 19851130