AU2004284884A1 - Pharmaceutical formulations for carrier-mediated transport statins and uses thereof - Google Patents
Pharmaceutical formulations for carrier-mediated transport statins and uses thereof Download PDFInfo
- Publication number
- AU2004284884A1 AU2004284884A1 AU2004284884A AU2004284884A AU2004284884A1 AU 2004284884 A1 AU2004284884 A1 AU 2004284884A1 AU 2004284884 A AU2004284884 A AU 2004284884A AU 2004284884 A AU2004284884 A AU 2004284884A AU 2004284884 A1 AU2004284884 A1 AU 2004284884A1
- Authority
- AU
- Australia
- Prior art keywords
- carrier
- mediated transport
- formulation
- statin
- transport statin
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
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Classifications
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- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D207/30—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members
- C07D207/34—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Epidemiology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Organic Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Diabetes (AREA)
- Urology & Nephrology (AREA)
- Vascular Medicine (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US51677003P | 2003-11-04 | 2003-11-04 | |
| US60/516,770 | 2003-11-04 | ||
| US10/967,167 US8987322B2 (en) | 2003-11-04 | 2004-10-19 | Pharmaceutical formulations for carrier-mediated transport statins and uses thereof |
| US10/967,167 | 2004-10-19 | ||
| PCT/IB2004/003849 WO2005041939A1 (en) | 2003-11-04 | 2004-10-29 | Pharmaceutical formulations for carrier-mediated transport statins and uses thereof |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AU2004284884A1 true AU2004284884A1 (en) | 2005-05-12 |
Family
ID=34556205
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AU2004284884A Abandoned AU2004284884A1 (en) | 2003-11-04 | 2004-10-29 | Pharmaceutical formulations for carrier-mediated transport statins and uses thereof |
Country Status (9)
| Country | Link |
|---|---|
| US (2) | US8987322B2 (cg-RX-API-DMAC7.html) |
| EP (2) | EP1682095B1 (cg-RX-API-DMAC7.html) |
| JP (1) | JP2007510714A (cg-RX-API-DMAC7.html) |
| AU (1) | AU2004284884A1 (cg-RX-API-DMAC7.html) |
| CA (1) | CA2543716C (cg-RX-API-DMAC7.html) |
| ES (2) | ES2509869T3 (cg-RX-API-DMAC7.html) |
| IL (1) | IL175134A0 (cg-RX-API-DMAC7.html) |
| NO (1) | NO20062432L (cg-RX-API-DMAC7.html) |
| WO (1) | WO2005041939A1 (cg-RX-API-DMAC7.html) |
Families Citing this family (17)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US7658938B2 (en) | 1999-02-22 | 2010-02-09 | Merrion Reasearch III Limited | Solid oral dosage form containing an enhancer |
| CA2628666A1 (en) * | 2005-11-21 | 2007-05-24 | Teva Pharmaceutical Industries Ltd. | Atorvastatin formulation |
| WO2007071357A2 (en) * | 2005-12-20 | 2007-06-28 | Lek Pharmaceuticals D.D. | Pharmaceutical composition comprising (e) -7- [4- (4-fluorophenyl) -6-isopropyl-2- [methyl (methylsulfonyl) amino] pyrimidin-5 -yl- (3r, 5s) -3, 5-dihydr0xyhept-6-en0ic acid |
| WO2007103453A1 (en) * | 2006-03-06 | 2007-09-13 | Teva Pharmaceutical Industries Ltd. | Ezetimibe compositions |
| BRPI0710503A2 (pt) * | 2006-04-07 | 2011-08-16 | Merrion Res Iii Ltd | uso de uma composição farmacêutica, composição farmacêutica, e, forma de dosagem oral |
| ES2300188B1 (es) * | 2006-05-24 | 2009-05-01 | Ferrer Internacional, S.A. | Comprimido bicapa para la prevencion de los accidentes cardiovasculares. |
| WO2008154339A2 (en) * | 2007-06-08 | 2008-12-18 | Addrenex Pharmaceuticals, Inc. | Extended release formulation and method of treating adrenergic dysregulation |
| US20090082315A1 (en) * | 2007-09-05 | 2009-03-26 | Raif Tawakol | Compositions and Methods for Controlling Cholesterol Levels |
| TR200800269A2 (tr) * | 2008-01-15 | 2009-08-21 | Bi̇li̇m İlaç Sanayi̇ Ti̇caret A.Ş. | Stabil farmasötik formülasyon ve hazırlama yöntemleri |
| TWI391150B (zh) * | 2008-01-22 | 2013-04-01 | Taiwan Biotech Co Ltd | 腸溶性長效塗覆芯與藥物劑型及其製造方法 |
| WO2009095934A1 (en) * | 2008-01-30 | 2009-08-06 | Lupin Limited | Modified release formulations of hmg coa reductase inhibitors |
| US20090280169A1 (en) | 2008-05-07 | 2009-11-12 | Merrion Research Iii Limited | Compositions of peptides and processes of preparation thereof |
| TWI480286B (zh) * | 2009-02-25 | 2015-04-11 | Merrion Res Iii Ltd | 雙膦酸鹽類組合物及藥物遞送 |
| US20110182985A1 (en) * | 2010-01-28 | 2011-07-28 | Coughlan David C | Solid Pharmaceutical Composition with Enhancers and Methods of Preparing thereof |
| US9089484B2 (en) * | 2010-03-26 | 2015-07-28 | Merrion Research Iii Limited | Pharmaceutical compositions of selective factor Xa inhibitors for oral administration |
| EP2661273A4 (en) | 2011-01-07 | 2014-06-04 | Merrion Res Iii Ltd | IRON PHARMACEUTICAL COMPOSITIONS FOR ORAL ADMINISTRATION |
| JP7211704B2 (ja) | 2015-01-29 | 2023-01-24 | ノヴォ ノルディスク アー／エス | Ｇｌｐ－１アゴニスト及び腸溶コーティングを含む錠剤 |
Family Cites Families (24)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3845770A (en) | 1972-06-05 | 1974-11-05 | Alza Corp | Osmatic dispensing device for releasing beneficial agent |
| US3916899A (en) | 1973-04-25 | 1975-11-04 | Alza Corp | Osmotic dispensing device with maximum and minimum sizes for the passageway |
| GB1478759A (en) | 1974-11-18 | 1977-07-06 | Alza Corp | Process for forming outlet passageways in pills using a laser |
| US4088884A (en) * | 1976-01-26 | 1978-05-09 | The United States Of America As Represented By The Secretary Of The Navy | Wide aperture optical communications detector |
| US4200098A (en) | 1978-10-23 | 1980-04-29 | Alza Corporation | Osmotic system with distribution zone for dispensing beneficial agent |
| US4557925A (en) | 1982-07-08 | 1985-12-10 | Ab Ferrosan | Membrane-coated sustained-release tablets and method |
| SE8601624D0 (sv) * | 1986-04-11 | 1986-04-11 | Haessle Ab | New pharmaceutical preparations |
| US4904474A (en) * | 1988-01-25 | 1990-02-27 | Alza Corporation | Delivery of drug to colon by oral disage form |
| CA2045428A1 (en) | 1990-06-26 | 1991-12-27 | Alfred W. Alberts | Method for enhancing the lowering of plasma cholesterol levels |
| US6764697B1 (en) * | 1991-06-27 | 2004-07-20 | Alza Corporation | System for delaying drug delivery up to seven hours |
| US5573776A (en) | 1992-12-02 | 1996-11-12 | Alza Corporation | Oral osmotic device with hydrogel driving member |
| US5916595A (en) * | 1997-12-12 | 1999-06-29 | Andrx Pharmaceutials, Inc. | HMG co-reductase inhibitor |
| CO5140079A1 (es) | 1998-10-14 | 2002-03-22 | Novartis Ag | Composicion farmaceutica de liberacion sostenida y metodo para liberar un agente farmaceuticamente activo de liberacion sostenida y metodo para liberar un agente far- maceuticamente activo |
| US6248363B1 (en) * | 1999-11-23 | 2001-06-19 | Lipocine, Inc. | Solid carriers for improved delivery of active ingredients in pharmaceutical compositions |
| JP2002538202A (ja) * | 1999-03-08 | 2002-11-12 | メルク エンド カムパニー インコーポレーテッド | ＨＭＧ−ＣｏＡレダクターゼ阻害剤のジヒドロキシオープンアシッド及びその塩 |
| US6569461B1 (en) * | 1999-03-08 | 2003-05-27 | Merck & Co., Inc. | Dihydroxy open-acid and salts of HMG-CoA reductase inhibitors |
| SI20425A (sl) * | 1999-12-10 | 2001-06-30 | LEK tovarna farmacevtskih in kemi�nih izdelkov d.d. | Priprava amorfnega atorvastatina |
| AU5340101A (en) * | 2000-04-11 | 2001-10-23 | Atherogenics Inc | Compounds and methods to increase plasma hdl cholesterol levels and improve hdl functionality |
| US20020147232A1 (en) * | 2000-05-26 | 2002-10-10 | Claus Sundgreen | Pharmaceutical compositions comprising desglymidodrine as an active drug substance |
| IL156552A0 (en) * | 2000-12-21 | 2004-01-04 | Aventis Pharma Gmbh | Diphenyl azetidinone derivatives, method for the production thereof, medicaments containing these compounds, and their use |
| FR2834212B1 (fr) * | 2001-12-27 | 2004-07-09 | Besins Int Belgique | Utilisation d'une poudre a liberation immediate dans des compositions pharmaceutiques et nutraceutiques |
| MXPA04006780A (es) | 2002-01-11 | 2005-06-08 | Athpharma Ltd | Formulaciones farmaceuticas de pravastatina y metodos para usarlas. |
| US20040132802A1 (en) | 2002-09-03 | 2004-07-08 | Jackie Butler | Pharmaceutical formulations and methods for modified release of statin drugs |
| US20040132806A1 (en) | 2002-09-03 | 2004-07-08 | Jackie Butler | Pravastatin pharmaceutical formulations and methods of their use |
-
2004
- 2004-10-19 US US10/967,167 patent/US8987322B2/en not_active Expired - Fee Related
- 2004-10-29 ES ES04791793.5T patent/ES2509869T3/es not_active Expired - Lifetime
- 2004-10-29 CA CA2543716A patent/CA2543716C/en not_active Expired - Fee Related
- 2004-10-29 EP EP04791793.5A patent/EP1682095B1/en not_active Expired - Lifetime
- 2004-10-29 JP JP2006538993A patent/JP2007510714A/ja active Pending
- 2004-10-29 EP EP10185149.1A patent/EP2319501B1/en not_active Expired - Lifetime
- 2004-10-29 AU AU2004284884A patent/AU2004284884A1/en not_active Abandoned
- 2004-10-29 WO PCT/IB2004/003849 patent/WO2005041939A1/en not_active Ceased
- 2004-10-29 ES ES10185149.1T patent/ES2500924T3/es not_active Expired - Lifetime
-
2006
- 2006-04-24 IL IL175134A patent/IL175134A0/en unknown
- 2006-05-29 NO NO20062432A patent/NO20062432L/no not_active Application Discontinuation
-
2015
- 2015-02-23 US US14/629,232 patent/US20150164893A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| EP1682095A1 (en) | 2006-07-26 |
| US8987322B2 (en) | 2015-03-24 |
| CA2543716C (en) | 2016-05-31 |
| US20050119331A1 (en) | 2005-06-02 |
| JP2007510714A (ja) | 2007-04-26 |
| EP2319501B1 (en) | 2014-06-18 |
| CA2543716A1 (en) | 2005-05-12 |
| ES2509869T3 (es) | 2014-10-20 |
| WO2005041939A1 (en) | 2005-05-12 |
| US20150164893A1 (en) | 2015-06-18 |
| EP1682095B1 (en) | 2014-07-02 |
| IL175134A0 (en) | 2006-09-05 |
| EP2319501A1 (en) | 2011-05-11 |
| ES2500924T3 (es) | 2014-10-01 |
| NO20062432L (no) | 2006-08-04 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| PC1 | Assignment before grant (sect. 113) |
Owner name: CIRC PHARMA RESEARCH AND DEVELOPMENT LIMITED Free format text: FORMER APPLICANT(S): ATHPHARMA LIMITED |
|
| MK1 | Application lapsed section 142(2)(a) - no request for examination in relevant period |