AU2001285981A1 - Biphenyl derivatives and their use as PPAR-GAMMA receptor activators - Google Patents

Biphenyl derivatives and their use as PPAR-GAMMA receptor activators

Info

Publication number
AU2001285981A1
AU2001285981A1 AU2001285981A AU2001285981A AU2001285981A1 AU 2001285981 A1 AU2001285981 A1 AU 2001285981A1 AU 2001285981 A AU2001285981 A AU 2001285981A AU 2001285981 A AU2001285981 A AU 2001285981A AU 2001285981 A1 AU2001285981 A1 AU 2001285981A1
Authority
AU
Australia
Prior art keywords
ppar
gamma receptor
biphenyl derivatives
receptor activators
activators
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
AU2001285981A
Other versions
AU2001285981B2 (en
Inventor
Jean-Michel Bernardon
Laurence Clary
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Galderma Research and Development SNC
Original Assignee
Galderma Research and Development SNC
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from FR0010447A external-priority patent/FR2812876B1/en
Application filed by Galderma Research and Development SNC filed Critical Galderma Research and Development SNC
Publication of AU2001285981A1 publication Critical patent/AU2001285981A1/en
Assigned to GALDERMA RESEARCH & DEVELOPMENT, S.N.C. reassignment GALDERMA RESEARCH & DEVELOPMENT, S.N.C. Amend patent request/document other than specification (104) Assignors: Refer to Publication History
Application granted granted Critical
Publication of AU2001285981B2 publication Critical patent/AU2001285981B2/en
Anticipated expiration legal-status Critical
Ceased legal-status Critical Current

Links

AU2001285981A 2000-08-08 2001-08-03 Biphenyl derivatives and their use as PPAR-GAMMA receptor activators Ceased AU2001285981B2 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
FR0010447A FR2812876B1 (en) 2000-08-08 2000-08-08 NOVEL BIAROMATIC COMPOUNDS THAT ACTIVATE PPAR-GAMMA TYPE RECEPTORS AND THEIR USE IN COSMETIC OR PHARMACEUTICAL COMPOSITIONS
FR00/10447 2000-08-08
PCT/FR2001/002543 WO2002012210A1 (en) 2000-08-08 2001-08-03 Biphenyl derivatives and their use as ppar-gamma receptor activators

Publications (2)

Publication Number Publication Date
AU2001285981A1 true AU2001285981A1 (en) 2002-05-16
AU2001285981B2 AU2001285981B2 (en) 2006-01-19

Family

ID=8853412

Family Applications (2)

Application Number Title Priority Date Filing Date
AU2001285981A Ceased AU2001285981B2 (en) 2000-08-08 2001-08-03 Biphenyl derivatives and their use as PPAR-GAMMA receptor activators
AU8598101A Pending AU8598101A (en) 2000-08-08 2001-08-03 Biphenyl derivatives and their use as ppar-gamma receptor activators

Family Applications After (1)

Application Number Title Priority Date Filing Date
AU8598101A Pending AU8598101A (en) 2000-08-08 2001-08-03 Biphenyl derivatives and their use as ppar-gamma receptor activators

Country Status (20)

Country Link
US (1) US6927228B2 (en)
EP (1) EP1309575B1 (en)
JP (1) JP2004505958A (en)
KR (1) KR20030051611A (en)
CN (1) CN1468226A (en)
AR (1) AR032888A1 (en)
AT (1) ATE297386T1 (en)
AU (2) AU2001285981B2 (en)
BR (1) BR0113251A (en)
CA (1) CA2418895A1 (en)
DE (1) DE60111393T2 (en)
DK (1) DK1309575T3 (en)
ES (1) ES2245373T3 (en)
FR (1) FR2812876B1 (en)
MX (1) MXPA03001184A (en)
PL (1) PL360292A1 (en)
PT (1) PT1309575E (en)
RU (1) RU2280033C2 (en)
WO (1) WO2002012210A1 (en)
ZA (1) ZA200300667B (en)

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EP1558591B1 (en) 2002-10-07 2014-05-07 The Regents of The University of California Modulation of anxiety through blockade of anandamide hydrolysis
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US20050038098A1 (en) * 2003-04-18 2005-02-17 Catherine Tachdjian Substituted dihydronaphthalene and isochroman compounds for the treatment of metabolic disorders, cancer and other diseases
FR2856401B1 (en) * 2003-06-20 2010-02-12 Galderma Res & Dev NOVEL MODULATING COMPOUNDS OF PPARGAMMA RECEPTORS AND THEIR USE IN COSMETIC OR PHARMACEUTICAL COMPOSITIONS
EP1638964B1 (en) * 2003-06-20 2011-07-27 Galderma Research & Development Novel compounds that modulate ppar-gamma type receptors, and use thereof in cosmetic or pharmaceutical compositions
FR2869903B1 (en) * 2004-05-06 2006-06-23 Galderma Res & Dev NOVEL BI-AROMATIC RECEPTOR ACTIVATOR COMPOUNDS OF THE PPARY TYPE, PROCESS FOR THEIR PREPARATION AND THEIR USE IN COSMETIC OR PHARMACEUTICAL COMPOSITIONS
DE602005019555D1 (en) * 2004-05-06 2010-04-08 Galderma Res & Dev BIAROMATIC COMPOUNDS ACTIVATING PPAR (GAMMA) TYPE RECEPTORS, PROCESS FOR THEIR PREPARATION AND THEIR USE IN COSMETIC OR PHARMACEUTICAL COMPOSITIONS
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FR2874379B1 (en) * 2004-08-17 2006-10-27 Galderma Res & Dev NOVEL BI-AROMATIC RECEPTOR ACTIVATOR COMPOUNDS OF THE PPAR TYPE AND THEIR USE IN COSMETIC OR PHARMACEUTICAL COMPOSITIONS
FR2874378B1 (en) * 2004-08-17 2006-10-27 Galderma Res & Dev NOVEL BI-AROMATIC RECEPTOR ACTIVATOR COMPOUNDS OF THE PPAR TYPE AND THEIR USE IN COSMETIC OR PHARMACEUTICAL COMPOSITIONS
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US20070059265A1 (en) * 2005-06-28 2007-03-15 L'oreal Benzylidene-1,3-thiazolidine-2,4-dione compounds for stimulating or inducing the growth and/or for reducing the loss and/or for increasing the density of keratin fibers
FR2892412B1 (en) * 2005-10-26 2008-05-16 Galderma Res & Dev BIAROMATIC COMPOUNDS MODULATORS OF PPARS
FR2897536A1 (en) * 2006-02-17 2007-08-24 Galderma Res & Dev USE OF MURAGLITAZAR FOR THE PREPARATION OF A PHARMACEUTICAL COMPOSITION FOR THE TREATMENT OF DERMATOLOGICAL DISEASES
US7754725B2 (en) 2006-03-01 2010-07-13 Astex Therapeutics Ltd. Dihydroxyphenyl isoindolymethanones
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JP5721949B2 (en) 2006-10-12 2015-05-20 アステックス、セラピューティックス、リミテッドＡｓｔｅｘ Ｔｈｅｒａｐｅｕｔｉｃｓ Ｌｉｍｉｔｅｄ Compound drug
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FR2917084B1 (en) * 2007-06-05 2009-07-17 Galderma Res & Dev NOVEL 3-PHENYL PROPANOIC ACID DERIVATIVES OF PPAR-TYPE RECEPTORS, THEIR METHOD OF PREPARATION AND THEIR USE IN COSMETIC OR PHARMACEUTICAL COMPOSITIONS
FR2917086B1 (en) * 2007-06-05 2009-07-17 Galderma Res & Dev NOVEL 3-PHENYL ACRYLIC ACIDIC ACID DERIVATIVES OF PPAR TYPE RECEPTORS, THEIR METHOD OF PREPARATION AND THEIR USE IN COSMETIC OR PHARMACEUTICAL COMPOSITIONS.
JP2011502148A (en) * 2007-10-31 2011-01-20 メルク・シャープ・エンド・ドーム・コーポレイション P2X3 receptor antagonist for the treatment of pain
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