AU6020890A - New esters of organic acids with alcohol derivatives of 19-nor steroids and their salts, their preparation process and the intermediates of this process, their use as medicaments and the compositions containing them - Google Patents
New esters of organic acids with alcohol derivatives of 19-nor steroids and their salts, their preparation process and the intermediates of this process, their use as medicaments and the compositions containing themInfo
- Publication number
- AU6020890A AU6020890A AU60208/90A AU6020890A AU6020890A AU 6020890 A AU6020890 A AU 6020890A AU 60208/90 A AU60208/90 A AU 60208/90A AU 6020890 A AU6020890 A AU 6020890A AU 6020890 A AU6020890 A AU 6020890A
- Authority
- AU
- Australia
- Prior art keywords
- denotes
- radical
- alkyl
- hydrogen atom
- optionally
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
- C07J41/0033—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005
- C07J41/0077—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005 substituted in position 11-beta by a carbon atom, further substituted by a group comprising at least one further carbon atom
- C07J41/0083—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005 substituted in position 11-beta by a carbon atom, further substituted by a group comprising at least one further carbon atom substituted in position 11-beta by an optionally substituted phenyl group not further condensed with other rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
- C07J1/0051—Estrane derivatives
- C07J1/0081—Substituted in position 17 alfa and 17 beta
- C07J1/0088—Substituted in position 17 alfa and 17 beta the substituent in position 17 alfa being an unsaturated hydrocarbon group
- C07J1/0096—Alkynyl derivatives
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J31/00—Normal steroids containing one or more sulfur atoms not belonging to a hetero ring
- C07J31/006—Normal steroids containing one or more sulfur atoms not belonging to a hetero ring not covered by C07J31/003
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Diabetes (AREA)
- Endocrinology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Steroid Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Abstract
Products of general formula (I): <IMAGE> in which R1 denotes an aliphatic hydrocarbon radical, R2 and R3, which are identical or different, denote a hydrogen atom or an alkyl radical, G denotes a hydrocarbon group containing from one to eighteen carbon atoms and optionally one or a number of identical or different heteroatoms, which is linked to the steroid nucleus by a carbon atom, and either X denotes XA, XA being a hydrogen atom, an alkyl radical, an arylalkyl radical or an acyl radical, and in this case Y denotes YA, YA being a group -B-O-CO-A-Z in which B denotes a saturated or unsaturated, linear or branched, divalent aliphatic radical, A denotes either a saturated or unsaturated, linear or branched, divalent aliphatic radical optionally interrupted or terminated by a divalent aromatic radical, or A denotes a divalent aromatic radical and Z denotes one of the functional groups -COOH or -SO3H, it being possible for these functional groups to be optionally converted into salt form or X denotes XB, XB being a group -CO-A-Z in which A and Z are as defined above and Y then denotes YB, YB being one of the groups chosen from -C IDENTICAL C-R4, -CH=CH-R4 or -CH2-CH2-R4, in which R4 denotes a hydrogen atom, a halogen atom, a trialkylsilyl radical, an alkyl radical or a phenyl radical, the said alkyl and phenyl radicals being optionally substituted.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR8910648A FR2650748B1 (en) | 1989-08-08 | 1989-08-08 | NOVEL ESTERS OF ORGANIC ACIDS WITH ALCOHOLS DERIVED FROM 19-NOR STEROIDS AND THEIR SALTS, THEIR PREPARATION METHOD AND THE INTERMEDIATES THEREOF, THEIR APPLICATION AS MEDICAMENTS AND THE COMPOSITIONS CONTAINING THEM |
| FR8910648 | 1989-08-08 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| AU6020890A true AU6020890A (en) | 1991-02-14 |
| AU633604B2 AU633604B2 (en) | 1993-02-04 |
Family
ID=9384560
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AU60208/90A Ceased AU633604B2 (en) | 1989-08-08 | 1990-08-07 | New esters of organic acids with alcohol derivatives of 19-nor steroids and their salts, their preparation process and the intermediates of this process, their use as medicaments and the compositions containing them |
Country Status (27)
| Country | Link |
|---|---|
| EP (1) | EP0412907B1 (en) |
| JP (1) | JP3056770B2 (en) |
| KR (1) | KR910004648A (en) |
| CN (1) | CN1036521C (en) |
| AT (1) | ATE113958T1 (en) |
| AU (1) | AU633604B2 (en) |
| CA (1) | CA2022647A1 (en) |
| DE (1) | DE69014012T2 (en) |
| DK (1) | DK0412907T3 (en) |
| EG (1) | EG19423A (en) |
| ES (1) | ES2063940T3 (en) |
| FI (1) | FI903905A0 (en) |
| FR (1) | FR2650748B1 (en) |
| HU (1) | HUT55031A (en) |
| IE (1) | IE65905B1 (en) |
| IL (1) | IL95272A (en) |
| MA (1) | MA21925A1 (en) |
| MX (1) | MX21771A (en) |
| NO (1) | NO177595C (en) |
| NZ (1) | NZ234824A (en) |
| OA (1) | OA09303A (en) |
| PT (1) | PT94935B (en) |
| RU (1) | RU2056431C1 (en) |
| TN (1) | TNSN90112A1 (en) |
| TW (1) | TW201313B (en) |
| YU (1) | YU47865B (en) |
| ZA (1) | ZA905812B (en) |
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO1996022387A1 (en) * | 1995-01-16 | 1996-07-25 | Garvan Institute Of Medical Research | Diagnostic method using estrogen receptor gene polymorphisms |
Families Citing this family (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2659233B1 (en) * | 1990-03-06 | 1994-01-21 | Roussel Uclaf | NEW USE OF ANTI-PROGESTOMIMETIC COMPOUNDS IN FARMING ANIMALS. |
| DE4434488A1 (en) * | 1994-09-14 | 1996-03-21 | Schering Ag | Steroid esters and amides, processes for their preparation and their pharmaceutical use |
| US6090798A (en) * | 1997-12-19 | 2000-07-18 | Alcon Laboratories, Inc. | Treatment of GLC1A glaucoma with glucocorticoid antagonists |
| DE19915871A1 (en) | 1998-04-09 | 1999-10-21 | Unisia Jecs Corp | Viscous fluid coupling, for driving auxiliary units such as cooling fans |
| JP2000130165A (en) | 1998-10-30 | 2000-05-09 | Unisia Jecs Corp | Fan coupling device |
| JP2001012511A (en) | 1999-06-25 | 2001-01-16 | Unisia Jecs Corp | Fluid coupling |
| CN110099688A (en) * | 2016-11-17 | 2019-08-06 | 赛途公司 | Bone myohypertrophia inducer |
| KR102518275B1 (en) * | 2022-07-27 | 2023-04-05 | 주식회사 화성케미칼 | Method of recycled neoprene fabric |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE3347126A1 (en) * | 1983-12-22 | 1985-07-11 | Schering AG, 1000 Berlin und 4709 Bergkamen | 11SS-ARYL-ESTRADIENE, THEIR PRODUCTION AND THE PHARMACEUTICAL PREPARATIONS CONTAINING THEM |
| DE3506785A1 (en) * | 1985-02-22 | 1986-08-28 | Schering AG, Berlin und Bergkamen, 1000 Berlin | 11SS-N, N-DIMETHYLAMINOPHENYL ESTRADIENE, THE PRODUCTION THEREOF AND PHARMACEUTICAL PREPARATIONS CONTAINING THEM |
| IE60780B1 (en) * | 1987-01-23 | 1994-08-10 | Akzo Nv | New 11-aryl steroid derivatives |
| DE3878198T2 (en) * | 1987-12-12 | 1993-06-24 | Akzo Nv | 11-ARYLSTEROID DERIVATIVES. |
| FR2643638B1 (en) * | 1989-02-24 | 1991-06-14 | Roussel Uclaf | NOVEL 19-NOR STEROIDS HAVING IN THE 11BETA POSITION A CARBON CHAIN COMPRISING AN AMIDE OR CARBAMATE FUNCTION, THEIR PREPARATION METHOD AND INTERMEDIATES THEREOF, THEIR APPLICATION AS MEDICAMENTS AND THE PHARMACEUTICAL COMPOSITIONS CONTAINING THEM |
-
1989
- 1989-08-08 FR FR8910648A patent/FR2650748B1/en not_active Expired - Fee Related
-
1990
- 1990-07-24 ZA ZA905812A patent/ZA905812B/en unknown
- 1990-07-30 MX MX2177190A patent/MX21771A/en unknown
- 1990-08-02 IL IL9527290A patent/IL95272A/en not_active IP Right Cessation
- 1990-08-02 MA MA22195A patent/MA21925A1/en unknown
- 1990-08-03 YU YU151390A patent/YU47865B/en unknown
- 1990-08-03 CA CA002022647A patent/CA2022647A1/en not_active Abandoned
- 1990-08-04 EG EG46190A patent/EG19423A/en active
- 1990-08-06 JP JP2206949A patent/JP3056770B2/en not_active Expired - Lifetime
- 1990-08-07 FI FI903905A patent/FI903905A0/en not_active Application Discontinuation
- 1990-08-07 PT PT94935A patent/PT94935B/en not_active IP Right Cessation
- 1990-08-07 HU HU904921A patent/HUT55031A/en unknown
- 1990-08-07 IE IE283990A patent/IE65905B1/en not_active IP Right Cessation
- 1990-08-07 NO NO903475A patent/NO177595C/en unknown
- 1990-08-07 AU AU60208/90A patent/AU633604B2/en not_active Ceased
- 1990-08-07 KR KR1019900012166A patent/KR910004648A/en active IP Right Grant
- 1990-08-08 OA OA59835A patent/OA09303A/en unknown
- 1990-08-08 ES ES90402266T patent/ES2063940T3/en not_active Expired - Lifetime
- 1990-08-08 DE DE69014012T patent/DE69014012T2/en not_active Expired - Lifetime
- 1990-08-08 CN CN90106741A patent/CN1036521C/en not_active Expired - Fee Related
- 1990-08-08 TN TNTNSN90112A patent/TNSN90112A1/en unknown
- 1990-08-08 DK DK90402266.2T patent/DK0412907T3/en active
- 1990-08-08 AT AT90402266T patent/ATE113958T1/en not_active IP Right Cessation
- 1990-08-08 EP EP90402266A patent/EP0412907B1/en not_active Expired - Lifetime
- 1990-08-08 NZ NZ234824A patent/NZ234824A/en unknown
- 1990-08-23 TW TW079107064A patent/TW201313B/zh active
-
1992
- 1992-07-07 RU SU925011906A patent/RU2056431C1/en active
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO1996022387A1 (en) * | 1995-01-16 | 1996-07-25 | Garvan Institute Of Medical Research | Diagnostic method using estrogen receptor gene polymorphisms |
Also Published As
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| MK14 | Patent ceased section 143(a) (annual fees not paid) or expired |