AU2013288319A1 - Complement pathway modulators and uses thereof - Google Patents

Complement pathway modulators and uses thereof Download PDF

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Publication number
AU2013288319A1
AU2013288319A1 AU2013288319A AU2013288319A AU2013288319A1 AU 2013288319 A1 AU2013288319 A1 AU 2013288319A1 AU 2013288319 A AU2013288319 A AU 2013288319A AU 2013288319 A AU2013288319 A AU 2013288319A AU 2013288319 A1 AU2013288319 A1 AU 2013288319A1
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Australia
Prior art keywords
alkyl
alkoxy
hydrogen
halogen
compound
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AU2013288319A
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Inventor
Ulrich Hommel
Edwige Liliane Jeanne Lorthiois
Juergen Klaus Maibaum
Nils Ostermann
Stefan Andreas Randl
Olivier Rogel
Anna Vulpetti
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Novartis AG
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Novartis AG
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    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing three or more hetero rings
    • A—HUMAN NECESSITIES
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    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/403—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
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    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/415—1,2-Diazoles
    • A61K31/4155—1,2-Diazoles non condensed and containing further heterocyclic rings
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    • C07D471/04—Ortho-condensed systems

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  • Child & Adolescent Psychology (AREA)
  • Tropical Medicine & Parasitology (AREA)
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  • Obesity (AREA)
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AU2013288319A 2012-07-12 2013-06-27 Complement pathway modulators and uses thereof Abandoned AU2013288319A1 (en)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US201261670868P 2012-07-12 2012-07-12
US61/670,868 2012-07-12
US201361774234P 2013-03-07 2013-03-07
US61/774,234 2013-03-07
PCT/IB2013/055302 WO2014009833A2 (en) 2012-07-12 2013-06-27 Complement pathway modulators and uses thereof

Publications (1)

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AU2013288319A1 true AU2013288319A1 (en) 2015-02-05

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AU2013288319A Abandoned AU2013288319A1 (en) 2012-07-12 2013-06-27 Complement pathway modulators and uses thereof

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US (1) US9550755B2 (h)
EP (1) EP2872503B1 (h)
JP (1) JP6238980B2 (h)
KR (1) KR20150036481A (h)
CN (1) CN104684910B (h)
AU (1) AU2013288319A1 (h)
BR (1) BR112015000578A2 (h)
CA (1) CA2882724A1 (h)
EA (1) EA201590200A1 (h)
ES (1) ES2687983T3 (h)
IN (1) IN2015DN00185A (h)
MX (1) MX2015000537A (h)
WO (1) WO2014009833A2 (h)

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KR20210093855A (ko) 2018-09-25 2021-07-28 아칠리온 파르마세우티칼스 인코포레이티드 보체 인자 d 억제제의 형태체 형태
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US20150148374A1 (en) 2015-05-28
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US9550755B2 (en) 2017-01-24
MX2015000537A (es) 2015-05-11
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