BE754606A - Nouvelles 2-aminoalcoylamino-thieno(3,2-d)pyrimidines et leurs procedesde fabrication - Google Patents

Nouvelles 2-aminoalcoylamino-thieno(3,2-d)pyrimidines et leurs procedesde fabrication

Info

Publication number
BE754606A
BE754606A BE754606DA BE754606A BE 754606 A BE754606 A BE 754606A BE 754606D A BE754606D A BE 754606DA BE 754606 A BE754606 A BE 754606A
Authority
BE
Belgium
Prior art keywords
aminoalcoylamino
thieno
pyrimidines
new
manufacturing processes
Prior art date
Application number
Other languages
English (en)
French (fr)
Original Assignee
Thomae Gmbh Dr K
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Publication date
Priority claimed from DE19691940572 external-priority patent/DE1940572A1/de
Priority claimed from DE19702032687 external-priority patent/DE2032687A1/de
Priority claimed from DE19702032686 external-priority patent/DE2032686A1/de
Publication of BE754606A publication Critical patent/BE754606A/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D495/00Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04Ortho-condensed systems
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Slide Fasteners (AREA)
BE754606D 1969-08-08 Nouvelles 2-aminoalcoylamino-thieno(3,2-d)pyrimidines et leurs procedesde fabrication BE754606A (fr)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
DE19691940572 DE1940572A1 (de) 1969-08-08 1969-08-08 Neue 2-Aminoalkylamino-thieno[3,2-d]pyrimidine und Verfahren zu ihrer Herstellung
DE19702032687 DE2032687A1 (en) 1970-07-02 1970-07-02 Cardiovascular 2-aminoalkylamino-thienopyrimidines - and 4-morpholino derivatives from 4-diethanolamino-compounds by intramolecular cyclisa
DE19702032686 DE2032686A1 (de) 1970-07-02 1970-07-02 Verfahren zur Herstellung von neuen 2 Aminoalkylamino thieno eckige Klammer auf 3,2 d eckige Klammer zu Pynmidinen

Publications (1)

Publication Number Publication Date
BE754606A true BE754606A (fr) 1971-02-08

Family

ID=27182086

Family Applications (1)

Application Number Title Priority Date Filing Date
BE754606D BE754606A (fr) 1969-08-08 Nouvelles 2-aminoalcoylamino-thieno(3,2-d)pyrimidines et leurs procedesde fabrication

Country Status (14)

Country Link
US (1) US3838121A (cs)
JP (1) JPS519759B1 (cs)
BE (1) BE754606A (cs)
BG (1) BG17591A3 (cs)
CH (5) CH547299A (cs)
ES (5) ES382548A1 (cs)
FI (1) FI51939C (cs)
FR (1) FR2068478B1 (cs)
IE (1) IE34687B1 (cs)
IL (1) IL35078A (cs)
NL (1) NL7011592A (cs)
NO (1) NO130538C (cs)
PH (1) PH9574A (cs)
SE (1) SE386449B (cs)

Families Citing this family (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6187777B1 (en) 1998-02-06 2001-02-13 Amgen Inc. Compounds and methods which modulate feeding behavior and related diseases
WO2004087707A1 (en) * 2003-03-31 2004-10-14 Vernalis (Cambridge) Limited Pyrazolopyrimidine compounds and their use in medicine
GB0423653D0 (en) * 2004-10-25 2004-11-24 Piramed Ltd Pharmaceutical compounds
CN101163706A (zh) * 2005-04-21 2008-04-16 贝林格尔·英格海姆国际有限公司 用于治疗炎性疾病的二氢噻吩并嘧啶
EP1847543A1 (de) 2006-04-19 2007-10-24 Boehringer Ingelheim Pharma GmbH & Co. KG Dihydrothienopyrimidine zur Behandlung von entzündlichen Erkrankungen
AR060632A1 (es) 2006-04-26 2008-07-02 Genentech Inc Compuestos inhibidores de fosfoinositida 3- quinasa y metodos de uso
ATE532788T1 (de) * 2006-04-26 2011-11-15 Hoffmann La Roche Pharmazeutische verbindungen
KR101533461B1 (ko) 2006-04-26 2015-07-02 에프. 호프만-라 로슈 아게 Pi3k저해제로 유용한 티에노[3,2-d]피리미딘 유도체
CN101675053B (zh) * 2006-12-07 2014-03-12 健泰科生物技术公司 磷酸肌醇3-激酶抑制剂化合物及使用方法
PE20081679A1 (es) * 2006-12-07 2008-12-18 Hoffmann La Roche Compuestos del inhibidor de fosfoinositida 3-cinasa y metodos de uso
KR20100075930A (ko) * 2007-10-19 2010-07-05 베링거 인겔하임 인터내셔날 게엠베하 헤테로사이클-치환된 피페라지노-디하이드로티에노피리미딘
EP2215093B1 (de) 2007-10-19 2011-12-14 Boehringer Ingelheim International GmbH Neue piperazino-dihydrothienopyrimidin-derivate
RS52271B (en) * 2007-10-19 2012-10-31 Boehringer Ingelheim International Gmbh SUBSTITUISANI PIPERIDINO-DIHIDROTIENOPIRIMIDIN
GB0721095D0 (en) * 2007-10-26 2007-12-05 Piramed Ltd Pharmaceutical compounds
BRPI1009022A2 (pt) * 2009-05-27 2016-03-08 Hoffmann La Roche "composto, composição farmacêutica, processo para produzir uma composição farmacêutica, uso de um composto, método para tratamento de uma doença ou transtorno e kit"
US8158625B2 (en) * 2009-05-27 2012-04-17 Genentech, Inc. Bicyclic indole-pyrimidine PI3K inhibitor compounds selective for P110 delta, and methods of use
MA33974B1 (fr) * 2009-10-12 2013-02-01 Hoffmann La Roche Combinaisons d'un inhibiteur de pi3k et d'un inhibiteur de mek
US20130059866A1 (en) 2011-08-24 2013-03-07 Boehringer Ingelheim International Gmbh Novel piperidino-dihydrothienopyrimidine sulfoxides and their use for treating copd and asthma
US9802954B2 (en) 2011-08-24 2017-10-31 Boehringer Ingelheim International Gmbh Piperidino-dihydrothienopyrimidine sulfoxides and their use for treating COPD and asthma

Also Published As

Publication number Publication date
IE34687B1 (en) 1975-07-23
ES382551A1 (es) 1973-04-01
NL7011592A (cs) 1971-02-10
JPS519759B1 (cs) 1976-03-30
IL35078A (en) 1974-09-10
NO130538B (cs) 1974-09-23
US3838121A (en) 1974-09-24
CH547299A (de) 1974-03-29
SE386449B (sv) 1976-08-09
IL35078A0 (en) 1970-10-30
NO130538C (cs) 1975-01-08
FI51939B (cs) 1977-01-31
BG17591A3 (bg) 1973-11-10
FR2068478A1 (cs) 1971-08-27
CH547301A (de) 1974-03-29
ES382552A1 (es) 1973-04-16
ES382549A1 (es) 1973-04-01
IE34687L (en) 1971-02-08
FR2068478B1 (cs) 1974-08-30
CH547300A (de) 1974-03-29
CH547304A (de) 1974-03-29
PH9574A (en) 1976-01-16
ES382548A1 (es) 1973-04-01
ES382550A1 (es) 1973-04-16
CH546251A (de) 1974-02-28
FI51939C (fi) 1977-05-10

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