ATE69219T1 - Stereospezifisches verfahren zur herstellung von indolderivaten. - Google Patents
Stereospezifisches verfahren zur herstellung von indolderivaten.Info
- Publication number
- ATE69219T1 ATE69219T1 AT87401563T AT87401563T ATE69219T1 AT E69219 T1 ATE69219 T1 AT E69219T1 AT 87401563 T AT87401563 T AT 87401563T AT 87401563 T AT87401563 T AT 87401563T AT E69219 T1 ATE69219 T1 AT E69219T1
- Authority
- AT
- Austria
- Prior art keywords
- derivatives
- compound
- indold
- production
- image
- Prior art date
Links
- 238000000034 method Methods 0.000 title abstract 2
- 230000000707 stereoselective effect Effects 0.000 title abstract 2
- IZXIZTKNFFYFOF-UHFFFAOYSA-N 2-Oxazolidone Chemical compound O=C1NCCO1 IZXIZTKNFFYFOF-UHFFFAOYSA-N 0.000 abstract 2
- 150000001875 compounds Chemical class 0.000 abstract 2
- OKTJSMMVPCPJKN-UHFFFAOYSA-N Carbon Chemical compound [C] OKTJSMMVPCPJKN-UHFFFAOYSA-N 0.000 abstract 1
- ISWSIDIOOBJBQZ-UHFFFAOYSA-N Phenol Chemical compound OC1=CC=CC=C1 ISWSIDIOOBJBQZ-UHFFFAOYSA-N 0.000 abstract 1
- 229940054051 antipsychotic indole derivative Drugs 0.000 abstract 1
- SIKJAQJRHWYJAI-UHFFFAOYSA-N benzopyrrole Natural products C1=CC=C2NC=CC2=C1 SIKJAQJRHWYJAI-UHFFFAOYSA-N 0.000 abstract 1
- 230000015572 biosynthetic process Effects 0.000 abstract 1
- 229910052799 carbon Inorganic materials 0.000 abstract 1
- 238000009833 condensation Methods 0.000 abstract 1
- 230000005494 condensation Effects 0.000 abstract 1
- PZOUSPYUWWUPPK-UHFFFAOYSA-N indole Natural products CC1=CC=CC2=C1C=CN2 PZOUSPYUWWUPPK-UHFFFAOYSA-N 0.000 abstract 1
- -1 indole compound Chemical class 0.000 abstract 1
- RKJUIXBNRJVNHR-UHFFFAOYSA-N indolenine Natural products C1=CC=C2CC=NC2=C1 RKJUIXBNRJVNHR-UHFFFAOYSA-N 0.000 abstract 1
- 150000002475 indoles Chemical class 0.000 abstract 1
- 125000002924 primary amino group Chemical class [H]N([H])* 0.000 abstract 1
- 238000003786 synthesis reaction Methods 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/04—Indoles; Hydrogenated indoles
- C07D209/10—Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
- C07D209/14—Radicals substituted by nitrogen atoms, not forming part of a nitro radical
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/04—Indoles; Hydrogenated indoles
- C07D209/10—Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
- C07D209/14—Radicals substituted by nitrogen atoms, not forming part of a nitro radical
- C07D209/16—Tryptamines
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Indole Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR8609680A FR2601008B1 (fr) | 1986-07-03 | 1986-07-03 | Procede de synthese stereospecifique de derives de l'indole |
| EP87401563A EP0251938B1 (de) | 1986-07-03 | 1987-07-03 | Stereospezifisches Verfahren zur Herstellung von Indolderivaten |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ATE69219T1 true ATE69219T1 (de) | 1991-11-15 |
Family
ID=9337041
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AT87401563T ATE69219T1 (de) | 1986-07-03 | 1987-07-03 | Stereospezifisches verfahren zur herstellung von indolderivaten. |
Country Status (11)
| Country | Link |
|---|---|
| US (1) | US4806655A (de) |
| EP (1) | EP0251938B1 (de) |
| JP (1) | JPS6322559A (de) |
| KR (1) | KR880001592A (de) |
| AT (1) | ATE69219T1 (de) |
| CA (1) | CA1298303C (de) |
| DE (1) | DE3774342D1 (de) |
| DK (1) | DK338687A (de) |
| ES (1) | ES2028890T3 (de) |
| FR (1) | FR2601008B1 (de) |
| GR (1) | GR3003562T3 (de) |
Families Citing this family (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5030640A (en) * | 1989-01-05 | 1991-07-09 | Merck & Co., Inc. | Novel β-adrenergic agonists and pharmaceutical compositions thereof |
| US5747501A (en) * | 1992-04-07 | 1998-05-05 | Pfizer, Inc. | Indole derivatives |
| TW456052B (en) * | 1995-11-14 | 2001-09-21 | Sumitomo Chemical Co | Process for producing group III-V compound semiconductor |
| JP2003055344A (ja) * | 1999-01-29 | 2003-02-26 | Dainippon Pharmaceut Co Ltd | ３，７−ジ置換インドール誘導体及びそれを含有する医薬組成物 |
| TWI316511B (en) | 2002-11-26 | 2009-11-01 | Smithkline Beecham Corp | Calcilytic compounds |
| JPWO2008120655A1 (ja) * | 2007-03-30 | 2010-07-15 | 株式会社医薬分子設計研究所 | Ｉ型１１βヒドロキシステロイド脱水素酵素阻害活性を有するオキサゾリジノン誘導体 |
| US8927190B2 (en) * | 2010-01-25 | 2015-01-06 | Rohm And Haas Electronic Materials Llc | Photoresist comprising nitrogen-containing compound |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA1116598A (en) * | 1977-07-13 | 1982-01-19 | William T. Comer | 3-indolyl-tertiary butylaminopropanols |
| US4234595A (en) * | 1977-07-13 | 1980-11-18 | Mead Johnson & Company | 3-Indolyl-tertiary butylaminopropanols |
| FR2463765A1 (fr) * | 1979-08-17 | 1981-02-27 | Clin Midy | Nouveaux derives de l'indole actifs sur le systeme cardiovasculaire |
| FR2523964B1 (fr) * | 1982-03-23 | 1985-09-27 | Sanofi Sa | Nouveaux derives de la tryptamine actifs notamment sur le systeme cardiovasculaire et procede pour leur preparation |
| NZ208337A (en) * | 1983-06-10 | 1988-10-28 | Bristol Myers Co | 2-(2-hydroxy-3-((2-(ar-hydroxy-1h-aminopropoxy-yl)ethyl benzonitriles and pharmaceutical compositions |
-
1986
- 1986-07-03 FR FR8609680A patent/FR2601008B1/fr not_active Expired - Fee Related
-
1987
- 1987-06-29 US US07/067,273 patent/US4806655A/en not_active Expired - Fee Related
- 1987-06-30 CA CA000541037A patent/CA1298303C/en not_active Expired - Fee Related
- 1987-07-01 DK DK338687A patent/DK338687A/da not_active Application Discontinuation
- 1987-07-02 JP JP62167660A patent/JPS6322559A/ja active Pending
- 1987-07-03 EP EP87401563A patent/EP0251938B1/de not_active Expired - Lifetime
- 1987-07-03 ES ES198787401563T patent/ES2028890T3/es not_active Expired - Lifetime
- 1987-07-03 AT AT87401563T patent/ATE69219T1/de not_active IP Right Cessation
- 1987-07-03 DE DE8787401563T patent/DE3774342D1/de not_active Expired - Fee Related
- 1987-07-03 KR KR1019870007112A patent/KR880001592A/ko not_active Withdrawn
-
1992
- 1992-01-13 GR GR920400019T patent/GR3003562T3/el unknown
Also Published As
| Publication number | Publication date |
|---|---|
| ES2028890T3 (es) | 1992-07-16 |
| FR2601008A1 (fr) | 1988-01-08 |
| DK338687D0 (da) | 1987-07-01 |
| EP0251938B1 (de) | 1991-11-06 |
| DE3774342D1 (de) | 1991-12-12 |
| EP0251938A1 (de) | 1988-01-07 |
| CA1298303C (en) | 1992-03-31 |
| GR3003562T3 (de) | 1993-03-16 |
| FR2601008B1 (fr) | 1990-03-30 |
| JPS6322559A (ja) | 1988-01-30 |
| US4806655A (en) | 1989-02-21 |
| KR880001592A (ko) | 1988-04-25 |
| DK338687A (da) | 1988-01-04 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| RER | Ceased as to paragraph 5 lit. 3 law introducing patent treaties |