AU2254692A - Methods and compositions for treating emesis, nausea and other disorders using optically pure s(-) ondansetron - Google Patents
Methods and compositions for treating emesis, nausea and other disorders using optically pure s(-) ondansetronInfo
- Publication number
- AU2254692A AU2254692A AU22546/92A AU2254692A AU2254692A AU 2254692 A AU2254692 A AU 2254692A AU 22546/92 A AU22546/92 A AU 22546/92A AU 2254692 A AU2254692 A AU 2254692A AU 2254692 A AU2254692 A AU 2254692A
- Authority
- AU
- Australia
- Prior art keywords
- ondansetron
- administered
- composition according
- pharmaceutically acceptable
- composition
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
Links
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- 239000007921 spray Substances 0.000 description 1
- 230000000638 stimulation Effects 0.000 description 1
- 239000000126 substance Substances 0.000 description 1
- 231100000736 substance abuse Toxicity 0.000 description 1
- 235000000346 sugar Nutrition 0.000 description 1
- 150000008163 sugars Chemical class 0.000 description 1
- QAOWNCQODCNURD-UHFFFAOYSA-N sulfuric acid group Chemical class S(O)(O)(=O)=O QAOWNCQODCNURD-UHFFFAOYSA-N 0.000 description 1
- 239000004094 surface-active agent Substances 0.000 description 1
- 210000000225 synapse Anatomy 0.000 description 1
- 208000011580 syndromic disease Diseases 0.000 description 1
- 235000002906 tartaric acid Nutrition 0.000 description 1
- 239000011975 tartaric acid Substances 0.000 description 1
- 231100000462 teratogen Toxicity 0.000 description 1
- 239000003439 teratogenic agent Substances 0.000 description 1
- 229960003433 thalidomide Drugs 0.000 description 1
- 238000011287 therapeutic dose Methods 0.000 description 1
- 231100001274 therapeutic index Toxicity 0.000 description 1
- 210000001519 tissue Anatomy 0.000 description 1
- 235000019505 tobacco product Nutrition 0.000 description 1
- 229940125725 tranquilizer Drugs 0.000 description 1
- 239000003204 tranquilizing agent Substances 0.000 description 1
- 230000002936 tranquilizing effect Effects 0.000 description 1
- 230000001052 transient effect Effects 0.000 description 1
- 210000001186 vagus nerve Anatomy 0.000 description 1
- 230000000007 visual effect Effects 0.000 description 1
- 230000004580 weight loss Effects 0.000 description 1
- 208000016261 weight loss Diseases 0.000 description 1
- 229950004681 zacopride Drugs 0.000 description 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/415—1,2-Diazoles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/08—Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
Landscapes
- Health & Medical Sciences (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- Veterinary Medicine (AREA)
- General Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Otolaryngology (AREA)
- Organic Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Hospice & Palliative Care (AREA)
- Engineering & Computer Science (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (4)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US721723 | 1985-04-10 | ||
| US750801 | 1985-07-01 | ||
| US72172391A | 1991-06-26 | 1991-06-26 | |
| US75080191A | 1991-08-27 | 1991-08-27 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AU2254692A true AU2254692A (en) | 1993-01-25 |
Family
ID=27110471
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AU22546/92A Abandoned AU2254692A (en) | 1991-06-26 | 1992-06-25 | Methods and compositions for treating emesis, nausea and other disorders using optically pure s(-) ondansetron |
Country Status (5)
| Country | Link |
|---|---|
| EP (1) | EP0591395A1 (enrdf_load_stackoverflow) |
| JP (1) | JPH06509073A (enrdf_load_stackoverflow) |
| AU (1) | AU2254692A (enrdf_load_stackoverflow) |
| CA (1) | CA2112488A1 (enrdf_load_stackoverflow) |
| WO (1) | WO1993000075A1 (enrdf_load_stackoverflow) |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO1993000074A1 (en) * | 1991-06-26 | 1993-01-07 | Sepracor, Inc. | Method and compositions for treating emesis, nausea and other disorders using optically pure r(+) ondansetron |
| CN1078465C (zh) * | 1996-10-10 | 2002-01-30 | 沈阳药科大学 | 一种含奥坦西酮的透皮吸收制剂 |
| AU779696B2 (en) | 1999-03-01 | 2005-02-10 | Sepracor, Inc. | Methods for treating apnea and apnea disorders using optically pure R(+)ondansetron |
| US20030114475A1 (en) * | 2001-10-31 | 2003-06-19 | Addiction Therapies, Inc. | Methods for the treatment of addiction |
| WO2006085497A1 (ja) * | 2005-02-09 | 2006-08-17 | Kissei Pharmaceutical Co., Ltd. | 口腔内崩壊錠 |
| US20110288115A1 (en) * | 2010-05-24 | 2011-11-24 | Avmedis Llc | Treatment of vagally-mediated spectrum disorders |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4695578A (en) * | 1984-01-25 | 1987-09-22 | Glaxo Group Limited | 1,2,3,9-tetrahydro-3-imidazol-1-ylmethyl-4H-carbazol-4-ones, composition containing them, and method of using them to treat neuronal 5HT function disturbances |
| GB8516083D0 (en) * | 1985-06-25 | 1985-07-31 | Glaxo Group Ltd | Heterocyclic compounds |
| GB8518745D0 (en) * | 1985-07-24 | 1985-08-29 | Glaxo Group Ltd | Heterocyclic compounds |
| DK662687A (da) * | 1986-12-17 | 1988-06-18 | Glaxo Group Ltd | Anvendelse af tricycliske carbazoloner |
-
1992
- 1992-06-25 EP EP92914351A patent/EP0591395A1/en not_active Withdrawn
- 1992-06-25 AU AU22546/92A patent/AU2254692A/en not_active Abandoned
- 1992-06-25 JP JP5501665A patent/JPH06509073A/ja active Pending
- 1992-06-25 WO PCT/US1992/005377 patent/WO1993000075A1/en not_active Application Discontinuation
- 1992-06-25 CA CA002112488A patent/CA2112488A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| WO1993000075A1 (en) | 1993-01-07 |
| CA2112488A1 (en) | 1993-01-07 |
| JPH06509073A (ja) | 1994-10-13 |
| EP0591395A4 (enrdf_load_stackoverflow) | 1994-08-31 |
| EP0591395A1 (en) | 1994-04-13 |
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