AU605522B2 - Carboxamido ethyl-imidazole and-1,2,4-triazole derivatives - Google Patents

Carboxamido ethyl-imidazole and-1,2,4-triazole derivatives Download PDF

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Publication number
AU605522B2
AU605522B2 AU81962/87A AU8196287A AU605522B2 AU 605522 B2 AU605522 B2 AU 605522B2 AU 81962/87 A AU81962/87 A AU 81962/87A AU 8196287 A AU8196287 A AU 8196287A AU 605522 B2 AU605522 B2 AU 605522B2
Authority
AU
Australia
Prior art keywords
halogen
substituted
compound
cyano
heteroaryl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
AU81962/87A
Other languages
English (en)
Other versions
AU8196287A (en
Inventor
Helmut Egger
Rudolf Walchli
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Sandoz AG
Original Assignee
Sandoz AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sandoz AG filed Critical Sandoz AG
Publication of AU8196287A publication Critical patent/AU8196287A/en
Application granted granted Critical
Publication of AU605522B2 publication Critical patent/AU605522B2/en
Anticipated expiration legal-status Critical
Ceased legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/56—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Endocrinology (AREA)
  • Reproductive Health (AREA)
  • Urology & Nephrology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
AU81962/87A 1986-12-03 1987-12-01 Carboxamido ethyl-imidazole and-1,2,4-triazole derivatives Ceased AU605522B2 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE3641320 1986-12-03
DE3641320 1986-12-03

Publications (2)

Publication Number Publication Date
AU8196287A AU8196287A (en) 1988-06-16
AU605522B2 true AU605522B2 (en) 1991-01-17

Family

ID=6315380

Family Applications (1)

Application Number Title Priority Date Filing Date
AU81962/87A Ceased AU605522B2 (en) 1986-12-03 1987-12-01 Carboxamido ethyl-imidazole and-1,2,4-triazole derivatives

Country Status (24)

Country Link
JP (1) JPH0678318B2 (uk)
KR (1) KR880007481A (uk)
AT (1) AT395587B (uk)
AU (1) AU605522B2 (uk)
BE (1) BE1001235A4 (uk)
CH (1) CH677925A5 (uk)
DK (1) DK631287A (uk)
ES (1) ES2010235A6 (uk)
FI (1) FI875300A (uk)
FR (1) FR2607810B1 (uk)
GB (1) GB2199579B (uk)
GR (1) GR871897B (uk)
HU (1) HU198694B (uk)
IL (1) IL84665A (uk)
IT (1) IT1211944B (uk)
LU (1) LU87063A1 (uk)
MY (1) MY103004A (uk)
NL (1) NL8702897A (uk)
NZ (1) NZ222765A (uk)
PH (1) PH24666A (uk)
PL (1) PL151588B1 (uk)
PT (1) PT86255B (uk)
SE (1) SE8704792L (uk)
ZA (1) ZA879093B (uk)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8814277D0 (en) * 1988-06-16 1988-07-20 Glaxo Group Ltd Chemical compounds
HU220863B1 (en) * 1991-09-02 2002-06-29 Yamanouchi Pharma Co Ltd Triazolylated tertiary amines, process for producing them and pharmaceutical compositions containing them
GB9409882D0 (en) * 1994-05-18 1994-07-06 Sandoz Ltd Organic compounds
GB0128415D0 (en) * 2001-11-27 2002-01-16 Univ Sheffield Medicaments

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AT382868B (de) * 1983-03-11 1987-04-27 Sandoz Ag Verfahren zur herstellung neuer azolderivate und deren salze
JPH0625144B2 (ja) * 1986-02-24 1994-04-06 四国化成工業株式会社 新規イミダゾール化合物及び該化合物の合成方法

Also Published As

Publication number Publication date
GB2199579A (en) 1988-07-13
DK631287D0 (da) 1987-12-01
AT395587B (de) 1993-01-25
IT1211944B (it) 1989-11-08
LU87063A1 (fr) 1988-07-14
GR871897B (en) 1988-04-04
HUT45506A (en) 1988-07-28
FI875300A0 (fi) 1987-12-01
FR2607810B1 (fr) 1989-12-01
JPH0678318B2 (ja) 1994-10-05
FR2607810A1 (fr) 1988-06-10
AU8196287A (en) 1988-06-16
IT8748656A0 (it) 1987-12-01
SE8704792D0 (sv) 1987-12-01
BE1001235A4 (fr) 1989-08-29
KR880007481A (ko) 1988-08-27
PH24666A (en) 1990-09-07
ATA316887A (de) 1992-06-15
IL84665A0 (en) 1988-05-31
GB2199579B (en) 1990-07-18
NZ222765A (en) 1990-11-27
PL151588B1 (en) 1990-09-28
MY103004A (en) 1993-03-31
ZA879093B (en) 1989-07-26
SE8704792L (sv) 1988-06-04
HU198694B (en) 1989-11-28
DK631287A (da) 1988-06-04
ES2010235A6 (es) 1989-11-01
JPS63145270A (ja) 1988-06-17
CH677925A5 (uk) 1991-07-15
IL84665A (en) 1991-11-21
NL8702897A (nl) 1988-07-01
FI875300A (fi) 1988-06-04
GB8727978D0 (en) 1988-01-06
PT86255B (pt) 1990-11-07
PL269180A1 (en) 1988-08-18
PT86255A (en) 1988-06-01

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