AU2006317545B2 - Compositions and methods for modulating gated ion channels - Google Patents

Compositions and methods for modulating gated ion channels Download PDF

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AU2006317545B2
AU2006317545B2 AU2006317545A AU2006317545A AU2006317545B2 AU 2006317545 B2 AU2006317545 B2 AU 2006317545B2 AU 2006317545 A AU2006317545 A AU 2006317545A AU 2006317545 A AU2006317545 A AU 2006317545A AU 2006317545 B2 AU2006317545 B2 AU 2006317545B2
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alkoxy
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AU2006317545A1 (en
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Philip K. Ahring
Joachim Demnitz
Zhonghong Gan
Nachhattarpal Gill
Rahul Vohra
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Aros Pharma ApS
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AU2006317545A 2005-11-23 2006-11-22 Compositions and methods for modulating gated ion channels Ceased AU2006317545B2 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US73960005P 2005-11-23 2005-11-23
US60/739,600 2005-11-23
PCT/CA2006/001897 WO2007059608A1 (en) 2005-11-23 2006-11-22 Compositions and methods for modulating gated ion channels

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AU2006317545A1 AU2006317545A1 (en) 2007-05-31
AU2006317545B2 true AU2006317545B2 (en) 2012-04-12

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AU2006317545A Ceased AU2006317545B2 (en) 2005-11-23 2006-11-22 Compositions and methods for modulating gated ion channels

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US (2) US7718641B2 (ko)
EP (1) EP1957486A4 (ko)
JP (1) JP2009516712A (ko)
KR (1) KR20080070749A (ko)
CN (1) CN101346375B (ko)
AU (1) AU2006317545B2 (ko)
BR (1) BRPI0618863A2 (ko)
CA (1) CA2630617C (ko)
WO (1) WO2007059608A1 (ko)

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WO2008144931A1 (en) * 2007-05-30 2008-12-04 Painceptor Pharma Corporation Compositions and methods for modulating gated ion channels
EP2288922B1 (en) * 2008-05-08 2016-08-17 University of Utah Research Foundation Sensory receptors for chronic fatigue and pain and uses thereof
AU2009332651A1 (en) * 2008-12-26 2011-12-01 Glenmark Pharmaceuticals, S.A. Fused imidazole derivatives as TRPV3 antagonist
US9211313B2 (en) * 2011-01-14 2015-12-15 The Research Foundation Of State University Of New York Methods and compound to inhibit Ca2+ permeable cation conductance
JP5971657B2 (ja) 2011-04-20 2016-08-17 塩野義製薬株式会社 Ｔｒｐｖ４阻害活性を有する芳香族複素環誘導体
JO3154B1 (ar) * 2011-06-17 2017-09-20 Glaxosmithkline Llc عوامل مضادة لـ trpv4
US9499533B2 (en) 2012-03-27 2016-11-22 Shionogi & Co., Ltd. Aromatic 5-membered heterocyclic derivative having TRPV4-Inhibiting activity
WO2015021988A1 (en) 2013-08-12 2015-02-19 Aros Pharma Aps Pyrrolo-isoquinoline compounds for treatment of pain associated with interstitial cystitis/bladder pain syndrome
KR102084185B1 (ko) 2013-08-29 2020-03-04 주식회사 대웅제약 테트라히드로사이클로펜타피롤 유도체 및 이의 제조방법
JPWO2015046193A1 (ja) 2013-09-25 2017-03-09 塩野義製薬株式会社 Ｔｒｐｖ４阻害活性を有する芳香族複素環式アミン誘導体
WO2018151240A1 (ja) * 2017-02-17 2018-08-23 第一三共株式会社 ３，６，７，８－テトラヒドロシクロペンタ［ｅ］インドール化合物
WO2018151239A1 (ja) * 2017-02-17 2018-08-23 第一三共株式会社 ３，６－ジヒドロ－２Ｈ－フロ［２，３－ｅ］インドール化合物
CN109364248B (zh) * 2018-10-16 2021-05-18 哈尔滨医科大学 ENaC及其抑制剂在预防、缓解和/或治疗动脉粥样硬化中的应用

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AU2006317545A1 (en) 2007-05-31
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WO2007059608A1 (en) 2007-05-31
US7718641B2 (en) 2010-05-18
US20070191418A1 (en) 2007-08-16
CA2630617C (en) 2014-03-25
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CN101346375A (zh) 2009-01-14
BRPI0618863A2 (pt) 2016-09-13
US20100197721A1 (en) 2010-08-05
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KR20080070749A (ko) 2008-07-30
CA2630617A1 (en) 2007-05-31

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