AU2012224634B2 - Preparation of a 1-amino-3-hydroxy-cyclobutane-1-carboxylic acid derivative - Google Patents
Preparation of a 1-amino-3-hydroxy-cyclobutane-1-carboxylic acid derivative Download PDFInfo
- Publication number
- AU2012224634B2 AU2012224634B2 AU2012224634A AU2012224634A AU2012224634B2 AU 2012224634 B2 AU2012224634 B2 AU 2012224634B2 AU 2012224634 A AU2012224634 A AU 2012224634A AU 2012224634 A AU2012224634 A AU 2012224634A AU 2012224634 B2 AU2012224634 B2 AU 2012224634B2
- Authority
- AU
- Australia
- Prior art keywords
- compound
- group
- palladium
- catalyst
- formula
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
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Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C229/00—Compounds containing amino and carboxyl groups bound to the same carbon skeleton
- C07C229/46—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino or carboxyl groups bound to carbon atoms of rings other than six-membered aromatic rings of the same carbon skeleton
- C07C229/48—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino or carboxyl groups bound to carbon atoms of rings other than six-membered aromatic rings of the same carbon skeleton with amino groups and carboxyl groups bound to carbon atoms of the same non-condensed ring
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C227/00—Preparation of compounds containing amino and carboxyl groups bound to the same carbon skeleton
- C07C227/14—Preparation of compounds containing amino and carboxyl groups bound to the same carbon skeleton from compounds containing already amino and carboxyl groups or derivatives thereof
- C07C227/16—Preparation of compounds containing amino and carboxyl groups bound to the same carbon skeleton from compounds containing already amino and carboxyl groups or derivatives thereof by reactions not involving the amino or carboxyl groups
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K51/00—Preparations containing radioactive substances for use in therapy or testing in vivo
- A61K51/02—Preparations containing radioactive substances for use in therapy or testing in vivo characterised by the carrier, i.e. characterised by the agent or material covalently linked or complexing the radioactive nucleus
- A61K51/04—Organic compounds
- A61K51/0404—Lipids, e.g. triglycerides; Polycationic carriers
- A61K51/0406—Amines, polyamines, e.g. spermine, spermidine, amino acids, (bis)guanidines
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C269/00—Preparation of derivatives of carbamic acid, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups
- C07C269/06—Preparation of derivatives of carbamic acid, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups by reactions not involving the formation of carbamate groups
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C2601/00—Systems containing only non-condensed rings
- C07C2601/04—Systems containing only non-condensed rings with a four-membered ring
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- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Optics & Photonics (AREA)
- Epidemiology (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Physics & Mathematics (AREA)
- Medicinal Chemistry (AREA)
- Biophysics (AREA)
- Pharmacology & Pharmacy (AREA)
- Molecular Biology (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Catalysts (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201161450177P | 2011-03-08 | 2011-03-08 | |
| US61/450,177 | 2011-03-08 | ||
| PCT/EP2012/053867 WO2012120025A1 (en) | 2011-03-08 | 2012-03-07 | Preparation of a 1-amino-3-hydroxy-cyclobutane-1-carboxylic acid derivative |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| AU2012224634A1 AU2012224634A1 (en) | 2013-08-08 |
| AU2012224634B2 true AU2012224634B2 (en) | 2016-09-08 |
Family
ID=45808953
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AU2012224634A Active AU2012224634B2 (en) | 2011-03-08 | 2012-03-07 | Preparation of a 1-amino-3-hydroxy-cyclobutane-1-carboxylic acid derivative |
Country Status (14)
| Country | Link |
|---|---|
| US (1) | US9242924B2 (enExample) |
| EP (1) | EP2683684B1 (enExample) |
| JP (1) | JP5938422B2 (enExample) |
| KR (1) | KR101904565B1 (enExample) |
| CN (1) | CN103415503B (enExample) |
| AU (1) | AU2012224634B2 (enExample) |
| BR (1) | BR112013020627B1 (enExample) |
| CA (1) | CA2828975C (enExample) |
| DK (1) | DK2683684T3 (enExample) |
| ES (1) | ES2657894T3 (enExample) |
| MX (1) | MX341089B (enExample) |
| NO (1) | NO2683684T3 (enExample) |
| RU (1) | RU2596829C2 (enExample) |
| WO (1) | WO2012120025A1 (enExample) |
Citations (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP1978015A1 (en) * | 2005-11-29 | 2008-10-08 | Nihon Medi-Physics Co., Ltd. | Precursor compound of radioactive halogen labeled organic compound |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AU4314700A (en) | 1999-04-28 | 2000-11-17 | Banyu Pharmaceutical Co., Ltd. | Processes for the preparation of piperidylmethylpyridine derivatives |
| JP4744163B2 (ja) * | 2005-02-28 | 2011-08-10 | 広栄化学工業株式会社 | ビピリジン類の製造方法 |
| TW200736203A (en) * | 2005-11-18 | 2007-10-01 | Glaxo Group Ltd | New pleuromutilin derivative and its use |
| JP5518337B2 (ja) * | 2006-12-27 | 2014-06-11 | 日本メジフィジックス株式会社 | 放射性ハロゲン標識有機化合物の前駆体化合物の製造方法 |
| MX2010010012A (es) | 2008-03-11 | 2010-10-20 | Incyte Corp | Derivados de azetidina y ciclobutano como inhibidores de jak. |
| JP5718233B2 (ja) | 2008-10-20 | 2015-05-13 | ザ ガバメント オブ ザ ユナイテッド ステイツ オブ アメリカ アズ リプレゼンテッド バイ ザ セクレタリー オブ ザ デパートメント オブ ヘルス アンド ヒューマン サービシーズ | 甲状腺刺激ホルモン受容体(tshr)の低分子量アゴニスト |
| JP2012532834A (ja) | 2009-07-11 | 2012-12-20 | バイエル ファーマ アクチエンゲゼルシャフト | シクロアルキル基を用いる放射性標識方法 |
-
2012
- 2012-03-07 NO NO12707320A patent/NO2683684T3/no unknown
- 2012-03-07 US US14/002,184 patent/US9242924B2/en active Active
- 2012-03-07 DK DK12707320.3T patent/DK2683684T3/en active
- 2012-03-07 JP JP2013557076A patent/JP5938422B2/ja active Active
- 2012-03-07 WO PCT/EP2012/053867 patent/WO2012120025A1/en not_active Ceased
- 2012-03-07 CN CN201280012007.4A patent/CN103415503B/zh active Active
- 2012-03-07 RU RU2013139061/04A patent/RU2596829C2/ru active
- 2012-03-07 AU AU2012224634A patent/AU2012224634B2/en active Active
- 2012-03-07 KR KR1020137023602A patent/KR101904565B1/ko active Active
- 2012-03-07 MX MX2013010254A patent/MX341089B/es active IP Right Grant
- 2012-03-07 EP EP12707320.3A patent/EP2683684B1/en active Active
- 2012-03-07 ES ES12707320.3T patent/ES2657894T3/es active Active
- 2012-03-07 BR BR112013020627A patent/BR112013020627B1/pt active IP Right Grant
- 2012-03-07 CA CA2828975A patent/CA2828975C/en active Active
Patent Citations (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP1978015A1 (en) * | 2005-11-29 | 2008-10-08 | Nihon Medi-Physics Co., Ltd. | Precursor compound of radioactive halogen labeled organic compound |
Non-Patent Citations (2)
| Title |
|---|
| SHOUP, T.M. et al, Journal of Labelled Compounds and Radiopharmaceuticals, 1999, vol. 42, pp. 215-225 * |
| YU, W. et al, Bioorganic & Medicinal Chemistry, 2009, vol. 17, pp. 1982-1990 * |
Also Published As
| Publication number | Publication date |
|---|---|
| EP2683684A1 (en) | 2014-01-15 |
| CA2828975A1 (en) | 2012-09-13 |
| US9242924B2 (en) | 2016-01-26 |
| BR112013020627B1 (pt) | 2019-12-03 |
| WO2012120025A1 (en) | 2012-09-13 |
| MX2013010254A (es) | 2013-11-18 |
| DK2683684T3 (en) | 2018-02-05 |
| NO2683684T3 (enExample) | 2018-06-02 |
| JP2014514268A (ja) | 2014-06-19 |
| KR20140049975A (ko) | 2014-04-28 |
| CA2828975C (en) | 2019-07-09 |
| BR112013020627A2 (pt) | 2016-10-04 |
| RU2013139061A (ru) | 2015-04-20 |
| US20130345468A1 (en) | 2013-12-26 |
| ES2657894T3 (es) | 2018-03-07 |
| MX341089B (es) | 2016-08-08 |
| EP2683684B1 (en) | 2018-01-03 |
| CN103415503A (zh) | 2013-11-27 |
| JP5938422B2 (ja) | 2016-06-22 |
| KR101904565B1 (ko) | 2018-10-04 |
| RU2596829C2 (ru) | 2016-09-10 |
| CN103415503B (zh) | 2015-09-16 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FGA | Letters patent sealed or granted (standard patent) |