AU2001240674A1 - Dihydropyrimidine-5-carboxylic acid esters and use thereof as medicaments against viral diseases - Google Patents

Dihydropyrimidine-5-carboxylic acid esters and use thereof as medicaments against viral diseases

Info

Publication number
AU2001240674A1
AU2001240674A1 AU2001240674A AU4067401A AU2001240674A1 AU 2001240674 A1 AU2001240674 A1 AU 2001240674A1 AU 2001240674 A AU2001240674 A AU 2001240674A AU 4067401 A AU4067401 A AU 4067401A AU 2001240674 A1 AU2001240674 A1 AU 2001240674A1
Authority
AU
Australia
Prior art keywords
dihydropyrimidine
carboxylic acid
acid esters
viral diseases
against viral
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
AU2001240674A
Inventor
Karl Deres
Siegfried Goldmann
Erwin Graef
Thomas Kramer
Ulrich Niewohner
Arnold Paessens
Karl-Heinz Schlemmer
Jurgen Stoltefuss
Olaf Weber
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Bayer AG
Original Assignee
Bayer AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer AG filed Critical Bayer AG
Publication of AU2001240674A1 publication Critical patent/AU2001240674A1/en
Abandoned legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/04Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
AU2001240674A 2000-03-17 2001-03-05 Dihydropyrimidine-5-carboxylic acid esters and use thereof as medicaments against viral diseases Abandoned AU2001240674A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
DE10013125 2000-03-17
DE10013125A DE10013125A1 (en) 2000-03-17 2000-03-17 New 4-dihalophenyl-dihydropyrimidine-5-carboxylate ester derivatives, useful as antiviral agents having strong activity against hepatitis B virus and low cytotoxicity
PCT/EP2001/002441 WO2001068639A1 (en) 2000-03-17 2001-03-05 Dihydropyrimidine-5-carboxylic acid esters and use thereof as medicaments against viral diseases

Publications (1)

Publication Number Publication Date
AU2001240674A1 true AU2001240674A1 (en) 2001-09-24

Family

ID=7635174

Family Applications (1)

Application Number Title Priority Date Filing Date
AU2001240674A Abandoned AU2001240674A1 (en) 2000-03-17 2001-03-05 Dihydropyrimidine-5-carboxylic acid esters and use thereof as medicaments against viral diseases

Country Status (3)

Country Link
AU (1) AU2001240674A1 (en)
DE (1) DE10013125A1 (en)
WO (1) WO2001068639A1 (en)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN101225084A (en) * 2007-01-16 2008-07-23 北京摩力克科技有限公司 Dihydropyrimidine compound and use thereof in preparation of medicine treating and preventing virus diseases
WO2008154820A1 (en) * 2007-06-18 2008-12-24 Zhang, Zhongneng Carbethoxy-substituted thiazolyl dihydropyrimidines
WO2008154818A1 (en) * 2007-06-18 2008-12-24 Zhang, Zhongneng Fluorophenyl-substituted thiazolyl dihydropyrimidines
PL2159224T3 (en) 2007-06-18 2012-12-31 Ruyuan Wei Xiang Tech Co Ltd Bromo-phenyl substituted thiazolyl dihydropyrimidines
CN101328169B (en) * 2007-06-18 2011-05-25 张中能 Diethylcarbamyl-substituted thiazole dihydropyrimidine
CN101575318B (en) * 2009-06-25 2012-02-08 中国人民解放军军事医学科学院毒物药物研究所 Novel dihydropyridine compound and application thereof on preparing drugs for curing and/or preventing virus diseases
US20130267517A1 (en) 2012-03-31 2013-10-10 Hoffmann-La Roche Inc. Novel 4-methyl-dihydropyrimidines for the treatment and prophylaxis of hepatitis b virus infection
SG11201408791TA (en) 2012-08-24 2015-01-29 Sunshine Lake Pharma Co Ltd Dihydropyrimidine compounds and their application in pharmaceuticals
PE20150776A1 (en) 2012-09-10 2015-05-21 Hoffmann La Roche 6-AMINO ACID-HETEROARYLDIHYDROPYRIMIDINES FOR THE TREATMENT AND PROPHYLAXIS OF HEPATITIS B VIRUS INFECTION
US9498479B2 (en) 2013-11-19 2016-11-22 Sunshine Lake Pharma Co., Ltd. Dihydropyrimidine compounds and their application in pharmaceuticals
WO2015078392A1 (en) 2013-11-27 2015-06-04 Sunshine Lake Pharma Co., Ltd. Processes for preparing dihydropyrimidine derivatives and intermediates thereof
SG11201605896WA (en) 2014-03-28 2016-08-30 Sunshine Lake Pharma Co Ltd Dihydropyrimidine compounds and their application in pharmaceuticals
EP3253751B1 (en) 2015-02-07 2020-12-09 Sunshine Lake Pharma Co., Ltd. Complexes and salts of dihydropyrimidine derivatives and their application in pharmaceuticals

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE19817262A1 (en) * 1998-04-18 1999-10-21 Bayer Ag New dihydropyrimidine derivatives and their corresponding mesomers useful in treatment of hepatitis
DE19817264A1 (en) * 1998-04-18 1999-10-21 Bayer Ag New dihydropyrimidine derivatives and their corresponding mesomers useful as antiviral agents

Also Published As

Publication number Publication date
DE10013125A1 (en) 2001-09-20
WO2001068639A1 (en) 2001-09-20

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