AU2002357164A1 - Pyrazolopyridazine derivatives - Google Patents

Pyrazolopyridazine derivatives

Info

Publication number
AU2002357164A1
AU2002357164A1 AU2002357164A AU2002357164A AU2002357164A1 AU 2002357164 A1 AU2002357164 A1 AU 2002357164A1 AU 2002357164 A AU2002357164 A AU 2002357164A AU 2002357164 A AU2002357164 A AU 2002357164A AU 2002357164 A1 AU2002357164 A1 AU 2002357164A1
Authority
AU
Australia
Prior art keywords
pyrazolopyridazine derivatives
pyrazolopyridazine
derivatives
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
AU2002357164A
Other languages
English (en)
Other versions
AU2002357164A8 (en
Inventor
Phillip Anthony Harris
David Kendall Jung
Michael Robert Peel
Michael John Reno
Tara Renae Rheault
Jennifer Badiang Stanford
Kirk Lawrence Stevens
James Marvin Veal
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
SmithKline Beecham Corp
Original Assignee
SmithKline Beecham Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by SmithKline Beecham Corp filed Critical SmithKline Beecham Corp
Publication of AU2002357164A8 publication Critical patent/AU2002357164A8/xx
Publication of AU2002357164A1 publication Critical patent/AU2002357164A1/en
Abandoned legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
AU2002357164A 2001-12-17 2002-12-11 Pyrazolopyridazine derivatives Abandoned AU2002357164A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US34179801P 2001-12-17 2001-12-17
US60/341,798 2001-12-17
PCT/US2002/039672 WO2003051886A1 (en) 2001-12-17 2002-12-11 Pyrazolopyridazine derivatives

Publications (2)

Publication Number Publication Date
AU2002357164A8 AU2002357164A8 (en) 2003-06-30
AU2002357164A1 true AU2002357164A1 (en) 2003-06-30

Family

ID=23339081

Family Applications (1)

Application Number Title Priority Date Filing Date
AU2002357164A Abandoned AU2002357164A1 (en) 2001-12-17 2002-12-11 Pyrazolopyridazine derivatives

Country Status (10)

Country Link
US (1) US7279473B2 (enExample)
EP (1) EP1463730B1 (enExample)
JP (1) JP2005524609A (enExample)
AR (1) AR037826A1 (enExample)
AT (1) ATE323706T1 (enExample)
AU (1) AU2002357164A1 (enExample)
DE (1) DE60210819T2 (enExample)
ES (1) ES2262899T3 (enExample)
TW (1) TW200301119A (enExample)
WO (1) WO2003051886A1 (enExample)

Families Citing this family (29)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP4291696B2 (ja) 2002-01-22 2009-07-08 ワーナー−ランバート カンパニー リミテッド ライアビリティー カンパニー ２−（ピリジン−２−イルアミノ）−ピリド［２，３−ｄ］ピリミジン−７−オン
JP2006504755A (ja) * 2002-10-15 2006-02-09 スミスクライン ビーチャム コーポレーション Ｇｓｋ−３阻害薬としてのピリダジン化合物
JP4053073B2 (ja) * 2003-07-11 2008-02-27 ワーナー−ランバート カンパニー リミテッド ライアビリティー カンパニー 選択的ｃｄｋ４阻害剤のイセチオン酸塩
DE10344223A1 (de) * 2003-09-24 2005-04-21 Merck Patent Gmbh 1,3-Benzoxazolylderivate als Kinase-Inhibitoren
WO2006050076A1 (en) 2004-10-29 2006-05-11 Janssen Pharmaceutica, N.V. Pyrimidinyl substituted fused-pyrrolyl compounds useful in treating kinase disorders
JP2009507032A (ja) 2005-09-02 2009-02-19 アボット・ラボラトリーズ 新規なイミダゾ系複素環
WO2008068171A1 (en) * 2006-12-08 2008-06-12 F. Hoffmann-La Roche Ag Substituted pyrimidines and their use as jnk modulators
KR20100098521A (ko) * 2007-12-07 2010-09-07 노파르티스 아게 피라졸 유도체 및 그의 사이클린 의존성 키나제 억제제로서의 용도
HRP20170317T1 (hr) 2008-02-15 2017-04-21 Rigel Pharmaceuticals, Inc. Spojevi pirimidin-2-amina i njihova uporaba kao inhibitora jak kinaza
TW201433568A (zh) * 2008-06-30 2014-09-01 Janssen Pharmaceutica Nv 製備經取代之嘧啶衍生物的方法
AR074870A1 (es) * 2008-12-24 2011-02-16 Palau Pharma Sa Derivados de pirazolo (1,5-a ) piridina
JP5959537B2 (ja) * 2011-01-28 2016-08-02 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング 置換ピリジニル−ピリミジン及び医薬としてのその使用
US20150203812A1 (en) * 2014-01-20 2015-07-23 Francesco Tombola Inhibitors of Voltage Gated Ion Channels
GB201605126D0 (en) * 2016-03-24 2016-05-11 Univ Nottingham Inhibitors and their uses
CN106699608A (zh) * 2016-12-26 2017-05-24 常州大学 一种含有强吸电子基团的苯胍及其盐的制备方法
GB201715342D0 (en) * 2017-09-22 2017-11-08 Univ Nottingham Compounds
US11066404B2 (en) 2018-10-11 2021-07-20 Incyte Corporation Dihydropyrido[2,3-d]pyrimidinone compounds as CDK2 inhibitors
WO2020168197A1 (en) 2019-02-15 2020-08-20 Incyte Corporation Pyrrolo[2,3-d]pyrimidinone compounds as cdk2 inhibitors
WO2020180959A1 (en) 2019-03-05 2020-09-10 Incyte Corporation Pyrazolyl pyrimidinylamine compounds as cdk2 inhibitors
WO2020205560A1 (en) 2019-03-29 2020-10-08 Incyte Corporation Sulfonylamide compounds as cdk2 inhibitors
WO2020223469A1 (en) 2019-05-01 2020-11-05 Incyte Corporation N-(1-(methylsulfonyl)piperidin-4-yl)-4,5-di hydro-1h-imidazo[4,5-h]quinazolin-8-amine derivatives and related compounds as cyclin-dependent kinase 2 (cdk2) inhibitors for treating cancer
US11447494B2 (en) 2019-05-01 2022-09-20 Incyte Corporation Tricyclic amine compounds as CDK2 inhibitors
WO2021003517A1 (en) * 2019-07-10 2021-01-14 Aucentra Therapeutics Pty Ltd Derivatives of 4-(imidazo[l,2-a]pyridin-3-yl)-n-(pyridinyl)pyrimidin- 2-amine as therapeutic agents
PH12022550361A1 (en) 2019-08-14 2023-02-27 Incyte Corp Imidazolyl pyrimidinylamine compounds as cdk2 inhibitors
PE20221905A1 (es) 2019-10-11 2022-12-23 Incyte Corp Aminas biciclicas como inhibidoras de la cdk2
US11981671B2 (en) 2021-06-21 2024-05-14 Incyte Corporation Bicyclic pyrazolyl amines as CDK2 inhibitors
US11976073B2 (en) 2021-12-10 2024-05-07 Incyte Corporation Bicyclic amines as CDK2 inhibitors
WO2023107705A1 (en) 2021-12-10 2023-06-15 Incyte Corporation Bicyclic amines as cdk12 inhibitors
CN118005948B (zh) * 2024-04-09 2024-06-28 蓝固(湖州)新能源科技有限公司 一种电解液添加剂及其制备方法和应用

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU622330B2 (en) 1989-06-23 1992-04-02 Takeda Chemical Industries Ltd. Condensed heterocyclic compounds having a nitrogen atom in the bridgehead for use as fungicides
AU734009B2 (en) * 1997-05-30 2001-05-31 Merck & Co., Inc. Novel angiogenesis inhibitors
ATE281458T1 (de) 1997-09-05 2004-11-15 Glaxo Group Ltd Pharmazeutische zusammensetzung, enthaltend 2,3- diaryl-pyrazolo(1,5-b)pyridazin derivate
WO1999032447A2 (en) 1997-12-11 1999-07-01 American Home Products Corporation 2,4,6-trisubstituted pyridines with estrogenic activity and methods for the solid phase synthesis thereof
GB9919778D0 (en) 1999-08-21 1999-10-27 Zeneca Ltd Chemical compounds
KR20010089805A (ko) 1999-11-10 2001-10-08 오르토-맥네일 파마슈티칼, 인코퍼레이티드 치환된 2-아릴-3-(헤테로아릴)-이미다조[1,2-ａ]피리미딘,및 관련 약제학적 조성물 및 방법
AU2001296871A1 (en) 2000-09-15 2002-03-26 Vertex Pharmaceuticals Incorporated Pyrazole compounds useful as protein kinase inhibitors
GB0103926D0 (en) 2001-02-17 2001-04-04 Astrazeneca Ab Chemical compounds

Also Published As

Publication number Publication date
ES2262899T3 (es) 2006-12-01
JP2005524609A (ja) 2005-08-18
EP1463730A1 (en) 2004-10-06
DE60210819T2 (de) 2007-04-19
ATE323706T1 (de) 2006-05-15
US20050090507A1 (en) 2005-04-28
AU2002357164A8 (en) 2003-06-30
WO2003051886A8 (en) 2004-08-19
TW200301119A (en) 2003-07-01
EP1463730B1 (en) 2006-04-19
DE60210819D1 (en) 2006-05-24
US7279473B2 (en) 2007-10-09
AR037826A1 (es) 2004-12-09
WO2003051886A1 (en) 2003-06-26

Similar Documents

Publication Publication Date Title
AU2002357164A1 (en) Pyrazolopyridazine derivatives
AU2002349676A1 (en) 4-oxoquinoline derivatives
AU2002313565A1 (en) Putter-heads
AU2002358715A1 (en) Tetrahydrobenzfluorene derivatives
AU2002313943A1 (en) Electromobile
AU2002226571A1 (en) Biligands
AU2001100406A4 (en) DriverSMS
AU2002313073A1 (en) Phytocystatin
AU2002257925A1 (en) Numberplates
AU2002255269B8 (en) 2-Iminopyrrolidine derivatives
AU2001100522A4 (en) e-Trans
AU2001100532A4 (en) FonePark
AU2001100338A4 (en) Sunglove
AU2001100214A4 (en) Dolly-trolley
AU2002100746A4 (en) Adrail
AU2002255269A1 (en) 2-Iminopyrrolidine derivatives
AU2002354530A1 (en) 4-phenylpyran-2-one derivatives
AU2002225034A1 (en) Rustmicin derivatives
AU2002350425A1 (en) 6-phenyldihydropyrrolopyrimidinedione derivatives
AU2002325368A1 (en) Benzoylcyclohexenone derivatives
AU2002249205A1 (en) Bis-triazinylaminobenzoxazole derivatives
HK1062431A (en) A-amino-n-hydroxy-acetamide derivatives
AU2002230196A1 (en) Dicarba-closo-dodecarborane derivatives
AU2002253080A1 (en) Biurethane derivatives
AU2002305184A1 (en) Cycloalkenylsulfonamide derivatives

Legal Events

Date Code Title Description
MK6 Application lapsed section 142(2)(f)/reg. 8.3(3) - pct applic. not entering national phase