AU2009254176A1 - 4, 6-diphenylpyrid-2-0nes against cancer - Google Patents
4, 6-diphenylpyrid-2-0nes against cancer Download PDFInfo
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- AU2009254176A1 AU2009254176A1 AU2009254176A AU2009254176A AU2009254176A1 AU 2009254176 A1 AU2009254176 A1 AU 2009254176A1 AU 2009254176 A AU2009254176 A AU 2009254176A AU 2009254176 A AU2009254176 A AU 2009254176A AU 2009254176 A1 AU2009254176 A1 AU 2009254176A1
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- lower alkyl
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- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/18—Drugs for disorders of the alimentary tract or the digestive system for pancreatic disorders, e.g. pancreatic enzymes
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/08—Drugs for disorders of the urinary system of the prostate
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/10—Drugs for disorders of the urinary system of the bladder
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/12—Drugs for disorders of the urinary system of the kidneys
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/04—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Urology & Nephrology (AREA)
- Endocrinology (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Reproductive Health (AREA)
- Gastroenterology & Hepatology (AREA)
- Dermatology (AREA)
- Pulmonology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Pyridine Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GBGB0810228.7A GB0810228D0 (en) | 2008-06-04 | 2008-06-04 | Novel compounds |
| GB0810228.7 | 2008-06-04 | ||
| PCT/EP2009/004005 WO2009146910A1 (en) | 2008-06-04 | 2009-06-04 | 4, 6-diphenylpyrid-2-0nes against cancer |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AU2009254176A1 true AU2009254176A1 (en) | 2009-12-10 |
Family
ID=39638174
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AU2009254176A Abandoned AU2009254176A1 (en) | 2008-06-04 | 2009-06-04 | 4, 6-diphenylpyrid-2-0nes against cancer |
Country Status (7)
| Country | Link |
|---|---|
| US (2) | US8236827B2 (enExample) |
| EP (1) | EP2310370A1 (enExample) |
| JP (1) | JP2011521986A (enExample) |
| AU (1) | AU2009254176A1 (enExample) |
| CA (1) | CA2726939A1 (enExample) |
| GB (1) | GB0810228D0 (enExample) |
| WO (1) | WO2009146910A1 (enExample) |
Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2012058550A2 (en) * | 2010-10-29 | 2012-05-03 | Fox Chase Cancer Center | Methods for screening compounds for capability to inhibit premalignant squamous epithelial cell progression to a malignant state |
| WO2012075136A2 (en) * | 2010-11-30 | 2012-06-07 | Fox Chase Cancer Center | Targeting of cyp1b1 in the treatment of head and neck cancer and lung cancer |
| CN103387574A (zh) * | 2012-05-07 | 2013-11-13 | 北京以岭药业有限公司 | 一种表小檗碱的合成方法 |
| CN107591180A (zh) * | 2016-07-07 | 2018-01-16 | 中芯国际集成电路制造(上海)有限公司 | 非挥发性存储器及其读取数据的方法 |
| WO2018011376A1 (en) * | 2016-07-13 | 2018-01-18 | Centre National De La Recherche Scientifique - Cnrs - | Pyrimidinone derivatives and uses thereof to neutralize the biological activity of chemokines |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB0123777D0 (en) | 2001-10-03 | 2001-11-21 | Cancer Res Ventures Ltd | Substituted chalcones as therapeutic agents |
| US7910742B2 (en) | 2005-09-29 | 2011-03-22 | Abbott Laboratories | Survivin inhibitors |
| JP2010525062A (ja) * | 2007-04-25 | 2010-07-22 | エグゼリクシス， インコーポレイテッド | Ｐｉｍモジュレーターとしてのピリミジノン類 |
-
2008
- 2008-06-04 GB GBGB0810228.7A patent/GB0810228D0/en not_active Ceased
-
2009
- 2009-06-04 EP EP09757293A patent/EP2310370A1/en not_active Withdrawn
- 2009-06-04 AU AU2009254176A patent/AU2009254176A1/en not_active Abandoned
- 2009-06-04 US US12/478,587 patent/US8236827B2/en not_active Expired - Fee Related
- 2009-06-04 JP JP2011512021A patent/JP2011521986A/ja active Pending
- 2009-06-04 WO PCT/EP2009/004005 patent/WO2009146910A1/en not_active Ceased
- 2009-06-04 CA CA2726939A patent/CA2726939A1/en not_active Abandoned
-
2012
- 2012-07-25 US US13/557,508 patent/US20130023567A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| WO2009146910A1 (en) | 2009-12-10 |
| US8236827B2 (en) | 2012-08-07 |
| EP2310370A1 (en) | 2011-04-20 |
| CA2726939A1 (en) | 2009-12-10 |
| US20100168180A1 (en) | 2010-07-01 |
| US20130023567A1 (en) | 2013-01-24 |
| WO2009146910A8 (en) | 2011-04-07 |
| GB0810228D0 (en) | 2008-07-09 |
| JP2011521986A (ja) | 2011-07-28 |
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