AU2011339150B2 - Complex formulation comprising lercanidipine hydrochloride and valsartan and method for the preparation thereof - Google Patents
Complex formulation comprising lercanidipine hydrochloride and valsartan and method for the preparation thereof Download PDFInfo
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- AU2011339150B2 AU2011339150B2 AU2011339150A AU2011339150A AU2011339150B2 AU 2011339150 B2 AU2011339150 B2 AU 2011339150B2 AU 2011339150 A AU2011339150 A AU 2011339150A AU 2011339150 A AU2011339150 A AU 2011339150A AU 2011339150 B2 AU2011339150 B2 AU 2011339150B2
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- Prior art keywords
- valsartan
- lercanidipine hydrochloride
- composition according
- granules
- lercanidipine
- Prior art date
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- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
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- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
- A61K9/1605—Excipients; Inactive ingredients
- A61K9/1629—Organic macromolecular compounds
- A61K9/1652—Polysaccharides, e.g. alginate, cellulose derivatives; Cyclodextrin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/2027—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
- A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
- A61K9/2086—Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat
- A61K9/209—Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat containing drug in at least two layers or in the core and in at least one outer layer
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2095—Tabletting processes; Dosage units made by direct compression of powders or specially processed granules, by eliminating solvents, by melt-extrusion, by injection molding, by 3D printing
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
- A61K9/5084—Mixtures of one or more drugs in different galenical forms, at least one of which being granules, microcapsules or (coated) microparticles according to A61K9/16 or A61K9/50, e.g. for obtaining a specific release pattern or for combining different drugs
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
Landscapes
- Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical & Material Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- Epidemiology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| KR20100125804 | 2010-12-09 | ||
| KR10-2010-0125804 | 2010-12-09 | ||
| PCT/KR2011/009413 WO2012077968A2 (en) | 2010-12-09 | 2011-12-07 | Complex formulation comprising lercanidipine hydrochloride and valsartan and method for the preparation thereof |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| AU2011339150A1 AU2011339150A1 (en) | 2013-06-06 |
| AU2011339150B2 true AU2011339150B2 (en) | 2015-09-10 |
Family
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AU2011339150A Ceased AU2011339150B2 (en) | 2010-12-09 | 2011-12-07 | Complex formulation comprising lercanidipine hydrochloride and valsartan and method for the preparation thereof |
Country Status (17)
| Country | Link |
|---|---|
| EP (1) | EP2648730A4 (es) |
| KR (1) | KR101414814B1 (es) |
| CN (1) | CN103249415B (es) |
| AR (1) | AR084195A1 (es) |
| AU (1) | AU2011339150B2 (es) |
| BR (1) | BR112013013415A2 (es) |
| CL (1) | CL2013001626A1 (es) |
| CO (1) | CO6721030A2 (es) |
| DO (1) | DOP2013000115A (es) |
| EA (1) | EA201390844A1 (es) |
| IL (1) | IL226449A0 (es) |
| MX (1) | MX2013005716A (es) |
| PE (1) | PE20140699A1 (es) |
| SG (1) | SG190326A1 (es) |
| UA (1) | UA108277C2 (es) |
| UY (1) | UY33772A (es) |
| WO (1) | WO2012077968A2 (es) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN102755322B (zh) * | 2012-07-24 | 2013-12-11 | 兆科药业（广州）有限公司 | 一种乐卡地平和阿托伐他汀复方制剂 |
| US20160045497A1 (en) * | 2013-03-12 | 2016-02-18 | Lg Life Sciences Ltd. | Complex preparation including valsartan and rosuvastatin calcium and manufacturing method therefor |
| WO2019008485A1 (en) | 2017-07-06 | 2019-01-10 | Mankind Pharma Ltd | FIXED DOSE PHARMACEUTICAL COMPOSITION BASED ON VALSARTAN AND SACUBITRIL |
| KR102233986B1 (ko) * | 2019-06-25 | 2021-03-30 | 경남과학기술대학교 산학협력단 | 라푸티딘 및 이르소글라딘을 함유하는 고형 약제학적 조성물 및 이의 제조방법 |
Citations (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20040198789A1 (en) * | 2003-02-28 | 2004-10-07 | Recordati Ireland Limited | Lercanidipine/ARB/diuretic therapeutic combinations |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP1694305B1 (en) * | 2003-12-01 | 2019-10-16 | Recordati Ireland Limited | Pharmaceutical compositions comprising lercanidipine |
| WO2007001067A2 (en) | 2005-06-27 | 2007-01-04 | Daiichi Sankyo Company, Limited | Solid dosage form comprising an angiotensin ii receptor antagonist and a calcium channel blocker |
| KR100888131B1 (ko) * | 2006-10-10 | 2009-03-11 | 한올제약주식회사 | 시간차 투약 원리를 이용한 심혈관계 질환 치료용 복합제제 |
-
2011
- 2011-12-06 UY UY0001033772A patent/UY33772A/es not_active Application Discontinuation
- 2011-12-07 AR ARP110104583A patent/AR084195A1/es unknown
- 2011-12-07 BR BR112013013415A patent/BR112013013415A2/pt not_active IP Right Cessation
- 2011-12-07 MX MX2013005716A patent/MX2013005716A/es unknown
- 2011-12-07 EA EA201390844A patent/EA201390844A1/ru unknown
- 2011-12-07 CN CN201180058951.9A patent/CN103249415B/zh active Active
- 2011-12-07 UA UAA201307936A patent/UA108277C2/ru unknown
- 2011-12-07 WO PCT/KR2011/009413 patent/WO2012077968A2/en active Application Filing
- 2011-12-07 AU AU2011339150A patent/AU2011339150B2/en not_active Ceased
- 2011-12-07 SG SG2013038211A patent/SG190326A1/en unknown
- 2011-12-07 KR KR1020110130400A patent/KR101414814B1/ko active IP Right Grant
- 2011-12-07 PE PE2013001346A patent/PE20140699A1/es not_active Application Discontinuation
- 2011-12-07 EP EP11847739.7A patent/EP2648730A4/en not_active Withdrawn
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2013
- 2013-05-20 IL IL226449A patent/IL226449A0/en unknown
- 2013-05-21 DO DO2013000115A patent/DOP2013000115A/es unknown
- 2013-06-06 CL CL2013001626A patent/CL2013001626A1/es unknown
- 2013-06-21 CO CO13147794A patent/CO6721030A2/es unknown
Patent Citations (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20040198789A1 (en) * | 2003-02-28 | 2004-10-07 | Recordati Ireland Limited | Lercanidipine/ARB/diuretic therapeutic combinations |
Also Published As
| Publication number | Publication date |
|---|---|
| KR20120089787A (ko) | 2012-08-13 |
| MX2013005716A (es) | 2013-06-12 |
| UA108277C2 (ru) | 2015-04-10 |
| DOP2013000115A (es) | 2014-07-31 |
| BR112013013415A2 (pt) | 2019-09-24 |
| EP2648730A4 (en) | 2014-08-06 |
| UY33772A (es) | 2012-07-31 |
| CN103249415B (zh) | 2017-12-12 |
| PE20140699A1 (es) | 2014-06-13 |
| EA201390844A1 (ru) | 2013-11-29 |
| SG190326A1 (en) | 2013-06-28 |
| EP2648730A2 (en) | 2013-10-16 |
| IL226449A0 (en) | 2013-07-31 |
| CO6721030A2 (es) | 2013-07-31 |
| WO2012077968A2 (en) | 2012-06-14 |
| CL2013001626A1 (es) | 2013-10-04 |
| KR101414814B1 (ko) | 2014-07-21 |
| CN103249415A (zh) | 2013-08-14 |
| AU2011339150A1 (en) | 2013-06-06 |
| WO2012077968A3 (en) | 2012-07-26 |
| AR084195A1 (es) | 2013-04-24 |
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| FGA | Letters patent sealed or granted (standard patent) | ||
| HB | Alteration of name in register |
Owner name: LG CHEM, LTD. Free format text: FORMER NAME(S): LG LIFE SCIENCES LTD. |