AU2003282892A1 - Synergistic methods and compositions for treating cancer - Google Patents

Synergistic methods and compositions for treating cancer Download PDF

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Publication number
AU2003282892A1
AU2003282892A1 AU2003282892A AU2003282892A AU2003282892A1 AU 2003282892 A1 AU2003282892 A1 AU 2003282892A1 AU 2003282892 A AU2003282892 A AU 2003282892A AU 2003282892 A AU2003282892 A AU 2003282892A AU 2003282892 A1 AU2003282892 A1 AU 2003282892A1
Authority
AU
Australia
Prior art keywords
methyl
hydroxy
pyridin
phenyl
ethylamino
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
AU2003282892A
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English (en)
Inventor
Joan M. Carboni
Marco M. Gottardis
Warren W. Hurlburt
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Bristol Myers Squibb Co
Original Assignee
Bristol Myers Squibb Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bristol Myers Squibb Co filed Critical Bristol Myers Squibb Co
Publication of AU2003282892A1 publication Critical patent/AU2003282892A1/en
Abandoned legal-status Critical Current

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Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/513Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim having oxo groups directly attached to the heterocyclic ring, e.g. cytosine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/54Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • A61P35/02Antineoplastic agents specific for leukemia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Epidemiology (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Hematology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Oncology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Plural Heterocyclic Compounds (AREA)
AU2003282892A 2002-10-02 2003-10-01 Synergistic methods and compositions for treating cancer Abandoned AU2003282892A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US41541602P 2002-10-02 2002-10-02
US60/415,416 2002-10-02
PCT/US2003/030933 WO2004030625A2 (en) 2002-10-02 2003-10-01 Synergistic methods and compositions for treating cancer

Publications (1)

Publication Number Publication Date
AU2003282892A1 true AU2003282892A1 (en) 2004-04-23

Family

ID=32069854

Family Applications (2)

Application Number Title Priority Date Filing Date
AU2003275364A Abandoned AU2003275364A1 (en) 2002-10-02 2003-10-01 Synergistic methods and compositions for treating cancer
AU2003282892A Abandoned AU2003282892A1 (en) 2002-10-02 2003-10-01 Synergistic methods and compositions for treating cancer

Family Applications Before (1)

Application Number Title Priority Date Filing Date
AU2003275364A Abandoned AU2003275364A1 (en) 2002-10-02 2003-10-01 Synergistic methods and compositions for treating cancer

Country Status (7)

Country Link
US (2) US20040106605A1 (enExample)
EP (2) EP1551411A2 (enExample)
JP (2) JP2006503866A (enExample)
AU (2) AU2003275364A1 (enExample)
CA (2) CA2500714A1 (enExample)
TW (2) TW200501960A (enExample)
WO (2) WO2004030625A2 (enExample)

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Also Published As

Publication number Publication date
EP1551411A2 (en) 2005-07-13
CA2500729A1 (en) 2004-04-15
AU2003275364A1 (en) 2004-04-23
TW200410689A (en) 2004-07-01
JP2006503866A (ja) 2006-02-02
JP2006503867A (ja) 2006-02-02
US20040106605A1 (en) 2004-06-03
TW200501960A (en) 2005-01-16
US20040072760A1 (en) 2004-04-15
WO2004030625A2 (en) 2004-04-15
WO2004030625A3 (en) 2004-06-24
WO2004030627A3 (en) 2004-07-01
CA2500714A1 (en) 2004-04-15
WO2004030627A2 (en) 2004-04-15
EP1556051A2 (en) 2005-07-27

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