ATE63307T1 - (3-amino-1h-pyrazol-4-yl)(aryl)ketone. - Google Patents
(3-amino-1h-pyrazol-4-yl)(aryl)ketone.Info
- Publication number
- ATE63307T1 ATE63307T1 AT84107102T AT84107102T ATE63307T1 AT E63307 T1 ATE63307 T1 AT E63307T1 AT 84107102 T AT84107102 T AT 84107102T AT 84107102 T AT84107102 T AT 84107102T AT E63307 T1 ATE63307 T1 AT E63307T1
- Authority
- AT
- Austria
- Prior art keywords
- aryl
- amino
- pyrazole
- ketones
- methanones
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D231/38—Nitrogen atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C255/00—Carboxylic acid nitriles
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/24—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
- C07D213/54—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
- C07D213/57—Nitriles
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
- C07D307/02—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings
- C07D307/34—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D307/38—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms
- C07D307/54—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D317/00—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms
- C07D317/08—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3
- C07D317/44—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 ortho- or peri-condensed with carbocyclic rings or ring systems
- C07D317/46—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 ortho- or peri-condensed with carbocyclic rings or ring systems condensed with one six-membered ring
- C07D317/48—Methylenedioxybenzenes or hydrogenated methylenedioxybenzenes, unsubstituted on the hetero ring
- C07D317/50—Methylenedioxybenzenes or hydrogenated methylenedioxybenzenes, unsubstituted on the hetero ring with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to atoms of the carbocyclic ring
- C07D317/60—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
- C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
- C07D333/06—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to the ring carbon atoms
- C07D333/24—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/06—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D409/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Neurosurgery (AREA)
- Life Sciences & Earth Sciences (AREA)
- Neurology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Anesthesiology (AREA)
- Pharmacology & Pharmacy (AREA)
- Biomedical Technology (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Cosmetics (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Pyridine Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US50731783A | 1983-06-23 | 1983-06-23 | |
| EP84107102A EP0129846B1 (de) | 1983-06-23 | 1984-06-20 | (3-Amino-1H-pyrazol-4-yl)(aryl)ketone |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ATE63307T1 true ATE63307T1 (de) | 1991-05-15 |
Family
ID=24018151
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AT84107102T ATE63307T1 (de) | 1983-06-23 | 1984-06-20 | (3-amino-1h-pyrazol-4-yl)(aryl)ketone. |
Country Status (17)
| Country | Link |
|---|---|
| EP (1) | EP0129846B1 (de) |
| JP (1) | JPS6013764A (de) |
| KR (1) | KR900001215B1 (de) |
| AT (1) | ATE63307T1 (de) |
| AU (1) | AU572157B2 (de) |
| CA (1) | CA1243029A (de) |
| DD (1) | DD223448A5 (de) |
| DE (2) | DE3484549D1 (de) |
| DK (1) | DK306884A (de) |
| ES (1) | ES533653A0 (de) |
| HK (1) | HK15292A (de) |
| HU (1) | HUT34956A (de) |
| IE (1) | IE58013B1 (de) |
| NZ (1) | NZ208555A (de) |
| PH (1) | PH21579A (de) |
| SG (1) | SG2292G (de) |
| ZA (1) | ZA844771B (de) |
Families Citing this family (16)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE3502935A1 (de) * | 1984-09-29 | 1986-04-10 | Bayer Ag, 5090 Leverkusen | 3-amino-2-benzoyl-acrylsaeurederivate und ein verfahren zu ihrer herstellung |
| JPH01211582A (ja) * | 1988-02-16 | 1989-08-24 | Tanabe Seiyaku Co Ltd | ベンゾジオキソール誘導体 |
| GB8814881D0 (en) * | 1988-06-22 | 1988-07-27 | Shell Int Research | Herbicidal acrylonitrile derivatives |
| GB8920519D0 (en) * | 1989-09-11 | 1989-10-25 | Rhone Poulenc Ltd | New compositions of matter |
| US5656573A (en) * | 1989-09-11 | 1997-08-12 | Rhone-Poulenc Agriculture Ltd. | Herbicidal 4-substituted isoxazoles |
| US5650533A (en) * | 1989-09-11 | 1997-07-22 | Rhone-Poulenc Agriculture Ltd. | Intermediates to herbicidal 4-substituted isoxazoles |
| US5747424A (en) * | 1989-09-11 | 1998-05-05 | Rhone-Poulenc Agriculture Ltd. | Herbicidal 4-substituted isoxazol |
| GB8928524D0 (en) * | 1989-12-18 | 1990-02-21 | Shell Int Research | Herbicidal acrylonitrile derivatives |
| US5059709A (en) * | 1990-11-13 | 1991-10-22 | American Cyanamid Company | Process for the synthesis of α-[(dialkylamino)substituted-methylene]-β-oxo-(substituted)propanentriles |
| US5426089A (en) * | 1990-11-21 | 1995-06-20 | Shell Research Limited | Herbicidal acrylonitrile derivatives |
| JP2549304Y2 (ja) * | 1991-05-17 | 1997-09-30 | エヌオーケー株式会社 | ゴムコーティング素材の打抜き装置 |
| US20020156114A1 (en) | 1998-05-05 | 2002-10-24 | Goldstein David Michael | Pyrazole derivatives - p38 MAP kinase inhibitors |
| US6316466B1 (en) | 1998-05-05 | 2001-11-13 | Syntex (U.S.A.) Llc | Pyrazole derivatives P-38 MAP kinase inhibitors |
| US6376527B1 (en) | 1998-05-05 | 2002-04-23 | Syntex (U.S.A.) Llc | Pyrazole derivatives-p38 map kinase inhibitors |
| GB0016787D0 (en) | 2000-07-07 | 2000-08-30 | Pfizer Ltd | Compounds useful in therapy |
| KR100612079B1 (ko) * | 2003-10-09 | 2006-08-11 | 주식회사 엘지화학 | 방사형 다분지 고분자 및 이를 이용한 다공성 막 |
Family Cites Families (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3558605A (en) * | 1969-05-14 | 1971-01-26 | Parke Davis & Co | Pyrazolo(3,4-e)(1,4)diazepin-7-(1h)-one compounds |
| AU451515B2 (en) * | 1970-07-30 | 1974-08-08 | Yoshitomi Pharmaceutical Industries, Ltd | 5 aminopyrazole derivatives |
| JPS5140365B2 (de) * | 1972-05-31 | 1976-11-02 | ||
| FR2294699A1 (fr) * | 1974-12-19 | 1976-07-16 | Bottu | Nouveaux derives du pyrazole et compositions pharmaceutiques les renfermant |
| US4178449A (en) * | 1978-04-17 | 1979-12-11 | American Cyanamid Company | Pyrazolo[1,5-a]pyrimidines and imidazo-[1,5-a]pyrimidines |
| US4281000A (en) * | 1979-07-09 | 1981-07-28 | American Cyanamid Company | Substituted pyrazolo (1,5-a)pyrimidines and their use as anxiolytic agents |
| NO822100L (no) * | 1981-06-26 | 1982-12-27 | Warner Lambert Co | Fremgangsmaate for fremstilling av terapeutisk aktive basiske acylamider av aminopyrazol-aryl-matanoner |
| IT1154024B (it) * | 1982-09-22 | 1987-01-21 | Lepetit Spa | Derivati pridinici e procedimento per la loro produzione |
| US4495195A (en) * | 1982-11-01 | 1985-01-22 | Eli Lilly And Company | Xanthine oxidase inhibiting 3(5)-phenyl-substituted-5(3)-pyrazole-carboxylic acid derivatives, compositions, and methods of use |
-
1984
- 1984-06-18 NZ NZ208555A patent/NZ208555A/en unknown
- 1984-06-20 DE DE8484107102T patent/DE3484549D1/de not_active Expired - Fee Related
- 1984-06-20 EP EP84107102A patent/EP0129846B1/de not_active Expired - Lifetime
- 1984-06-20 DE DE19843422876 patent/DE3422876A1/de not_active Ceased
- 1984-06-20 AT AT84107102T patent/ATE63307T1/de not_active IP Right Cessation
- 1984-06-21 CA CA000457123A patent/CA1243029A/en not_active Expired
- 1984-06-21 DD DD84264400A patent/DD223448A5/de unknown
- 1984-06-21 PH PH30864A patent/PH21579A/en unknown
- 1984-06-22 KR KR1019840003543A patent/KR900001215B1/ko not_active IP Right Cessation
- 1984-06-22 IE IE158184A patent/IE58013B1/en not_active IP Right Cessation
- 1984-06-22 JP JP59127649A patent/JPS6013764A/ja active Granted
- 1984-06-22 ES ES533653A patent/ES533653A0/es active Granted
- 1984-06-22 AU AU29769/84A patent/AU572157B2/en not_active Ceased
- 1984-06-22 HU HU842439A patent/HUT34956A/hu unknown
- 1984-06-22 ZA ZA844771A patent/ZA844771B/xx unknown
- 1984-06-22 DK DK306884A patent/DK306884A/da not_active Application Discontinuation
-
1992
- 1992-01-09 SG SG22/92A patent/SG2292G/en unknown
- 1992-02-27 HK HK152/92A patent/HK15292A/xx unknown
Also Published As
| Publication number | Publication date |
|---|---|
| EP0129846A2 (de) | 1985-01-02 |
| DK306884D0 (da) | 1984-06-22 |
| KR900001215B1 (ko) | 1990-02-28 |
| EP0129846A3 (en) | 1987-04-22 |
| NZ208555A (en) | 1987-06-30 |
| ES8505658A1 (es) | 1985-06-16 |
| AU2976984A (en) | 1985-01-03 |
| DK306884A (da) | 1984-12-24 |
| PH21579A (en) | 1987-12-11 |
| HUT34956A (en) | 1985-05-28 |
| DE3422876A1 (de) | 1985-01-10 |
| HK15292A (en) | 1992-03-06 |
| EP0129846B1 (de) | 1991-05-08 |
| KR850000404A (ko) | 1985-02-27 |
| IE841581L (en) | 1984-12-23 |
| ZA844771B (en) | 1985-02-27 |
| AU572157B2 (en) | 1988-05-05 |
| SG2292G (en) | 1992-03-20 |
| JPS6013764A (ja) | 1985-01-24 |
| CA1243029A (en) | 1988-10-11 |
| JPH0469155B2 (de) | 1992-11-05 |
| DD223448A5 (de) | 1985-06-12 |
| ES533653A0 (es) | 1985-06-16 |
| IE58013B1 (en) | 1993-06-16 |
| DE3484549D1 (de) | 1991-06-13 |
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| IE801395L (en) | SUBSTITUTED PYRAZOLO (1, 5-a) PYRIMIDINES, ANXIOLYTIC AGENTS |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| UEP | Publication of translation of european patent specification | ||
| REN | Ceased due to non-payment of the annual fee |