AU2018221889A1 - Compositions for treating acne - Google Patents
Compositions for treating acne Download PDFInfo
- Publication number
- AU2018221889A1 AU2018221889A1 AU2018221889A AU2018221889A AU2018221889A1 AU 2018221889 A1 AU2018221889 A1 AU 2018221889A1 AU 2018221889 A AU2018221889 A AU 2018221889A AU 2018221889 A AU2018221889 A AU 2018221889A AU 2018221889 A1 AU2018221889 A1 AU 2018221889A1
- Authority
- AU
- Australia
- Prior art keywords
- solvent
- ethanol
- pharmaceutical composition
- ethoxyethoxy
- alcohol
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
Links
- 239000000203 mixture Substances 0.000 title claims description 75
- 206010000496 acne Diseases 0.000 title claims description 60
- 208000002874 Acne Vulgaris Diseases 0.000 title claims description 54
- XXJWXESWEXIICW-UHFFFAOYSA-N diethylene glycol monoethyl ether Chemical compound CCOCCOCCO XXJWXESWEXIICW-UHFFFAOYSA-N 0.000 claims abstract description 159
- 239000002904 solvent Substances 0.000 claims abstract description 108
- 239000012049 topical pharmaceutical composition Substances 0.000 claims abstract description 12
- 238000011282 treatment Methods 0.000 claims description 49
- 229920001451 polypropylene glycol Polymers 0.000 claims description 45
- KPUWHANPEXNPJT-UHFFFAOYSA-N disiloxane Chemical group [SiH3]O[SiH3] KPUWHANPEXNPJT-UHFFFAOYSA-N 0.000 claims description 44
- 235000019441 ethanol Nutrition 0.000 claims description 44
- LFQSCWFLJHTTHZ-UHFFFAOYSA-N Ethanol Chemical compound CCO LFQSCWFLJHTTHZ-UHFFFAOYSA-N 0.000 claims description 43
- 239000008194 pharmaceutical composition Substances 0.000 claims description 39
- 229920001223 polyethylene glycol Polymers 0.000 claims description 39
- 125000000217 alkyl group Chemical group 0.000 claims description 36
- 230000000699 topical effect Effects 0.000 claims description 36
- 239000002202 Polyethylene glycol Substances 0.000 claims description 35
- KFZMGEQAYNKOFK-UHFFFAOYSA-N Isopropanol Chemical compound CC(C)O KFZMGEQAYNKOFK-UHFFFAOYSA-N 0.000 claims description 33
- RTZKZFJDLAIYFH-UHFFFAOYSA-N Diethyl ether Chemical compound CCOCC RTZKZFJDLAIYFH-UHFFFAOYSA-N 0.000 claims description 28
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Classifications
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/075—Ethers or acetals
- A61K31/08—Ethers or acetals acyclic, e.g. paraformaldehyde
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
- A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
- A61K47/10—Alcohols; Phenols; Salts thereof, e.g. glycerol; Polyethylene glycols [PEG]; Poloxamers; PEG/POE alkyl ethers
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
- A61K47/24—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing atoms other than carbon, hydrogen, oxygen, halogen, nitrogen or sulfur, e.g. cyclomethicone or phospholipids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0014—Skin, i.e. galenical aspects of topical compositions
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/08—Solutions
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/10—Anti-acne agents
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Epidemiology (AREA)
- General Chemical & Material Sciences (AREA)
- Engineering & Computer Science (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Dermatology (AREA)
- Oil, Petroleum & Natural Gas (AREA)
- Molecular Biology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Biophysics (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Medicinal Preparation (AREA)
- Cosmetics (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201762459312P | 2017-02-15 | 2017-02-15 | |
| AU2017900498A AU2017900498A0 (en) | 2017-02-15 | Compositions for Treating Acne | |
| US62/459,312 | 2017-02-15 | ||
| AU2017900498 | 2017-02-15 | ||
| PCT/AU2018/050117 WO2018148795A1 (en) | 2017-02-15 | 2018-02-14 | Compositions for treating acne |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AU2018221889A1 true AU2018221889A1 (en) | 2019-09-05 |
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AU2018221889A Abandoned AU2018221889A1 (en) | 2017-02-15 | 2018-02-14 | Compositions for treating acne |
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| Country | Link |
|---|---|
| US (2) | US20200022927A1 (enExample) |
| EP (1) | EP3582763A4 (enExample) |
| JP (1) | JP2020508993A (enExample) |
| CN (1) | CN110430872A (enExample) |
| AU (1) | AU2018221889A1 (enExample) |
| BR (1) | BR112019017045A2 (enExample) |
| CA (1) | CA3053507A1 (enExample) |
| IL (1) | IL268715A (enExample) |
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| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA2338124C (en) * | 2001-02-26 | 2010-08-03 | Valerie Dumont Dicianna | Self-tanning composition in sheeted substrate |
| FR2867682B1 (fr) * | 2004-03-22 | 2009-06-05 | Galderma Res & Dev | Composition pharmaceutique anhydre associant un agent silicone et un principe actif solubilise. |
| WO2009090495A2 (en) * | 2007-12-07 | 2009-07-23 | Foamix Ltd. | Oil and liquid silicone foamable carriers and formulations |
| US20100261795A1 (en) * | 2009-04-08 | 2010-10-14 | Pierre Fabre Dermocosmetique Usa | Antiacneic compositions |
| JP5964322B2 (ja) * | 2011-01-13 | 2016-08-03 | キュー エル ティー インク．ＱＬＴ Ｉｎｃ． | 光増感剤の局所送達用医薬組成物及びその使用 |
| US20150141389A1 (en) * | 2012-04-27 | 2015-05-21 | Dow Corning Corporation | Topical Formulation Compositions Containing Silicone Based Excipients To Deliver Actives To A Substrate |
| CA2888060C (en) * | 2012-10-24 | 2019-02-26 | John E. Kulesza | Low toxicity topical active agent delivery system |
| WO2014081674A1 (en) * | 2012-11-20 | 2014-05-30 | Allergan, Inc. | Topical dapsone and dapsone/adapalene compositions and methods for use thereof |
| WO2014116653A1 (en) * | 2013-01-22 | 2014-07-31 | Coty Inc. | Topical formulations and methods for the use thereof |
| EP3065702B1 (en) * | 2013-10-31 | 2023-06-07 | Sun Pharmaceutical Industries Ltd | Topical pharmaceutical composition of acitretin |
-
2018
- 2018-02-14 US US16/486,323 patent/US20200022927A1/en not_active Abandoned
- 2018-02-14 CA CA3053507A patent/CA3053507A1/en active Pending
- 2018-02-14 JP JP2019544856A patent/JP2020508993A/ja active Pending
- 2018-02-14 CN CN201880019063.8A patent/CN110430872A/zh active Pending
- 2018-02-14 AU AU2018221889A patent/AU2018221889A1/en not_active Abandoned
- 2018-02-14 EP EP18754614.8A patent/EP3582763A4/en not_active Withdrawn
- 2018-02-14 BR BR112019017045A patent/BR112019017045A2/pt not_active IP Right Cessation
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2019
- 2019-08-14 IL IL26871519A patent/IL268715A/en unknown
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2022
- 2022-07-01 US US17/856,781 patent/US20220331269A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| US20220331269A1 (en) | 2022-10-20 |
| JP2020508993A (ja) | 2020-03-26 |
| EP3582763A1 (en) | 2019-12-25 |
| CA3053507A1 (en) | 2018-08-23 |
| BR112019017045A2 (pt) | 2020-04-14 |
| CN110430872A (zh) | 2019-11-08 |
| IL268715A (en) | 2019-10-31 |
| EP3582763A4 (en) | 2020-11-25 |
| US20200022927A1 (en) | 2020-01-23 |
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| Date | Code | Title | Description |
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| MK5 | Application lapsed section 142(2)(e) - patent request and compl. specification not accepted |