AU2005282290B2 - Combination of organic compounds - Google Patents

Combination of organic compounds Download PDF

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Publication number
AU2005282290B2
AU2005282290B2 AU2005282290A AU2005282290A AU2005282290B2 AU 2005282290 B2 AU2005282290 B2 AU 2005282290B2 AU 2005282290 A AU2005282290 A AU 2005282290A AU 2005282290 A AU2005282290 A AU 2005282290A AU 2005282290 B2 AU2005282290 B2 AU 2005282290B2
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AU
Australia
Prior art keywords
phenyl
pharmaceutically acceptable
disease
disorder
dihydro
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
AU2005282290A
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English (en)
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AU2005282290A1 (en
Inventor
Hong Chen
William Maher
Michele Mercuri
Meenakshi Nevatia
Pei-Ran Wang
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Novartis AG
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Novartis AG
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Application filed by Novartis AG filed Critical Novartis AG
Publication of AU2005282290A1 publication Critical patent/AU2005282290A1/en
Application granted granted Critical
Publication of AU2005282290B2 publication Critical patent/AU2005282290B2/en
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

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Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/42—Oxazoles
    • A61K31/422—Oxazoles not condensed and containing further heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A61K31/52—Purines, e.g. adenine
    • A61K31/522—Purines, e.g. adenine having oxo groups directly attached to the heterocyclic ring, e.g. hypoxanthine, guanine, acyclovir
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
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    • A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
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    • A—HUMAN NECESSITIES
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    • A—HUMAN NECESSITIES
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    • A—HUMAN NECESSITIES
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    • A61P29/02—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID] without antiinflammatory effect
    • A—HUMAN NECESSITIES
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    • A—HUMAN NECESSITIES
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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    • A—HUMAN NECESSITIES
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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
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    • A—HUMAN NECESSITIES
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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    • A—HUMAN NECESSITIES
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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    • A—HUMAN NECESSITIES
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    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/38—Drugs for disorders of the endocrine system of the suprarenal hormones
    • A61P5/42—Drugs for disorders of the endocrine system of the suprarenal hormones for decreasing, blocking or antagonising the activity of mineralocorticosteroids
    • A—HUMAN NECESSITIES
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    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives

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  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Diabetes (AREA)
  • Epidemiology (AREA)
  • Hematology (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Cardiology (AREA)
  • Addiction (AREA)
  • Psychiatry (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pulmonology (AREA)
  • Obesity (AREA)
  • Urology & Nephrology (AREA)
  • Endocrinology (AREA)
  • Rheumatology (AREA)
  • Immunology (AREA)
  • Dermatology (AREA)
  • Pain & Pain Management (AREA)
  • Hospice & Palliative Care (AREA)
  • Reproductive Health (AREA)
  • Ophthalmology & Optometry (AREA)
  • Emergency Medicine (AREA)
  • Child & Adolescent Psychology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Gastroenterology & Hepatology (AREA)
AU2005282290A 2004-09-09 2005-09-08 Combination of organic compounds Expired - Fee Related AU2005282290B2 (en)

Applications Claiming Priority (7)

Application Number Priority Date Filing Date Title
US60831004P 2004-09-09 2004-09-09
US60/608,310 2004-09-09
US60957704P 2004-09-14 2004-09-14
US60/609,577 2004-09-14
US68973805P 2005-06-10 2005-06-10
US60/689,738 2005-06-10
PCT/US2005/032224 WO2006029349A1 (en) 2004-09-09 2005-09-08 Combination of organic compounds

Publications (2)

Publication Number Publication Date
AU2005282290A1 AU2005282290A1 (en) 2006-03-16
AU2005282290B2 true AU2005282290B2 (en) 2009-06-25

Family

ID=35385557

Family Applications (1)

Application Number Title Priority Date Filing Date
AU2005282290A Expired - Fee Related AU2005282290B2 (en) 2004-09-09 2005-09-08 Combination of organic compounds

Country Status (13)

Country Link
US (1) US20070299047A1 (OSRAM)
EP (1) EP1791600A1 (OSRAM)
JP (1) JP2008512486A (OSRAM)
KR (1) KR20070106677A (OSRAM)
AR (1) AR050631A1 (OSRAM)
AU (1) AU2005282290B2 (OSRAM)
BR (1) BRPI0515185A (OSRAM)
CA (1) CA2578290A1 (OSRAM)
GT (1) GT200500246A (OSRAM)
MX (1) MX2007002879A (OSRAM)
PE (1) PE20060594A1 (OSRAM)
TW (1) TW200621220A (OSRAM)
WO (1) WO2006029349A1 (OSRAM)

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SE521512C2 (sv) 2001-06-25 2003-11-11 Niconovum Ab Anordning för administrering av en substans till främre delen av en individs munhåla
ATE359075T1 (de) 2002-12-20 2007-05-15 Niconovum Ab Chemisch und physikalisch stabiles teilchenförmiges material enthaltend nikotin und microcrystalline cellulose
CA2646942C (en) 2006-03-16 2014-07-29 Niconovum Ab Improved snuff composition
EP1972335A1 (en) * 2007-03-23 2008-09-24 Krka Solid dosage forms comprising aliskiren and pharmaceutically acceptable salts thereof
AU2013201888B2 (en) * 2007-04-11 2016-02-25 Omeros Corporation Compositions and methods for prophylaxis and treatment of addictions
US11241420B2 (en) 2007-04-11 2022-02-08 Omeros Corporation Compositions and methods for prophylaxis and treatment of addictions
US20160331729A9 (en) * 2007-04-11 2016-11-17 Omeros Corporation Compositions and methods for prophylaxis and treatment of addictions
EP3053440B1 (en) 2007-04-11 2020-08-12 Omeros Corporation Compositions and methods for prophylaxis and treatment of addictions
IE20070928A1 (en) * 2007-12-21 2009-09-30 Giuliani Int Ltd Multi target ligands
WO2009154230A1 (ja) * 2008-06-17 2009-12-23 持田製薬株式会社 非アルコール性脂肪肝炎の予防／改善・治療薬
AU2010213093B2 (en) 2009-02-16 2016-01-07 Nogra Pharma Limited Alkylamido compounds and uses thereof
CA2754901A1 (en) 2009-03-11 2010-09-16 Omeros Corporation Compositions and methods for prophylaxis and treatment of addictions
WO2011100659A2 (en) * 2010-02-12 2011-08-18 Kitov Pharmaceutical Ltd. Ameliorating drug-induced elevations in blood pressure by adjunctive use of antihypertensive drugs
CN107899012A (zh) 2011-01-11 2018-04-13 戴麦里克斯生物科学有限公司 联合疗法
WO2013071077A1 (en) * 2011-11-09 2013-05-16 Cornell University The use of pan-ppar agonists for prevention and treatment of huntington's disease and tauopathies
CN104254327A (zh) 2012-02-09 2014-12-31 诺格拉制药有限公司 治疗纤维化的方法
JP2021534141A (ja) * 2018-08-10 2021-12-09 セルビシオ アンダルーサ デ サルー アルコール使用障害の治療剤
EP4495101A3 (en) 2019-02-08 2025-04-30 Nogra Pharma Limited Process of making 3-(4'-aminophenyl)-2-methoxypropionic acid, and analogs and intermediates thereof
IL303347A (en) 2020-12-03 2023-08-01 Delta 4 Gmbh Clopidogrel for use in the treatment of focal segmental glomerulosclerosis (fsgs)

Citations (3)

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WO2003043985A1 (en) * 2001-11-21 2003-05-30 Novartis Ag Heterocyclic compounds and methods of use
US20030139429A1 (en) * 2001-09-27 2003-07-24 Cohen David Saul Combinations
AU2004240754A1 (en) * 2003-05-20 2004-12-02 Novartis Ag N-acyl nitrogen heterocycles as ligands of Peroxisome Proliferator-Activated Receptors

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US3800038A (en) * 1972-04-21 1974-03-26 Biolog Concepts Inc Uterine administraton of eutectic solid solutions of steroid hormones in a steroidal lipid carrier
FR2530247B1 (fr) * 1982-07-13 1986-05-16 Sanofi Sa Nouveaux derives de la thieno (3, 2-c) pyridine, leur procede de preparation et leur application therapeutique
US5631365A (en) * 1993-09-21 1997-05-20 Schering Corporation Hydroxy-substituted azetidinone compounds useful as hypocholesterolemic agents
AR005245A1 (es) * 1995-12-21 1999-04-28 Astrazeneca Ab Prodrogas de inhibidores de trombina, una formulación farmaceutica que las comprende, el uso de dichas prodrogas para la manufactura de un medicamento y un procedimiento para su preparacion
US6071539A (en) * 1996-09-20 2000-06-06 Ethypharm, Sa Effervescent granules and methods for their preparation
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Patent Citations (3)

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Publication number Priority date Publication date Assignee Title
US20030139429A1 (en) * 2001-09-27 2003-07-24 Cohen David Saul Combinations
WO2003043985A1 (en) * 2001-11-21 2003-05-30 Novartis Ag Heterocyclic compounds and methods of use
AU2004240754A1 (en) * 2003-05-20 2004-12-02 Novartis Ag N-acyl nitrogen heterocycles as ligands of Peroxisome Proliferator-Activated Receptors

Also Published As

Publication number Publication date
AR050631A1 (es) 2006-11-08
AU2005282290A1 (en) 2006-03-16
BRPI0515185A (pt) 2008-07-22
CA2578290A1 (en) 2006-03-16
WO2006029349A1 (en) 2006-03-16
EP1791600A1 (en) 2007-06-06
MX2007002879A (es) 2007-04-23
KR20070106677A (ko) 2007-11-05
TW200621220A (en) 2006-07-01
JP2008512486A (ja) 2008-04-24
GT200500246A (es) 2006-04-17
PE20060594A1 (es) 2006-08-18
US20070299047A1 (en) 2007-12-27

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