AU2013223749A1 - Stable dosage forms of imatinib mesylate - Google Patents
Stable dosage forms of imatinib mesylate Download PDFInfo
- Publication number
- AU2013223749A1 AU2013223749A1 AU2013223749A AU2013223749A AU2013223749A1 AU 2013223749 A1 AU2013223749 A1 AU 2013223749A1 AU 2013223749 A AU2013223749 A AU 2013223749A AU 2013223749 A AU2013223749 A AU 2013223749A AU 2013223749 A1 AU2013223749 A1 AU 2013223749A1
- Authority
- AU
- Australia
- Prior art keywords
- dosage form
- pharmaceutical dosage
- oral pharmaceutical
- pharmaceutically acceptable
- stable oral
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
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- 229960003685 imatinib mesylate Drugs 0.000 title claims abstract description 53
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- 239000005517 L01XE01 - Imatinib Substances 0.000 claims abstract description 19
- KTUFNOKKBVMGRW-UHFFFAOYSA-N imatinib Chemical compound C1CN(C)CCN1CC1=CC=C(C(=O)NC=2C=C(NC=3N=C(C=CN=3)C=3C=NC=CC=3)C(C)=CC=2)C=C1 KTUFNOKKBVMGRW-UHFFFAOYSA-N 0.000 claims abstract description 18
- 229960002411 imatinib Drugs 0.000 claims abstract description 17
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- A61K9/2893—Tablet coating processes
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/4833—Encapsulating processes; Filling of capsules
-
- B—PERFORMING OPERATIONS; TRANSPORTING
- B65—CONVEYING; PACKING; STORING; HANDLING THIN OR FILAMENTARY MATERIAL
- B65D—CONTAINERS FOR STORAGE OR TRANSPORT OF ARTICLES OR MATERIALS, e.g. BAGS, BARRELS, BOTTLES, BOXES, CANS, CARTONS, CRATES, DRUMS, JARS, TANKS, HOPPERS, FORWARDING CONTAINERS; ACCESSORIES, CLOSURES, OR FITTINGS THEREFOR; PACKAGING ELEMENTS; PACKAGES
- B65D81/00—Containers, packaging elements, or packages, for contents presenting particular transport or storage problems, or adapted to be used for non-packaging purposes after removal of contents
- B65D81/24—Adaptations for preventing deterioration or decay of contents; Applications to the container or packaging material of food preservatives, fungicides, pesticides or animal repellants
- B65D81/26—Adaptations for preventing deterioration or decay of contents; Applications to the container or packaging material of food preservatives, fungicides, pesticides or animal repellants with provision for draining away, or absorbing, or removing by ventilation, fluids, e.g. exuded by contents; Applications of corrosion inhibitors or desiccators
- B65D81/264—Adaptations for preventing deterioration or decay of contents; Applications to the container or packaging material of food preservatives, fungicides, pesticides or animal repellants with provision for draining away, or absorbing, or removing by ventilation, fluids, e.g. exuded by contents; Applications of corrosion inhibitors or desiccators for absorbing liquids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
- A61K9/1605—Excipients; Inactive ingredients
- A61K9/1611—Inorganic compounds
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/2027—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/4841—Filling excipients; Inactive ingredients
- A61K9/4858—Organic compounds
Landscapes
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Epidemiology (AREA)
- Medicinal Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Food Science & Technology (AREA)
- Mechanical Engineering (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| IN499DE2012 | 2012-02-21 | ||
| IN499/DEL/2012 | 2012-02-21 | ||
| IN498DE2012 | 2012-02-21 | ||
| IN498/DEL/2012 | 2012-02-21 | ||
| PCT/IB2013/051261 WO2013124774A1 (en) | 2012-02-21 | 2013-02-15 | Stable dosage forms of imatinib mesylate |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AU2013223749A1 true AU2013223749A1 (en) | 2014-09-11 |
Family
ID=48093035
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AU2013223749A Abandoned AU2013223749A1 (en) | 2012-02-21 | 2013-02-15 | Stable dosage forms of imatinib mesylate |
Country Status (7)
| Country | Link |
|---|---|
| US (1) | US20160015708A1 (enExample) |
| EP (1) | EP2817030A1 (enExample) |
| AU (1) | AU2013223749A1 (enExample) |
| IN (1) | IN2014DN07898A (enExample) |
| SG (1) | SG11201405099UA (enExample) |
| WO (1) | WO2013124774A1 (enExample) |
| ZA (1) | ZA201406139B (enExample) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| ES2683361T3 (es) * | 2013-05-14 | 2018-09-26 | Hetero Research Foundation | Composiciones de Imatinib |
| WO2019229648A1 (en) * | 2018-05-28 | 2019-12-05 | Shivalik Rasayan Limited | Oral compositions of imatinib mesylate |
Family Cites Families (13)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5521184A (en) | 1992-04-03 | 1996-05-28 | Ciba-Geigy Corporation | Pyrimidine derivatives and processes for the preparation thereof |
| CO4940418A1 (es) | 1997-07-18 | 2000-07-24 | Novartis Ag | Modificacion de cristal de un derivado de n-fenil-2- pirimidinamina, procesos para su fabricacion y su uso |
| ITMI992711A1 (it) | 1999-12-27 | 2001-06-27 | Novartis Ag | Composti organici |
| AU2002218262B2 (en) | 2000-10-27 | 2005-09-29 | Novartis Pharma Ag | Treatment of gastrointestinal stromal tumors |
| EP1243524A3 (en) * | 2001-03-16 | 2004-04-07 | Pfizer Products Inc. | Pharmaceutical kit for oxygen-sensitive drugs |
| GB0209265D0 (en) | 2002-04-23 | 2002-06-05 | Novartis Ag | Organic compounds |
| US8048883B2 (en) | 2004-02-11 | 2011-11-01 | Natco Pharma Limited | Polymorphic form of imatinib mesylate and a process for its preparation |
| DE602006012671D1 (de) | 2005-06-03 | 2010-04-15 | Elan Pharma Int Ltd | Nanoteilchenförmige imatinib-mesylat-formulierungen |
| BRPI0602338A (pt) | 2006-03-24 | 2007-12-11 | Univ Kyushu Nat Univ Corp | compostos orgánicos |
| US8414918B2 (en) | 2007-09-25 | 2013-04-09 | Teva Pharmaceutical Industries Ltd. | Stable imatinib compositions |
| US20130011477A1 (en) | 2010-03-29 | 2013-01-10 | Hetero Research Foundation | Stable Pharmaceutical Composition of Imatinib |
| WO2011158255A1 (en) * | 2010-06-16 | 2011-12-22 | Aptuit Laurus Private Limited | Process for preparation of stable imatintb mesylate alpha form |
| EP2603288A1 (en) * | 2010-08-11 | 2013-06-19 | Synthon BV | Pharmaceutical granulate comprising imatinib mesylate |
-
2013
- 2013-02-15 AU AU2013223749A patent/AU2013223749A1/en not_active Abandoned
- 2013-02-15 US US14/379,681 patent/US20160015708A1/en not_active Abandoned
- 2013-02-15 EP EP13716050.3A patent/EP2817030A1/en not_active Withdrawn
- 2013-02-15 WO PCT/IB2013/051261 patent/WO2013124774A1/en not_active Ceased
- 2013-02-15 IN IN7898DEN2014 patent/IN2014DN07898A/en unknown
- 2013-02-15 SG SG11201405099UA patent/SG11201405099UA/en unknown
-
2014
- 2014-08-21 ZA ZA2014/06139A patent/ZA201406139B/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| ZA201406139B (en) | 2015-05-27 |
| IN2014DN07898A (enExample) | 2015-04-24 |
| WO2013124774A1 (en) | 2013-08-29 |
| EP2817030A1 (en) | 2014-12-31 |
| US20160015708A1 (en) | 2016-01-21 |
| SG11201405099UA (en) | 2014-10-30 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| MK5 | Application lapsed section 142(2)(e) - patent request and compl. specification not accepted |