SE8704792L - azole derivatives - Google Patents
azole derivativesInfo
- Publication number
- SE8704792L SE8704792L SE8704792A SE8704792A SE8704792L SE 8704792 L SE8704792 L SE 8704792L SE 8704792 A SE8704792 A SE 8704792A SE 8704792 A SE8704792 A SE 8704792A SE 8704792 L SE8704792 L SE 8704792L
- Authority
- SE
- Sweden
- Prior art keywords
- heteroaryl
- aryl
- substituted
- cycloalkyl
- mono
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/56—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
- C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
- C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Endocrinology (AREA)
- Reproductive Health (AREA)
- Urology & Nephrology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Abstract
Compounds of formula <IMAGE> [wherein R1 and R2 are the same or different and each represent unsubstituted or mono- or poly-substituted aryl or heteroaryl; R3 represents unsubstituted or mono- or poly-substituted alkyl, cycloalkyl, aryl, or heteroaryl; or cycloalkyl, aryl or heteroaryl condensed with a benzene ring; or alkoxy; and X represents CH or N; whereby when R3 represents methyl and R1 and R2 represent phenyl at least one of said phenyls must be substituted,] in free form or in acid addition salt form are indicated for use as pharmaceuticals in particular as aromatase inhibitors.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE3641320 | 1986-12-03 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| SE8704792D0 SE8704792D0 (en) | 1987-12-01 |
| SE8704792L true SE8704792L (en) | 1988-06-04 |
Family
ID=6315380
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| SE8704792A SE8704792L (en) | 1986-12-03 | 1987-12-01 | azole derivatives |
Country Status (24)
| Country | Link |
|---|---|
| JP (1) | JPH0678318B2 (en) |
| KR (1) | KR880007481A (en) |
| AT (1) | AT395587B (en) |
| AU (1) | AU605522B2 (en) |
| BE (1) | BE1001235A4 (en) |
| CH (1) | CH677925A5 (en) |
| DK (1) | DK631287A (en) |
| ES (1) | ES2010235A6 (en) |
| FI (1) | FI875300A (en) |
| FR (1) | FR2607810B1 (en) |
| GB (1) | GB2199579B (en) |
| GR (1) | GR871897B (en) |
| HU (1) | HU198694B (en) |
| IL (1) | IL84665A (en) |
| IT (1) | IT1211944B (en) |
| LU (1) | LU87063A1 (en) |
| MY (1) | MY103004A (en) |
| NL (1) | NL8702897A (en) |
| NZ (1) | NZ222765A (en) |
| PH (1) | PH24666A (en) |
| PL (1) | PL151588B1 (en) |
| PT (1) | PT86255B (en) |
| SE (1) | SE8704792L (en) |
| ZA (1) | ZA879093B (en) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB8814277D0 (en) * | 1988-06-16 | 1988-07-20 | Glaxo Group Ltd | Chemical compounds |
| US5674886A (en) * | 1991-09-02 | 1997-10-07 | Yamanouchi Pharmaceutical Co., Ltd. | Triazolylated teritiary amine compound or salt thereof |
| GB9409882D0 (en) * | 1994-05-18 | 1994-07-06 | Sandoz Ltd | Organic compounds |
| GB0128415D0 (en) * | 2001-11-27 | 2002-01-16 | Univ Sheffield | Medicaments |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AT382868B (en) * | 1983-03-11 | 1987-04-27 | Sandoz Ag | Process for the preparation of novel azole derivatives and salts thereof |
| JPH0625144B2 (en) * | 1986-02-24 | 1994-04-06 | 四国化成工業株式会社 | Novel imidazole compound and method for synthesizing the compound |
-
1987
- 1987-11-26 CH CH4607/87A patent/CH677925A5/de not_active IP Right Cessation
- 1987-11-30 GB GB8727978A patent/GB2199579B/en not_active Expired - Lifetime
- 1987-12-01 NZ NZ222765A patent/NZ222765A/en unknown
- 1987-12-01 FI FI875300A patent/FI875300A/en not_active IP Right Cessation
- 1987-12-01 AU AU81962/87A patent/AU605522B2/en not_active Ceased
- 1987-12-01 IT IT8748656A patent/IT1211944B/en active
- 1987-12-01 PH PH36145A patent/PH24666A/en unknown
- 1987-12-01 IL IL84665A patent/IL84665A/en unknown
- 1987-12-01 DK DK631287A patent/DK631287A/en not_active Application Discontinuation
- 1987-12-01 SE SE8704792A patent/SE8704792L/en not_active Application Discontinuation
- 1987-12-01 MY MYPI87003136A patent/MY103004A/en unknown
- 1987-12-02 PT PT86255A patent/PT86255B/en not_active IP Right Cessation
- 1987-12-02 KR KR870013695A patent/KR880007481A/en not_active Application Discontinuation
- 1987-12-02 FR FR878716736A patent/FR2607810B1/en not_active Expired
- 1987-12-02 AT AT0316887A patent/AT395587B/en not_active IP Right Cessation
- 1987-12-02 HU HU875414A patent/HU198694B/en unknown
- 1987-12-02 NL NL8702897A patent/NL8702897A/en not_active Application Discontinuation
- 1987-12-02 JP JP62305522A patent/JPH0678318B2/en not_active Expired - Lifetime
- 1987-12-02 BE BE8701375A patent/BE1001235A4/en not_active IP Right Cessation
- 1987-12-02 PL PL1987269180A patent/PL151588B1/en unknown
- 1987-12-03 ZA ZA879093A patent/ZA879093B/en unknown
- 1987-12-03 LU LU87063A patent/LU87063A1/en unknown
- 1987-12-03 ES ES8703470A patent/ES2010235A6/en not_active Expired
- 1987-12-14 GR GR871897A patent/GR871897B/en unknown
Also Published As
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| FI800047A (en) | NYA (PIPERIDINYL ALKYL) QUINAZOLE DERIVATIVES | |
| DE69028136D1 (en) | Alkoxyiminoacetamide derivatives and their use as antifungal agents | |
| NL350013I2 (en) | Antifungal. | |
| BR9709126A (en) | Ethylene derivatives and pesticides containing said derivatives | |
| NO983970L (en) | Tricyclic compounds, their preparation and use | |
| ES506115A0 (en) | PROCEDURE FOR THE OBTAINING OF B-LACTAMA COMPOUNDS. | |
| ES2061663T3 (en) | DERIVATIVES OF CARBAMOILPIRROLIDINA, ITS USE AND PREPARATION. | |
| KR860005794A (en) | Method for preparing an imidazole derivative | |
| DE3783754D1 (en) | PROLIN DERIVATIVES. | |
| SE8704792L (en) | azole derivatives | |
| ATE32894T1 (en) | THIOMETHYLPYRIDIN DERIVATIVES, PROCESSES FOR THEIR PREPARATION AND PHARMACEUTICALS CONTAINING THESE COMPOUNDS. | |
| GB1478338A (en) | Catalytic oxidation of diarylmethane and triarylmethane compounds | |
| NO974462D0 (en) | Compound for use in the preparation of alkyl derivatives of trazodone with CNS activity | |
| CA2158763A1 (en) | Novel process for preparation of clonidine derivatives | |
| WO2000071785A3 (en) | 2-cylcoalkylcarbonylcyclohexane-1,3-dione derivatives as herbicides | |
| SE7901250L (en) | NEW PROCEDURE FOR PREPARATION OF THIAZOLE DERIVATIVES | |
| TH14140EX (en) | Alkylsubstitutated Nitrotoluene derivatives | |
| GB1094045A (en) | Phthalazine derivatives |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| NAV | Patent application has lapsed |
Ref document number: 8704792-4 Effective date: 19940701 Format of ref document f/p: F |