BE1001464A3 - NOVEL PROCESS FOR THE PREPARATION OF PHARMACOLOGICALLY ACTIVE PIPERAZINE DERIVATIVES, DERIVATIVES AND NEW INTERMEDIATES OBTAINED. - Google Patents
NOVEL PROCESS FOR THE PREPARATION OF PHARMACOLOGICALLY ACTIVE PIPERAZINE DERIVATIVES, DERIVATIVES AND NEW INTERMEDIATES OBTAINED. Download PDFInfo
- Publication number
- BE1001464A3 BE1001464A3 BE8800218A BE8800218A BE1001464A3 BE 1001464 A3 BE1001464 A3 BE 1001464A3 BE 8800218 A BE8800218 A BE 8800218A BE 8800218 A BE8800218 A BE 8800218A BE 1001464 A3 BE1001464 A3 BE 1001464A3
- Authority
- BE
- Belgium
- Prior art keywords
- derivatives
- preparation
- pharmacologically active
- novel process
- new intermediates
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
Abstract
Nouveau procédé pour la préparation de dérivés des pipérazines. Ces dérivés correspondent à la formule générale ci-après. Utilistion : en tant que médicaments.New process for the preparation of piperazine derivatives. These derivatives correspond to the general formula below. Use: as medicine.
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
HU71887A HU198477B (en) | 1987-02-25 | 1987-02-25 | Process for producing pyrimidinyl piperazine derivatives |
HU71787A HU198204B (en) | 1987-02-25 | 1987-02-25 | Process for production of derivatives of piperasine |
HU71687A HU197313B (en) | 1987-02-25 | 1987-02-25 | Process for producing 8-azaspiro <4.5> decane-7,9-dione-8-propine-/2/ |
Publications (1)
Publication Number | Publication Date |
---|---|
BE1001464A3 true BE1001464A3 (en) | 1989-11-07 |
Family
ID=27269942
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BE8800218A BE1001464A3 (en) | 1987-02-25 | 1988-02-25 | NOVEL PROCESS FOR THE PREPARATION OF PHARMACOLOGICALLY ACTIVE PIPERAZINE DERIVATIVES, DERIVATIVES AND NEW INTERMEDIATES OBTAINED. |
Country Status (20)
Country | Link |
---|---|
KR (1) | KR880009955A (en) |
CN (1) | CN88100923A (en) |
AT (1) | AT395851B (en) |
BE (1) | BE1001464A3 (en) |
CA (1) | CA1300141C (en) |
CH (1) | CH677924A5 (en) |
CS (1) | CS274423B2 (en) |
DE (1) | DE3806009C2 (en) |
DK (1) | DK99388A (en) |
ES (1) | ES2009236A6 (en) |
FI (1) | FI880895A (en) |
FR (1) | FR2615853B1 (en) |
GB (1) | GB2201417B (en) |
GR (1) | GR1002245B (en) |
IL (1) | IL85545A (en) |
IT (1) | IT1217342B (en) |
NL (1) | NL8800484A (en) |
PL (1) | PL152958B1 (en) |
SE (1) | SE8800651L (en) |
YU (1) | YU46441B (en) |
Families Citing this family (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
HU217129B (en) * | 1993-07-16 | 1999-11-29 | EGIS Gyógyszergyár Rt. | Process for the preparation of buspiron as therapeutical active ingredient of high purity |
KR950014099A (en) * | 1993-11-10 | 1995-06-15 | 장기하 | Method for preparing N- (2-pyrimidyl) piperazinyl butylamide |
Citations (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3354178A (en) * | 1965-04-09 | 1967-11-21 | Sterling Drug Inc | Nu-(4-amino-2-butynyl)-nu-alkylcarboxamides |
US3444171A (en) * | 1964-07-03 | 1969-05-13 | Astra Apotekarnes Kem Fab | Acetylenic imides and method for their preparation |
FR2073406A1 (en) * | 1969-11-24 | 1971-10-01 | Bristol Myers Co |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE1545543B1 (en) * | 1964-07-03 | 1970-01-22 | Astra Apotekarnes Kem Fab | 4-aminobutinylimides, their salts and processes for their preparation |
JPS6310786A (en) * | 1986-07-01 | 1988-01-18 | Sumitomo Pharmaceut Co Ltd | Novel imide derivative and production thereof |
JPS6310760A (en) * | 1986-07-01 | 1988-01-18 | Sumitomo Pharmaceut Co Ltd | Novel production of imide derivative |
-
1988
- 1988-02-23 CH CH675/88A patent/CH677924A5/de not_active IP Right Cessation
- 1988-02-23 PL PL1988270815A patent/PL152958B1/en unknown
- 1988-02-24 CN CN198888100923A patent/CN88100923A/en active Pending
- 1988-02-25 ES ES8800543A patent/ES2009236A6/en not_active Expired
- 1988-02-25 DK DK099388A patent/DK99388A/en not_active Application Discontinuation
- 1988-02-25 AT AT0047688A patent/AT395851B/en not_active IP Right Cessation
- 1988-02-25 NL NL8800484A patent/NL8800484A/en not_active Application Discontinuation
- 1988-02-25 CS CS122288A patent/CS274423B2/en unknown
- 1988-02-25 YU YU36288A patent/YU46441B/en unknown
- 1988-02-25 BE BE8800218A patent/BE1001464A3/en not_active IP Right Cessation
- 1988-02-25 FR FR888802286A patent/FR2615853B1/en not_active Expired - Lifetime
- 1988-02-25 SE SE8800651A patent/SE8800651L/en not_active Application Discontinuation
- 1988-02-25 DE DE3806009A patent/DE3806009C2/en not_active Expired - Fee Related
- 1988-02-25 GB GB8804385A patent/GB2201417B/en not_active Expired - Lifetime
- 1988-02-25 GR GR880100108A patent/GR1002245B/en unknown
- 1988-02-25 FI FI880895A patent/FI880895A/en not_active Application Discontinuation
- 1988-02-25 IL IL85545A patent/IL85545A/en not_active IP Right Cessation
- 1988-02-25 CA CA000559846A patent/CA1300141C/en not_active Expired - Lifetime
- 1988-02-25 KR KR1019880001939A patent/KR880009955A/en not_active Application Discontinuation
- 1988-02-25 IT IT19545/88A patent/IT1217342B/en active
Patent Citations (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3444171A (en) * | 1964-07-03 | 1969-05-13 | Astra Apotekarnes Kem Fab | Acetylenic imides and method for their preparation |
US3354178A (en) * | 1965-04-09 | 1967-11-21 | Sterling Drug Inc | Nu-(4-amino-2-butynyl)-nu-alkylcarboxamides |
FR2073406A1 (en) * | 1969-11-24 | 1971-10-01 | Bristol Myers Co |
Also Published As
Publication number | Publication date |
---|---|
YU36288A (en) | 1989-10-31 |
SE8800651L (en) | 1988-08-26 |
DK99388D0 (en) | 1988-02-25 |
IL85545A (en) | 1992-05-25 |
FR2615853A1 (en) | 1988-12-02 |
GB8804385D0 (en) | 1988-03-23 |
NL8800484A (en) | 1988-09-16 |
DK99388A (en) | 1988-08-26 |
GB2201417B (en) | 1990-10-31 |
SE8800651D0 (en) | 1988-02-25 |
YU46441B (en) | 1993-10-20 |
IT8819545A0 (en) | 1988-02-25 |
CH677924A5 (en) | 1991-07-15 |
PL152958B1 (en) | 1991-02-28 |
FI880895A0 (en) | 1988-02-25 |
GR880100108A (en) | 1988-12-16 |
GR1002245B (en) | 1996-04-22 |
CA1300141C (en) | 1992-05-05 |
GB2201417A (en) | 1988-09-01 |
CS122288A2 (en) | 1990-08-14 |
ATA47688A (en) | 1992-08-15 |
FR2615853B1 (en) | 1991-01-04 |
ES2009236A6 (en) | 1989-09-16 |
CN88100923A (en) | 1988-09-28 |
DE3806009A1 (en) | 1988-09-08 |
PL270815A1 (en) | 1989-04-03 |
FI880895A (en) | 1988-08-26 |
CS274423B2 (en) | 1991-04-11 |
KR880009955A (en) | 1988-10-06 |
IL85545A0 (en) | 1988-08-31 |
AT395851B (en) | 1993-03-25 |
IT1217342B (en) | 1990-03-22 |
DE3806009C2 (en) | 1996-09-12 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
FR2391210A1 (en) | QUINOLEINECARBOXYLIC ACID DERIVATIVES AND THEIR USE AS ANTIBACTERIAL AGENTS | |
FR2430412A1 (en) | SUBSTITUTED PROPANOLAMINE DERIVATIVES USEFUL AS MEDICAMENTS AND PROCESS FOR THEIR PREPARATION | |
FR2378023A1 (en) | PROCESS FOR THE PREPARATION OF OXIMES, NEW PRODUCTS THUS OBTAINED AND THEIR APPLICATION IN THE SYNTHESIS OF COMPOUNDS OF 3,7-DISUBSTITUTED CEPHEMCARBOXYLIC ACID | |
FR2426681A1 (en) | HYDANTOINE DERIVATIVES, PROCESS FOR THEIR PREPARATION AND APPLICATION OF THESE COMPOUNDS AS MEDICINAL PRODUCTS | |
FR2383907A1 (en) | PROCESS FOR PREPARING DERIVATIVES OF ACETIC ACID AND DERIVATIVES OBTAINED BY THIS PROCESS | |
FR2428052A1 (en) | NOVEL 5-FLUORO- (B-URIDINE OR 2'-DESOXY-B-URIDINE) DERIVATIVES, PROCESS FOR PREPARING THEM AND CARCINOSTATIC AGENTS CONTAINING THEM | |
FR2435479A1 (en) | PROCESS FOR THE PREPARATION OF 3-CEPHEM-4-CARBOXYLIC ACID COMPOUNDS 3, 7-DISUBSTITUTED AND THEIR PHARMACEUTICALLY ACCEPTABLE SALTS, NOVEL PRODUCTS THUS OBTAINED AND THEIR USE FOR THEIR ANTIMICROBIAL ACTIVITIES | |
FR2363559A1 (en) | NEW DERIVATIVES OF PERHYDRO-AZA-HETEROCYCLES USEFUL AS MEDICINAL PRODUCTS AND PROCESS FOR THEIR PREPARATION | |
FR2403330A1 (en) | NEW DERIVATIVES OF BENZOYL-2-CHLORO-4-GLYCINANILIDES SUBSTITUTES, THEIR METHOD OF PREPARATION AND THEIR APPLICATION AS MEDICINAL PRODUCTS | |
FR2386544A1 (en) | PROCESS FOR THE PREPARATION OF DERIVATIVES OF IMIDAZODIAZEPINE | |
FR2388802A1 (en) | PROCESS FOR THE PRODUCTION OF UREA DERIVATIVES AND NEW PRODUCTS THUS OBTAINED | |
FR2381776A1 (en) | PROCESS FOR THE PREPARATION OF OXAZOLINOAZETIDINYLBUTYRIC ACID DERIVATIVES AND NEW PRODUCTS THUS OBTAINED | |
FR2395272A1 (en) | NEW MEDICINES DERIVED FROM AMIDINOPENICILLANIC ACID | |
FR2370020A2 (en) | PROCESS FOR PREPARING ALKYLPHENOLS | |
FR2384775A1 (en) | MORPHINE DERIVATIVES, THEIR METHOD OF PREPARATION AND THEIR APPLICATION AS A MEDICINAL PRODUCT | |
FR2399998A1 (en) | PRODUCT DERIVED FROM DIPHENOXY-1,3 PROPANONE-2, PROCESS FOR ITS PREPARATION AND ITS APPLICATION TO THE REALIZATION OF A MEDICINAL PRODUCT | |
FR2364913A1 (en) | NEW BENZOPYRANE DERIVATIVES USEFUL AS MEDICINAL PRODUCTS AND THEIR PROCESS FOR PREPARATION | |
BE1001464A3 (en) | NOVEL PROCESS FOR THE PREPARATION OF PHARMACOLOGICALLY ACTIVE PIPERAZINE DERIVATIVES, DERIVATIVES AND NEW INTERMEDIATES OBTAINED. | |
FR2404010A1 (en) | NEW DERIVATIVES OF PYRIMIDO- (2,1-A) ISOQUINOLEINE, THEIR PRODUCTION PROCESS AND PHARMACEUTICAL COMPOSITION CONTAINING THEM | |
FR2362841A1 (en) | ACYL HETEROCYCLYL-CARBOXYLIC ACID DERIVATIVES USEFUL AS MEDICINAL PRODUCTS AND PROCESS FOR THEIR PREPARATION | |
FR2432015A1 (en) | COMPOUNDS DERIVED FROM CYCLOHEXYLCARBOXYLIC ACID AND PROCESS FOR THEIR PREPARATION | |
BE904864A (en) | QUINOLEIN DERIVATIVES, THEIR PREPARATION PROCESS AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM. | |
FR2401160A1 (en) | NEW VINCAMINOL ESTERS, THEIR PREPARATION AND THEIR APPLICATION AS MEDICINAL PRODUCTS | |
FR2387983A1 (en) | NEW BENZODIAZEPINE DERIVATIVES USEFUL AS MEDICINAL PRODUCTS | |
FR2391218A1 (en) | AZACYCLYL COMPOUNDS AND PROCESS FOR THEIR PREPARATION AND APPLICATION AS A MEDICINAL PRODUCT |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
RE | Patent lapsed |
Owner name: EGIS GYOGYSZERGYAR Effective date: 19980228 |