AU2005230837A1 - 1,3,4-oxadiazol-2-ones as PPAR delta modulators - Google Patents
1,3,4-oxadiazol-2-ones as PPAR delta modulators Download PDFInfo
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- AU2005230837A1 AU2005230837A1 AU2005230837A AU2005230837A AU2005230837A1 AU 2005230837 A1 AU2005230837 A1 AU 2005230837A1 AU 2005230837 A AU2005230837 A AU 2005230837A AU 2005230837 A AU2005230837 A AU 2005230837A AU 2005230837 A1 AU2005230837 A1 AU 2005230837A1
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- Inks, Pencil-Leads, Or Crayons (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US55841904P | 2004-04-01 | 2004-04-01 | |
| US60/558,419 | 2004-04-01 | ||
| PCT/US2005/010854 WO2005097762A2 (en) | 2004-04-01 | 2005-03-30 | 1,3,4-oxadiazol-2-ones as ppar delta modulators |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AU2005230837A1 true AU2005230837A1 (en) | 2005-10-20 |
Family
ID=34972933
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AU2005230837A Abandoned AU2005230837A1 (en) | 2004-04-01 | 2005-03-30 | 1,3,4-oxadiazol-2-ones as PPAR delta modulators |
Country Status (17)
| Country | Link |
|---|---|
| US (1) | US7576109B2 (https=) |
| EP (1) | EP1735303B1 (https=) |
| JP (1) | JP4813460B2 (https=) |
| KR (1) | KR20060135854A (https=) |
| CN (1) | CN100516065C (https=) |
| AT (1) | ATE507226T1 (https=) |
| AU (1) | AU2005230837A1 (https=) |
| BR (1) | BRPI0509468A (https=) |
| CA (1) | CA2561738A1 (https=) |
| DE (1) | DE602005027677D1 (https=) |
| IL (1) | IL178167A0 (https=) |
| MA (1) | MA28562B1 (https=) |
| NO (1) | NO20064982L (https=) |
| NZ (1) | NZ550857A (https=) |
| RU (1) | RU2375358C2 (https=) |
| WO (1) | WO2005097762A2 (https=) |
| ZA (1) | ZA200607851B (https=) |
Families Citing this family (13)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AU2005230838A1 (en) * | 2004-04-01 | 2005-10-20 | Aventis Pharmaceuticals Inc. | 1,3,4-oxadiazol-2-ones as PPAR delta |
| DE602005024384D1 (de) | 2004-05-05 | 2010-12-09 | High Point Pharmaceuticals Llc | Neue verbindungen, ihre herstellung und verwendung |
| US8053598B2 (en) | 2004-05-05 | 2011-11-08 | High Point Pharmaceuticals, Llc | Compounds, their preparation and use |
| ES2372617T3 (es) | 2005-06-30 | 2012-01-24 | High Point Pharmaceuticals, Llc | Ácidos fenoxiacéticos como activadores de ppar-delta. |
| AU2006299092A1 (en) * | 2005-09-29 | 2007-04-12 | Sanofi-Aventis | Phenyl-(1,2,4)-oxadiazol-5-one derivatives with phenyl group, processes for their preparation and their use as pharmaceuticals |
| JP2009509988A (ja) | 2005-09-29 | 2009-03-12 | サノフィ−アベンティス | フェニル−及びピリジニル−１，２，４−オキサジアゾロン誘導体、その製造方法、及び医薬品としてのその使用 |
| CN103224477A (zh) | 2005-12-22 | 2013-07-31 | 高点制药有限责任公司 | 作为PPAR-δ活化剂的苯氧基乙酸 |
| US7943612B2 (en) | 2006-03-09 | 2011-05-17 | High Point Pharmaceuticals, Llc | Compounds that modulate PPAR activity, their preparation and use |
| US20080004281A1 (en) * | 2006-06-28 | 2008-01-03 | Kalypsys, Inc. | Methods for the modulation of crp by the selective modulation of ppar delta |
| US20120020931A1 (en) * | 2010-06-02 | 2012-01-26 | Rutgers, The State University Of New Jersey | Therapeutic encapsulated embryonic stem cells and mesenchymal stromal cells |
| EP3756661A1 (en) | 2013-09-09 | 2020-12-30 | vTv Therapeutics LLC | Use of a ppar-delta agonist for treating muscle atrophy |
| WO2021092279A1 (en) * | 2019-11-06 | 2021-05-14 | Board Of Regents, The University Of Texas System | Methods for the treatment of dysmyelinating/demyelinating diseases |
| WO2023147309A1 (en) | 2022-01-25 | 2023-08-03 | Reneo Pharmaceuticals, Inc. | Use of ppar-delta agonists in the treatment of disease |
Family Cites Families (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4895953A (en) * | 1987-09-30 | 1990-01-23 | American Home Products Corporation | 2-Aryl substituted heterocyclic compounds as antiallergic and antiinflammatory agents |
| US5103014A (en) * | 1987-09-30 | 1992-04-07 | American Home Products Corporation | Certain 3,3'-[[[(2-phenyl-4-thiazolyl)methoxy]phenyl]methylene]dithiobis-propanoic acid derivatives |
| US4826990A (en) * | 1987-09-30 | 1989-05-02 | American Home Products Corporation | 2-aryl substituted heterocyclic compounds as antiallergic and antiinflammatory agents |
| US5641796A (en) * | 1994-11-01 | 1997-06-24 | Eli Lilly And Company | Oral hypoglycemic agents |
| ES2277842T3 (es) * | 1999-06-18 | 2007-08-01 | MERCK & CO., INC. | Derivados de ariltiazolidindiona y de ariloxazolidindiona. |
| GB9914977D0 (en) * | 1999-06-25 | 1999-08-25 | Glaxo Group Ltd | Chemical compounds |
| US6506781B1 (en) * | 1999-09-08 | 2003-01-14 | Smithkline Beecham Corporation | Oxazole PPAR antagonist |
| JP4145230B2 (ja) * | 2002-11-01 | 2008-09-03 | 武田薬品工業株式会社 | 神経障害の予防・治療剤 |
| TW200505441A (en) * | 2003-03-24 | 2005-02-16 | Hoffmann La Roche | Non-nucleoside reverse transcriptase inhibitorsⅠ |
| AU2005230838A1 (en) * | 2004-04-01 | 2005-10-20 | Aventis Pharmaceuticals Inc. | 1,3,4-oxadiazol-2-ones as PPAR delta |
-
2005
- 2005-03-30 NZ NZ550857A patent/NZ550857A/en unknown
- 2005-03-30 CN CN200580010054.5A patent/CN100516065C/zh not_active Expired - Fee Related
- 2005-03-30 JP JP2007506540A patent/JP4813460B2/ja not_active Expired - Fee Related
- 2005-03-30 WO PCT/US2005/010854 patent/WO2005097762A2/en not_active Ceased
- 2005-03-30 AT AT05766888T patent/ATE507226T1/de not_active IP Right Cessation
- 2005-03-30 BR BRPI0509468-2A patent/BRPI0509468A/pt not_active IP Right Cessation
- 2005-03-30 DE DE602005027677T patent/DE602005027677D1/de not_active Expired - Lifetime
- 2005-03-30 RU RU2006138485/04A patent/RU2375358C2/ru not_active IP Right Cessation
- 2005-03-30 EP EP05766888A patent/EP1735303B1/en not_active Expired - Lifetime
- 2005-03-30 KR KR1020067020431A patent/KR20060135854A/ko not_active Ceased
- 2005-03-30 AU AU2005230837A patent/AU2005230837A1/en not_active Abandoned
- 2005-03-30 CA CA002561738A patent/CA2561738A1/en not_active Abandoned
-
2006
- 2006-09-18 IL IL178167A patent/IL178167A0/en unknown
- 2006-09-19 ZA ZA200607851A patent/ZA200607851B/en unknown
- 2006-09-26 US US11/535,227 patent/US7576109B2/en not_active Expired - Fee Related
- 2006-10-31 NO NO20064982A patent/NO20064982L/no not_active Application Discontinuation
- 2006-10-31 MA MA29428A patent/MA28562B1/fr unknown
Also Published As
| Publication number | Publication date |
|---|---|
| WO2005097762A2 (en) | 2005-10-20 |
| RU2375358C2 (ru) | 2009-12-10 |
| CN1938305A (zh) | 2007-03-28 |
| CA2561738A1 (en) | 2005-10-20 |
| JP2007531763A (ja) | 2007-11-08 |
| US20070060626A1 (en) | 2007-03-15 |
| MA28562B1 (fr) | 2007-04-03 |
| NZ550857A (en) | 2009-12-24 |
| IL178167A0 (en) | 2006-12-31 |
| RU2006138485A (ru) | 2008-05-10 |
| EP1735303A2 (en) | 2006-12-27 |
| ZA200607851B (en) | 2008-06-25 |
| US7576109B2 (en) | 2009-08-18 |
| DE602005027677D1 (de) | 2011-06-09 |
| JP4813460B2 (ja) | 2011-11-09 |
| BRPI0509468A (pt) | 2007-09-11 |
| KR20060135854A (ko) | 2006-12-29 |
| ATE507226T1 (de) | 2011-05-15 |
| CN100516065C (zh) | 2009-07-22 |
| NO20064982L (no) | 2006-10-31 |
| WO2005097762A3 (en) | 2005-12-15 |
| EP1735303B1 (en) | 2011-04-27 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| MK4 | Application lapsed section 142(2)(d) - no continuation fee paid for the application |