AU662077B2 - Androst-4-eno(4,5-b)pyrrole derivatives and process for their preparation - Google Patents

Androst-4-eno(4,5-b)pyrrole derivatives and process for their preparation Download PDF

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Publication number
AU662077B2
AU662077B2 AU47072/93A AU4707293A AU662077B2 AU 662077 B2 AU662077 B2 AU 662077B2 AU 47072/93 A AU47072/93 A AU 47072/93A AU 4707293 A AU4707293 A AU 4707293A AU 662077 B2 AU662077 B2 AU 662077B2
Authority
AU
Australia
Prior art keywords
formula
compound
document
androsta
international
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
AU47072/93A
Other languages
English (en)
Other versions
AU4707293A (en
Inventor
Franco Buzzetti
Enrico Di Salle
Antonio Longo
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pfizer Italia SRL
Original Assignee
Farmitalia Carlo Erba SRL
Carlo Erba SpA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Farmitalia Carlo Erba SRL, Carlo Erba SpA filed Critical Farmitalia Carlo Erba SRL
Publication of AU4707293A publication Critical patent/AU4707293A/en
Application granted granted Critical
Publication of AU662077B2 publication Critical patent/AU662077B2/en
Anticipated expiration legal-status Critical
Ceased legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J71/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton is condensed with a heterocyclic ring
    • C07J71/0036—Nitrogen-containing hetero ring
    • C07J71/0042—Nitrogen only
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J7/00—Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of two carbon atoms
    • C07J7/008—Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of two carbon atoms substituted in position 21
    • C07J7/0085—Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of two carbon atoms substituted in position 21 by an halogen atom

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Steroid Compounds (AREA)
  • Pyrrole Compounds (AREA)
  • Fats And Perfumes (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
AU47072/93A 1992-08-11 1993-08-05 Androst-4-eno(4,5-b)pyrrole derivatives and process for their preparation Ceased AU662077B2 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GB929217035A GB9217035D0 (en) 1992-08-11 1992-08-11 Androst-4-eno(4,5-b)pyrrole derivatives and process for their preparation
GB9217035 1992-08-11
PCT/EP1993/002080 WO1994004554A1 (en) 1992-08-11 1993-08-05 ANDROST-4-ENO[4,5-b]PYRROLE DERIVATIVES AND PROCESS FOR THEIR PREPARATION

Publications (2)

Publication Number Publication Date
AU4707293A AU4707293A (en) 1994-03-15
AU662077B2 true AU662077B2 (en) 1995-08-17

Family

ID=10720180

Family Applications (1)

Application Number Title Priority Date Filing Date
AU47072/93A Ceased AU662077B2 (en) 1992-08-11 1993-08-05 Androst-4-eno(4,5-b)pyrrole derivatives and process for their preparation

Country Status (21)

Country Link
US (1) US5457097A (enExample)
EP (1) EP0608404B1 (enExample)
JP (1) JPH07500119A (enExample)
CN (1) CN1086220A (enExample)
AT (1) ATE136036T1 (enExample)
AU (1) AU662077B2 (enExample)
CA (1) CA2120726A1 (enExample)
DE (1) DE69302007T2 (enExample)
DK (1) DK0608404T3 (enExample)
ES (1) ES2088289T3 (enExample)
FI (1) FI941635A7 (enExample)
GB (1) GB9217035D0 (enExample)
GR (1) GR3019729T3 (enExample)
HU (1) HUT67662A (enExample)
IL (1) IL106597A (enExample)
MX (1) MX9304852A (enExample)
MY (1) MY108957A (enExample)
NZ (1) NZ254805A (enExample)
TW (1) TW276257B (enExample)
WO (1) WO1994004554A1 (enExample)
ZA (1) ZA935769B (enExample)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5510340A (en) * 1992-06-12 1996-04-23 Sri International Antihypercholesterolemic compounds and related pharmaceutical compositions and methods of use
CA2794565C (en) 2010-04-08 2018-08-21 Emory University Substituted androst-4-ene diones

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3032551A (en) * 1961-05-25 1962-05-01 Syntex Sa Pyrrolo(3', 2'-2, 3)-androstanes and process therefor
US3282928A (en) * 1964-04-23 1966-11-01 American Cyanamid Co 1, 11-iminoestratetraenes
GB8503940D0 (en) * 1985-02-15 1985-03-20 Erba Farmitalia 4-substituted androstendione derivatives
GB8617107D0 (en) * 1986-07-14 1986-08-20 Erba Farmitalia 6-/7-methylenandrosta-1 4-diene-3 17-dione derivatives
GB8622330D0 (en) * 1986-09-17 1986-10-22 Erba Farmitalia 4-substituted 6-alkylidenandrostene-3,17-dione derivatives
GB8721384D0 (en) * 1987-09-11 1987-10-21 Erba Farmitalia 17-substituted andro-sta-1 4-dien-3-one derivatives

Also Published As

Publication number Publication date
IL106597A0 (en) 1993-12-08
JPH07500119A (ja) 1995-01-05
FI941635A0 (fi) 1994-04-08
US5457097A (en) 1995-10-10
ES2088289T3 (es) 1996-08-01
DE69302007D1 (de) 1996-05-02
GR3019729T3 (en) 1996-07-31
DE69302007T2 (de) 1996-08-29
GB9217035D0 (en) 1992-09-23
EP0608404A1 (en) 1994-08-03
EP0608404B1 (en) 1996-03-27
CA2120726A1 (en) 1994-03-03
HU9401003D0 (en) 1994-07-28
MY108957A (en) 1996-11-30
AU4707293A (en) 1994-03-15
CN1086220A (zh) 1994-05-04
HUT67662A (en) 1995-04-28
DK0608404T3 (da) 1996-04-29
NZ254805A (en) 1995-11-27
FI941635A7 (fi) 1994-04-08
MX9304852A (es) 1994-02-28
TW276257B (enExample) 1996-05-21
ZA935769B (en) 1994-03-08
WO1994004554A1 (en) 1994-03-03
ATE136036T1 (de) 1996-04-15
IL106597A (en) 1997-09-30

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