BE771330A - - Google Patents

Info

Publication number
BE771330A
BE771330A BE771330A BE771330A BE771330A BE 771330 A BE771330 A BE 771330A BE 771330 A BE771330 A BE 771330A BE 771330 A BE771330 A BE 771330A BE 771330 A BE771330 A BE 771330A
Authority
BE
Belgium
Application number
BE771330A
Original Assignee
Thomae Gmbh Dr K
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from DE2040510A external-priority patent/DE2040510C3/de
Priority claimed from DE19712127267 external-priority patent/DE2127267A1/de
Application filed by Thomae Gmbh Dr K filed Critical Thomae Gmbh Dr K
Publication of BE771330A publication Critical patent/BE771330A/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D513/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
BE771330A 1970-08-14 1971-08-13 BE771330A (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE2040510A DE2040510C3 (de) 1970-08-14 1970-08-14 Oxazole- und Thiazole eckige Klammer auf 5,4-d] azepin- Derivate
DE19712127267 DE2127267A1 (en) 1971-06-02 1971-06-02 2-amino-4,5,7,8-tetrahydro-6h-thiazolo-or oxazolo(5,4-d) - azepines - as hypotensive, antiphlogistic, sedative and bechic agents

Publications (1)

Publication Number Publication Date
BE771330A true BE771330A (ru) 1972-02-14

Family

ID=25759588

Family Applications (1)

Application Number Title Priority Date Filing Date
BE771330A BE771330A (ru) 1970-08-14 1971-08-13

Country Status (23)

Country Link
US (1) US3804849A (ru)
JP (1) JPS5246236B1 (ru)
AT (1) AT310174B (ru)
AU (1) AU462319B2 (ru)
BE (1) BE771330A (ru)
BG (3) BG17785A3 (ru)
CA (1) CA965423A (ru)
CH (1) CH571003A5 (ru)
CS (1) CS178084B2 (ru)
DK (1) DK136654C (ru)
ES (3) ES393881A1 (ru)
FI (1) FI54925C (ru)
FR (1) FR2102192B1 (ru)
GB (1) GB1321509A (ru)
HU (1) HU162343B (ru)
IE (1) IE35517B1 (ru)
IL (1) IL37492A (ru)
NL (1) NL168516C (ru)
NO (1) NO131887C (ru)
PL (1) PL85080B1 (ru)
RO (4) RO59127A (ru)
SE (1) SE380529B (ru)
YU (5) YU35027B (ru)

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2820808A1 (de) * 1978-05-12 1979-11-22 Thomae Gmbh Dr K Arzneimittel mit einer antanginoesen wirksamkeit
EP0192098A2 (de) 1985-02-06 1986-08-27 Boehringer Ingelheim Kg Verwendung des 2-Amino-6-allyl-5,6,7,8-tetrahydro-4H-thiazolo[4,5-d]azepins zur Herstellung eines zur Behandlung der Parkinsonschen Erkrankung bzw. des Parkinsonismus geeigneten Arzneimittels

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3907996A (en) * 1970-08-14 1975-09-23 Boehringer Sohn Ingelheim Pharmaceutical composition containing a 2-amino-4,5,7,8-tetrahydro-6H-thiazolo or -oxazolo 5,4-D azepine and method of use
BE795257A (fr) * 1972-02-10 1973-08-09 Thomae Gmbh Dr K Nouveaux oxazols
US4400378A (en) * 1981-11-02 1983-08-23 Karl Thomae Gesellschaft Mit Beschrankter Haftung Pharmaceutical composition for the treatment of glaucoma
US4826686A (en) * 1985-12-14 1989-05-02 Boehringer Ingelheim Kg Therapeutic system
DE3820775A1 (de) * 1988-06-20 1989-12-21 Thomae Gmbh Dr K Neue 4,5,7,8-tetrahydro-6h-thiazolo(5,4,-d)azepine, ihre herstellung und ihre verwendung als arzneimittel
JP3054738B2 (ja) * 1988-07-22 2000-06-19 武田薬品工業株式会社 チアゾロ[5,4―b]アゼピン誘導体
US5424431A (en) * 1990-10-24 1995-06-13 Yamanouchi Pharmaceutical Co., Ltd. Thiazole derivatives
US6369222B1 (en) * 2000-07-18 2002-04-09 Hoffmann-La Roche Inc. mGluR antagonists and a method for their synthesis
WO2007065767A1 (en) * 2005-12-08 2007-06-14 Huntsman International Llc Process for preparing diaminodiphenylmethanes
EP2236511A4 (en) 2007-12-21 2011-04-13 Alla Chem Llc LIGANDS OF ALPHA ADRENOCEPTORS AND OF DOPAMINE, HISTAMIN, IMIDAZOLIN AND SEROTONIN RECEPTORS AND THEIR APPLICATION THEREOF
RU2374245C1 (ru) 2008-08-22 2009-11-27 Андрей Александрович Иващенко Лиганд с широким спектром одновременной рецепторной активности, фармацевтическая композиция, способ ее получения и лекарственное средство
EP2327704A4 (en) * 2008-08-29 2012-05-09 Shionogi & Co RING-CONDENSED AZOL DERIVATIVE WITH PI3K-INHIBITING EFFECT
TWI537274B (zh) 2011-03-14 2016-06-11 橘生藥品工業股份有限公司 新穎之八氫噻吩并喹啉衍生物、含有其之醫藥組成物及該等之用途
EP2930175A4 (en) 2012-12-10 2016-12-21 Kissei Pharmaceutical NOVEL OCTAHYDROPYRIDOQUINAZOLINE DERIVATIVE, PHARMACEUTICAL COMPOSITION CONTAINING THE SAME, AND USES THEREFOR, AND THE DERIVATIVE THEREOF
CN104031072A (zh) * 2014-06-24 2014-09-10 重庆植恩药业有限公司 一种盐酸他利克索的制备方法

Cited By (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2820808A1 (de) * 1978-05-12 1979-11-22 Thomae Gmbh Dr K Arzneimittel mit einer antanginoesen wirksamkeit
EP0005732A1 (de) * 1978-05-12 1979-12-12 Dr. Karl Thomae GmbH Verwendung von 2-Amino-oxazolo- oder 2-Amino-thiazolo-[5,4-d]azepinen sowie deren Säureadditionssalzen zur Herstellung eines Arzneimittels für die Verwendung bei der Bekämpfung von Angina Pectoris
EP0192098A2 (de) 1985-02-06 1986-08-27 Boehringer Ingelheim Kg Verwendung des 2-Amino-6-allyl-5,6,7,8-tetrahydro-4H-thiazolo[4,5-d]azepins zur Herstellung eines zur Behandlung der Parkinsonschen Erkrankung bzw. des Parkinsonismus geeigneten Arzneimittels

Also Published As

Publication number Publication date
RO59127A (ru) 1976-02-15
NL168516C (nl) 1982-04-16
IE35517B1 (en) 1976-03-03
YU35027B (en) 1980-06-30
RO59129A (ru) 1976-01-15
NO131887B (ru) 1975-05-12
PL85080B1 (ru) 1976-04-30
JPS5246236B1 (ru) 1977-11-22
FR2102192A1 (ru) 1972-04-07
YU42168B (en) 1988-06-30
YU35028B (en) 1980-06-30
CS178084B2 (ru) 1977-08-31
CH571003A5 (ru) 1975-12-31
YU288178A (en) 1979-12-31
NL7111176A (ru) 1972-02-16
BG17786A3 (ru) 1973-12-25
RO59925A (ru) 1976-08-15
IE35517L (en) 1972-02-14
ES396454A1 (es) 1974-05-16
FI54925B (fi) 1978-12-29
NL168516B (nl) 1981-11-16
YU208471A (en) 1979-12-31
YU35029B (en) 1980-06-30
NO131887C (ru) 1975-08-20
FI54925C (fi) 1979-04-10
DK136654B (da) 1977-11-07
YU40542B (en) 1986-02-28
HU162343B (ru) 1973-01-29
US3804849A (en) 1974-04-16
DK136654C (da) 1978-04-10
BG17785A3 (ru) 1973-12-25
AU3241171A (en) 1973-02-22
BG17968A3 (ru) 1974-03-05
AT310174B (de) 1973-09-25
YU288378A (en) 1979-12-31
RO60635A (ru) 1976-10-15
YU288278A (en) 1982-06-30
IL37492A0 (en) 1971-11-29
SE380529B (sv) 1975-11-10
YU288478A (en) 1982-06-30
ES393881A1 (es) 1973-09-16
AU462319B2 (en) 1975-06-19
CA965423A (en) 1975-04-01
IL37492A (en) 1974-03-14
FR2102192B1 (ru) 1974-11-15
GB1321509A (en) 1973-06-27
ES396453A1 (es) 1974-05-16

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