MY103004A - Azole derivatives - Google Patents

Azole derivatives

Info

Publication number
MY103004A
MY103004A MYPI87003136A MYPI19873136A MY103004A MY 103004 A MY103004 A MY 103004A MY PI87003136 A MYPI87003136 A MY PI87003136A MY PI19873136 A MYPI19873136 A MY PI19873136A MY 103004 A MY103004 A MY 103004A
Authority
MY
Malaysia
Prior art keywords
heteroaryl
aryl
substituted
cycloalkyl
mono
Prior art date
Application number
MYPI87003136A
Inventor
Helmut Egger Dr
Rudolf Walchli Dr
Original Assignee
Sandoz Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sandoz Ltd filed Critical Sandoz Ltd
Publication of MY103004A publication Critical patent/MY103004A/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D231/00Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/02Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D233/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/56Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D249/00Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/081,2,4-Triazoles; Hydrogenated 1,2,4-triazoles

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Endocrinology (AREA)
  • Reproductive Health (AREA)
  • Urology & Nephrology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)

Abstract

COMPOUNDS OF FORMULA I (FORMULA. 1)WHEREIN R1 AND R2 ARE THE SAME OR DIFFERENT AND EACH REPRESENT UNSUBSTITUTED OR MONO- OR POLY-SUBSTITUTED ARYL OR HETEROARYL, R3 REPRESENTS UNSUBSTITUTED OR MONO- OR POLY-SUBSTITUTED ALKYL, CYCLOALKYL, ARYL, OR HETEROARYL; OR CYCLOALKYL, ARYL OR HETEROARYL CONDENSED WITH A BENZENE RING; OR ALKOXY, AND X REPRESENTS CH OR N, WHEREBY WHEN R3 REPRESENTS METHYL AND R1 AND R2 REPRESENT PHENYL AT LEAST ONE OF SAID PHENYLS MUST BE SUBSTITUTED, IN FREE FORM OR IN ACID ADDITION SALT FORM. THE COMPOUNDS ARE INDICATED FOR USE AS PHARMACEUTICALS IN PARTICULAR AS AROMATASE INHIBITORS.
MYPI87003136A 1986-12-03 1987-12-01 Azole derivatives MY103004A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE3641320 1986-12-03

Publications (1)

Publication Number Publication Date
MY103004A true MY103004A (en) 1993-03-31

Family

ID=6315380

Family Applications (1)

Application Number Title Priority Date Filing Date
MYPI87003136A MY103004A (en) 1986-12-03 1987-12-01 Azole derivatives

Country Status (24)

Country Link
JP (1) JPH0678318B2 (en)
KR (1) KR880007481A (en)
AT (1) AT395587B (en)
AU (1) AU605522B2 (en)
BE (1) BE1001235A4 (en)
CH (1) CH677925A5 (en)
DK (1) DK631287A (en)
ES (1) ES2010235A6 (en)
FI (1) FI875300A (en)
FR (1) FR2607810B1 (en)
GB (1) GB2199579B (en)
GR (1) GR871897B (en)
HU (1) HU198694B (en)
IL (1) IL84665A (en)
IT (1) IT1211944B (en)
LU (1) LU87063A1 (en)
MY (1) MY103004A (en)
NL (1) NL8702897A (en)
NZ (1) NZ222765A (en)
PH (1) PH24666A (en)
PL (1) PL151588B1 (en)
PT (1) PT86255B (en)
SE (1) SE8704792L (en)
ZA (1) ZA879093B (en)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8814277D0 (en) * 1988-06-16 1988-07-20 Glaxo Group Ltd Chemical compounds
UA41295C2 (en) * 1991-09-02 2001-09-17 Яманугі Фармасетікл Ко., Лтд Triazol-substituted tertiary amine compounds or salts thereof as inhibitor of aromatase and a pharmaceutical composition based thereon
GB9409882D0 (en) * 1994-05-18 1994-07-06 Sandoz Ltd Organic compounds
GB0128415D0 (en) * 2001-11-27 2002-01-16 Univ Sheffield Medicaments

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AT382868B (en) * 1983-03-11 1987-04-27 Sandoz Ag Process for the preparation of novel azole derivatives and salts thereof
JPH0625144B2 (en) * 1986-02-24 1994-04-06 四国化成工業株式会社 Novel imidazole compound and method for synthesizing the compound

Also Published As

Publication number Publication date
LU87063A1 (en) 1988-07-14
AU8196287A (en) 1988-06-16
AU605522B2 (en) 1991-01-17
FR2607810B1 (en) 1989-12-01
SE8704792L (en) 1988-06-04
IL84665A (en) 1991-11-21
FI875300A0 (en) 1987-12-01
JPS63145270A (en) 1988-06-17
IT8748656A0 (en) 1987-12-01
PL151588B1 (en) 1990-09-28
NL8702897A (en) 1988-07-01
ES2010235A6 (en) 1989-11-01
GB8727978D0 (en) 1988-01-06
DK631287A (en) 1988-06-04
IT1211944B (en) 1989-11-08
JPH0678318B2 (en) 1994-10-05
ATA316887A (en) 1992-06-15
AT395587B (en) 1993-01-25
BE1001235A4 (en) 1989-08-29
GB2199579A (en) 1988-07-13
KR880007481A (en) 1988-08-27
PT86255A (en) 1988-06-01
NZ222765A (en) 1990-11-27
FR2607810A1 (en) 1988-06-10
ZA879093B (en) 1989-07-26
PT86255B (en) 1990-11-07
PL269180A1 (en) 1988-08-18
GR871897B (en) 1988-04-04
PH24666A (en) 1990-09-07
HUT45506A (en) 1988-07-28
FI875300A (en) 1988-06-04
DK631287D0 (en) 1987-12-01
IL84665A0 (en) 1988-05-31
CH677925A5 (en) 1991-07-15
GB2199579B (en) 1990-07-18
SE8704792D0 (en) 1987-12-01
HU198694B (en) 1989-11-28

Similar Documents

Publication Publication Date Title
AU536175B2 (en) (piperidinylalky) quinazoline derivatives
EG19678A (en) Derivatives of propenoic acid useful as fungicides
ZA86596B (en) Derivatives of imidazole,their preparation and utilisation,and pharmaceutical compositions containing these derivates
EP0275482A3 (en) Novel prolinal derivatives
MY103004A (en) Azole derivatives
ATE281462T1 (en) 4-CYKLOHEXYL-1,3,2-OXAZABOROLIDINE AS CHIRAL AGENTS
DK0413278T3 (en) Use of xanthine derivatives against peptic ulcer
WO2000071785A3 (en) 2-cylcoalkylcarbonylcyclohexane-1,3-dione derivatives as herbicides
GB1481158A (en) Derivatives of 1,2,4-oxadiazolidine-3-one and pesticidal compositions containing them
NO952937L (en) Newly substituted thiosemicarbazone derivatives
MY103558A (en) Fungicides
EP0132278A4 (en) Pyran derivatives.
MX9504262A (en) Novel process for preparation of clonidine derivatives.
JPS6463569A (en) Heteroaryl derivative