AU530456B2 - Thio-substituted benzoylpropionyl-l-prolines - Google Patents
Thio-substituted benzoylpropionyl-l-prolinesInfo
- Publication number
- AU530456B2 AU530456B2 AU49351/79A AU4935179A AU530456B2 AU 530456 B2 AU530456 B2 AU 530456B2 AU 49351/79 A AU49351/79 A AU 49351/79A AU 4935179 A AU4935179 A AU 4935179A AU 530456 B2 AU530456 B2 AU 530456B2
- Authority
- AU
- Australia
- Prior art keywords
- proline
- formula
- hydrogen
- aryl
- carbon atoms
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Ceased
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D207/46—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with hetero atoms directly attached to the ring nitrogen atom
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C327/00—Thiocarboxylic acids
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C59/00—Compounds having carboxyl groups bound to acyclic carbon atoms and containing any of the groups OH, O—metal, —CHO, keto, ether, groups, groups, or groups
- C07C59/40—Unsaturated compounds
- C07C59/76—Unsaturated compounds containing keto groups
- C07C59/84—Unsaturated compounds containing keto groups containing six membered aromatic rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C59/00—Compounds having carboxyl groups bound to acyclic carbon atoms and containing any of the groups OH, O—metal, —CHO, keto, ether, groups, groups, or groups
- C07C59/40—Unsaturated compounds
- C07C59/76—Unsaturated compounds containing keto groups
- C07C59/88—Unsaturated compounds containing keto groups containing halogen
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D207/10—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D207/16—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Pyrrole Compounds (AREA)
- Peptides Or Proteins (AREA)
Applications Claiming Priority (4)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US93956478A | 1978-09-05 | 1978-09-05 | |
| US939564 | 1978-09-05 | ||
| US06/044,733 US4226775A (en) | 1979-06-01 | 1979-06-01 | Substituted thio-substituted benzyl-propionyl-L-prolines |
| US44733 | 1979-06-01 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| AU4935179A AU4935179A (en) | 1980-03-13 |
| AU530456B2 true AU530456B2 (en) | 1983-07-14 |
Family
ID=26721935
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AU49351/79A Ceased AU530456B2 (en) | 1978-09-05 | 1979-07-30 | Thio-substituted benzoylpropionyl-l-prolines |
Country Status (19)
| Country | Link |
|---|---|
| EP (1) | EP0010347B1 (enExample) |
| AR (2) | AR230624A1 (enExample) |
| AU (1) | AU530456B2 (enExample) |
| CA (1) | CA1114821A (enExample) |
| DD (1) | DD147236A5 (enExample) |
| DE (1) | DE2934592A1 (enExample) |
| DK (1) | DK161198C (enExample) |
| ES (1) | ES483846A1 (enExample) |
| FI (1) | FI75152C (enExample) |
| GR (1) | GR73190B (enExample) |
| HU (1) | HU180651B (enExample) |
| IE (1) | IE48939B1 (enExample) |
| IL (1) | IL57802A (enExample) |
| NO (1) | NO155240C (enExample) |
| NZ (1) | NZ190995A (enExample) |
| PH (1) | PH19468A (enExample) |
| PT (1) | PT70025A (enExample) |
| YU (1) | YU205479A (enExample) |
| ZA (1) | ZA793536B (enExample) |
Families Citing this family (13)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4303583A (en) | 1979-08-13 | 1981-12-01 | American Home Products Corporation | 1H,5H-[1,4]Thiazepino[4,3-a]indole-1,5-diones |
| IE51409B1 (en) * | 1980-07-24 | 1986-12-24 | Ici Ltd | Amide derivatives |
| DE3169110D1 (en) * | 1980-11-24 | 1985-03-28 | Ici Plc | Amide derivatives |
| US4438031A (en) | 1982-02-24 | 1984-03-20 | American Home Products Corporation | N-(Alkylsulfonyl)-L-proline amide and N-(alkylsulfonyl)-2-carboxylic acid amide-indoline derivatives |
| JPH0623190B2 (ja) * | 1985-04-16 | 1994-03-30 | サントリー株式会社 | インヒビタ−活性を有するｎ−アシルピロリジン誘導体及びその製法並びに用途 |
| US4880827A (en) * | 1986-03-18 | 1989-11-14 | Sumitomo Pharmaceuticals Company, Ltd. | Pyrrolidine derivatives having inhibitory action for proline specific endopepidase |
| HU198012B (en) * | 1987-07-03 | 1989-07-28 | Richter Gedeon Vegyeszet | Process for producing cyclic amino-acid derivatives and pharmaceutical compositions containing them |
| CA2113288A1 (en) * | 1993-01-29 | 1994-07-30 | Kan Takamine | Process for producing aromatic amide compounds |
| DE4302957A1 (de) * | 1993-02-03 | 1994-08-04 | Bayer Ag | Imidazolyl-substituierte Phenylessigsäureprolinamide |
| JPH09501920A (ja) * | 1993-08-19 | 1997-02-25 | ワーナー−ランバート・コンパニー | 非ペプチドエンドセリンアンタゴニスト▲ｉ▼ |
| US5922759A (en) * | 1996-06-21 | 1999-07-13 | Warner-Lambert Company | Butenolide endothelin antagonists |
| AU6603996A (en) * | 1995-08-24 | 1997-03-19 | Warner-Lambert Company | Furanone endothelin antagonists |
| US5891892A (en) * | 1996-10-29 | 1999-04-06 | Warner-Lambert Company | Small molecule biaryl compounds as inhibitors of endothelin converting enzyme |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AU509899B2 (en) * | 1976-02-13 | 1980-05-29 | E.R. Squibb & Sons, Inc. | Proline derivatives and related compounds |
| US4052511A (en) * | 1976-02-13 | 1977-10-04 | E. R. Squibb & Sons, Inc. | Carboxyacylproline derivatives |
| US4116962A (en) * | 1976-12-03 | 1978-09-26 | E. R. Squibb & Sons, Inc. | Pyrrolidine and piperidine-2-carboxylic acid derivatives |
-
1978
- 1978-07-12 NZ NZ190995A patent/NZ190995A/xx unknown
-
1979
- 1979-06-25 CA CA332,486A patent/CA1114821A/en not_active Expired
- 1979-07-13 ZA ZA00793536A patent/ZA793536B/xx unknown
- 1979-07-13 IL IL57802A patent/IL57802A/xx not_active IP Right Cessation
- 1979-07-18 GR GR59636A patent/GR73190B/el unknown
- 1979-07-30 AU AU49351/79A patent/AU530456B2/en not_active Ceased
- 1979-08-02 AR AR277577A patent/AR230624A1/es active
- 1979-08-03 PT PT70025A patent/PT70025A/pt unknown
- 1979-08-21 EP EP79301712A patent/EP0010347B1/en not_active Expired
- 1979-08-21 FI FI792595A patent/FI75152C/fi not_active IP Right Cessation
- 1979-08-21 YU YU02054/79A patent/YU205479A/xx unknown
- 1979-08-27 DE DE19792934592 patent/DE2934592A1/de active Granted
- 1979-08-31 PH PH22988A patent/PH19468A/en unknown
- 1979-09-03 ES ES483846A patent/ES483846A1/es not_active Expired
- 1979-09-04 IE IE1682/79A patent/IE48939B1/en not_active IP Right Cessation
- 1979-09-04 HU HU79AE580A patent/HU180651B/hu not_active IP Right Cessation
- 1979-09-04 DK DK369079A patent/DK161198C/da not_active IP Right Cessation
- 1979-09-04 NO NO792849A patent/NO155240C/no unknown
- 1979-09-05 DD DD79215364A patent/DD147236A5/de unknown
-
1981
- 1981-02-04 AR AR284203A patent/AR229953A1/es active
Also Published As
| Publication number | Publication date |
|---|---|
| YU205479A (en) | 1983-01-21 |
| IL57802A0 (en) | 1979-11-30 |
| AR229953A1 (es) | 1984-01-31 |
| IL57802A (en) | 1983-05-15 |
| DD147236A5 (de) | 1981-03-25 |
| FI75152B (fi) | 1988-01-29 |
| EP0010347A1 (en) | 1980-04-30 |
| IE791682L (en) | 1980-03-05 |
| AU4935179A (en) | 1980-03-13 |
| CA1114821A (en) | 1981-12-22 |
| IE48939B1 (en) | 1985-06-26 |
| HU180651B (en) | 1983-04-29 |
| DK369079A (da) | 1980-03-06 |
| DE2934592C2 (enExample) | 1989-10-05 |
| FI75152C (fi) | 1988-05-09 |
| DE2934592A1 (de) | 1980-03-20 |
| NO792849L (no) | 1980-03-06 |
| ZA793536B (en) | 1980-07-30 |
| DK161198B (da) | 1991-06-10 |
| GR73190B (enExample) | 1984-02-14 |
| DK161198C (da) | 1991-12-02 |
| NO155240C (no) | 1987-03-04 |
| FI792595A7 (fi) | 1980-03-06 |
| NZ190995A (en) | 1982-03-09 |
| PT70025A (en) | 1979-09-01 |
| EP0010347B1 (en) | 1983-11-09 |
| ES483846A1 (es) | 1980-04-16 |
| NO155240B (no) | 1986-11-24 |
| AR230624A1 (es) | 1984-05-31 |
| PH19468A (en) | 1986-05-14 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| AU520788B2 (en) | Cycloalkyltriazoles | |
| AU518718B2 (en) | 9-amino-dibenzopyrans | |
| AU4782679A (en) | Oxygenerator | |
| AU4569779A (en) | 4-aza-17-substituted-5a-androstan-3-ones | |
| AU1328683A (en) | O-alkoxycarbonyl benzenesulfonylisocyanates | |
| AU5035479A (en) | 2-nitroimidazoles | |
| AU4876779A (en) | Oxybenzylidiene-bornanones | |
| AU4655479A (en) | Ear-plugs | |
| AU4825779A (en) | Benzofuranyl-piperidines | |
| AU5009279A (en) | Spiro-oxazolidindiones | |
| AU4406379A (en) | 1-aryloxy-3-hitratoalkylamino-2-propanols | |
| AU4506179A (en) | Nitrodiarylamines | |
| AU4530579A (en) | Plansifters | |
| AU4754479A (en) | Carbamimido thiaotes | |
| AU4642179A (en) | 4-quinolinylaminobenzoylpiperidines | |
| AU5064479A (en) | 3-unsubstituted-3-cephems | |
| AU4935179A (en) | Thio-substituted benzoylpropionyl-l-prolines | |
| AU4571479A (en) | 2-aminopyrimidones | |
| AU4946279A (en) | Imidazoquinoxalines | |
| AU4830279A (en) | Indolealylamines | |
| AU4814679A (en) | Rid-mowse | |
| AU4398479A (en) | N-azolylalkyl-halogenoacetanilides | |
| AU5169879A (en) | Episcope | |
| AU4507279A (en) | Phenoxyalkylamines | |
| AU4519079A (en) | Dilignols |