AU2010298169B2 - Bridged heterocyclic compounds and methods of use - Google Patents

Bridged heterocyclic compounds and methods of use Download PDF

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Publication number
AU2010298169B2
AU2010298169B2 AU2010298169A AU2010298169A AU2010298169B2 AU 2010298169 B2 AU2010298169 B2 AU 2010298169B2 AU 2010298169 A AU2010298169 A AU 2010298169A AU 2010298169 A AU2010298169 A AU 2010298169A AU 2010298169 B2 AU2010298169 B2 AU 2010298169B2
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substituted
unsubstituted
variation
formula
alkyl
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AU2010298169A1 (en
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Sarvajit Chakravarty
Rajendra Parasmal Jain
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Medivation Technologies LLC
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Medivation Technologies LLC
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Priority to AU2013203658A priority Critical patent/AU2013203658A1/en
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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/08Bridged systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/18Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/08Bridged systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/12Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
    • C07D471/18Bridged systems

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  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Psychiatry (AREA)
  • Hospice & Palliative Care (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
AU2010298169A 2009-09-23 2010-09-23 Bridged heterocyclic compounds and methods of use Ceased AU2010298169B2 (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
AU2013203658A AU2013203658A1 (en) 2009-09-23 2013-04-11 Bridged heterocyclic compounds and methods of use

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US24515109P 2009-09-23 2009-09-23
US61/245,151 2009-09-23
PCT/US2010/050081 WO2011038164A1 (en) 2009-09-23 2010-09-23 Bridged heterocyclic compounds and methods of use

Related Child Applications (1)

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AU2013203658A Division AU2013203658A1 (en) 2009-09-23 2013-04-11 Bridged heterocyclic compounds and methods of use

Publications (2)

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AU2010298169A1 AU2010298169A1 (en) 2012-04-19
AU2010298169B2 true AU2010298169B2 (en) 2015-10-29

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AU2010298169A Ceased AU2010298169B2 (en) 2009-09-23 2010-09-23 Bridged heterocyclic compounds and methods of use

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US (2) US9006234B2 (enExample)
EP (1) EP2480081A4 (enExample)
JP (1) JP5869484B2 (enExample)
CN (1) CN102711466A (enExample)
AU (1) AU2010298169B2 (enExample)
BR (1) BR112012006648A2 (enExample)
CA (1) CA2775216A1 (enExample)
WO (1) WO2011038164A1 (enExample)

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RU2544856C2 (ru) 2008-01-25 2015-03-20 Сергей Олегович Бачурин НОВЫЕ ПРОИЗВОДНЫЕ 2,3,4,5-ТЕТРАГИДРО-1-ПИРИДО[4,3-b]ИНДОЛА И СПОСОБЫ ИХ ПРИМЕНЕНИЯ
JP5586577B2 (ja) 2008-03-24 2014-09-10 メディベイション テクノロジーズ, インコーポレイテッド 架橋複素環化合物およびその使用
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JP5827943B2 (ja) 2009-04-29 2015-12-02 メディベイション テクノロジーズ, インコーポレイテッド ピリド[4,3−b]インドールおよびその使用方法
US9255094B2 (en) 2009-04-29 2016-02-09 Medivation Technologies, Inc. Pyrido[4,3-B]indoles and methods of use
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EP2480078A4 (en) 2009-09-23 2013-03-06 Medivation Technologies Inc PYRIDO- [4,3-B] INDOLE AND USE METHOD THEREFOR
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