ATE556083T1 - Avermectin derivate - Google Patents
Avermectin derivateInfo
- Publication number
- ATE556083T1 ATE556083T1 AT00902857T AT00902857T ATE556083T1 AT E556083 T1 ATE556083 T1 AT E556083T1 AT 00902857 T AT00902857 T AT 00902857T AT 00902857 T AT00902857 T AT 00902857T AT E556083 T1 ATE556083 T1 AT E556083T1
- Authority
- AT
- Austria
- Prior art keywords
- line
- carbon atom
- avermectin derivatives
- double bond
- avermectin
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
- C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
- C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/70—Carbohydrates; Sugars; Derivatives thereof
- A61K31/7042—Compounds having saccharide radicals and heterocyclic rings
- A61K31/7048—Compounds having saccharide radicals and heterocyclic rings having oxygen as a ring hetero atom, e.g. leucoglucosan, hesperidin, erythromycin, nystatin, digitoxin or digoxin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Molecular Biology (AREA)
- Veterinary Medicine (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- Biochemistry (AREA)
- Epidemiology (AREA)
- Genetics & Genomics (AREA)
- Biotechnology (AREA)
- Engineering & Computer Science (AREA)
- Tropical Medicine & Parasitology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Saccharide Compounds (AREA)
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP3105899 | 1999-02-09 | ||
JP24863399 | 1999-09-02 | ||
PCT/JP2000/000691 WO2000047597A1 (fr) | 1999-02-09 | 2000-02-09 | Derives de l'avermectine |
Publications (1)
Publication Number | Publication Date |
---|---|
ATE556083T1 true ATE556083T1 (de) | 2012-05-15 |
Family
ID=26369507
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AT00902857T ATE556083T1 (de) | 1999-02-09 | 2000-02-09 | Avermectin derivate |
Country Status (14)
Country | Link |
---|---|
US (1) | US6605595B1 (de) |
EP (2) | EP1160252B1 (de) |
JP (1) | JP4832645B2 (de) |
KR (1) | KR20010101819A (de) |
CN (2) | CN1202116C (de) |
AT (1) | ATE556083T1 (de) |
AU (1) | AU769612B2 (de) |
BR (1) | BR0009861A (de) |
CA (1) | CA2362253C (de) |
ES (1) | ES2387384T3 (de) |
HK (1) | HK1040083A1 (de) |
MX (1) | MXPA01007963A (de) |
NZ (1) | NZ514026A (de) |
WO (1) | WO2000047597A1 (de) |
Families Citing this family (17)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JPWO2002012261A1 (ja) * | 2000-08-09 | 2004-01-15 | 社団法人北里研究所 | エバーメクチン誘導体 |
CA2418975C (en) * | 2000-08-09 | 2012-01-17 | Satoshi Omura | Avermectin derivatives |
CR6574A (es) | 2001-02-27 | 2004-10-28 | Syngenta Participations Ag | Sales de avermectinas substituidas en la posicion 4 con propiedades plaguicidas |
EG23124A (en) | 2001-02-27 | 2004-04-28 | Syngenta Participations Ag | Avermectins substituted in the 4-position having pesticidal properties |
AR036486A1 (es) | 2001-08-28 | 2004-09-15 | Syngenta Participations Ag | Derivados 4"-desoxi-4"-(s)-amino avermectina, composicion plaguicida, procedimiento para la preparacion de esa composicion, metodo para controlar plagas, y uso de estos derivados para preparar una composicion |
MXPA04003854A (es) * | 2001-10-25 | 2005-02-17 | Sankyo Lifetech Company Ltd | Composicion antihelmintica. |
TW200407330A (en) | 2002-05-07 | 2004-05-16 | Syngenta Participations Ag | 4"-Deoxy-4"-(S)-amido avermectin derivatives |
GB0302308D0 (en) | 2003-01-31 | 2003-03-05 | Syngenta Participations Ag | Avermectin and avermectin monosaccharide derivatives substituted in the 4"- or 4'-position having pesticidal properties |
GB0302309D0 (en) * | 2003-01-31 | 2003-03-05 | Syngenta Participations Ag | Avermectin monosaccharide derivatives substituted in the 4 -position having pesticidal properties |
GB0302310D0 (en) | 2003-01-31 | 2003-03-05 | Syngenta Participations Ag | Avermectin- and avermectin monosaccharide derivatives substituted in the 4"- or 4' - positionhaving pesticidal properties |
GB0302547D0 (en) * | 2003-02-04 | 2003-03-12 | Syngenta Participations Ag | Avermectins and avermectin monosaccharide substituted in the 4'- and 4" position having pesticidal properties |
US7396819B2 (en) * | 2003-08-08 | 2008-07-08 | Virbac Corporation | Anthelmintic formulations |
GB0320176D0 (en) | 2003-08-28 | 2003-10-01 | Syngenta Participations Ag | Avermectins and avermectin monosaccharides substitued in the 4'-and 4"-positionhaving pesticidal properties |
US7582612B2 (en) * | 2004-03-12 | 2009-09-01 | Hartz Mountain Corporation | Multi-action anthelmintic formulations |
CN103360444B (zh) | 2012-04-03 | 2016-05-11 | 浙江海正药业股份有限公司 | 抗寄生虫药赛拉菌素的合成新工艺 |
CN104231022B (zh) * | 2013-06-14 | 2018-10-09 | 南开大学 | 一种大环内酯类化合物的制备及应用 |
CN103421065B (zh) * | 2013-07-03 | 2016-05-18 | 大庆志飞生物化工有限公司 | 一类新型阿维菌素衍生物及其制备方法 |
Family Cites Families (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4427663A (en) | 1982-03-16 | 1984-01-24 | Merck & Co., Inc. | 4"-Keto-and 4"-amino-4"-deoxy avermectin compounds and substituted amino derivatives thereof |
US4833168A (en) * | 1986-10-03 | 1989-05-23 | Merck & Co., Inc. | Avermectin reformatsky adducts |
US4895837A (en) * | 1988-01-29 | 1990-01-23 | Merck & Co., Inc. | Avermectin derivatives |
US4906619A (en) * | 1988-07-22 | 1990-03-06 | Merck & Co., Inc. | Alkyl avermectin derivatives |
US5030622A (en) * | 1989-06-02 | 1991-07-09 | Merck & Co., Inc. | Avermectin derivatives |
JPH0325467A (ja) | 1989-06-22 | 1991-02-04 | Konica Corp | カラー画像形成装置 |
JP2888586B2 (ja) | 1990-03-05 | 1999-05-10 | 社団法人北里研究所 | エバーメクチンの特定成分を選択生産するための微生物およびその選択的製造法 |
JPH0633273A (ja) | 1992-07-16 | 1994-02-08 | Asahi Chem Ind Co Ltd | Alcの埋込金属部材用の防錆剤 |
GB9312154D0 (en) * | 1993-06-12 | 1993-07-28 | Pfizer Ltd | Antiparasitic agents |
-
2000
- 2000-02-09 US US09/890,824 patent/US6605595B1/en not_active Expired - Lifetime
- 2000-02-09 JP JP2000598515A patent/JP4832645B2/ja not_active Expired - Lifetime
- 2000-02-09 EP EP00902857A patent/EP1160252B1/de not_active Expired - Lifetime
- 2000-02-09 ES ES00902857T patent/ES2387384T3/es not_active Expired - Lifetime
- 2000-02-09 BR BR0009861-2A patent/BR0009861A/pt not_active Application Discontinuation
- 2000-02-09 AU AU24590/00A patent/AU769612B2/en not_active Ceased
- 2000-02-09 NZ NZ514026A patent/NZ514026A/en not_active IP Right Cessation
- 2000-02-09 AT AT00902857T patent/ATE556083T1/de active
- 2000-02-09 CN CNB008060657A patent/CN1202116C/zh not_active Expired - Fee Related
- 2000-02-09 CN CNA2004100855716A patent/CN1637011A/zh active Pending
- 2000-02-09 MX MXPA01007963A patent/MXPA01007963A/es active IP Right Grant
- 2000-02-09 EP EP10010449A patent/EP2332949A1/de not_active Withdrawn
- 2000-02-09 WO PCT/JP2000/000691 patent/WO2000047597A1/ja not_active Application Discontinuation
- 2000-02-09 CA CA002362253A patent/CA2362253C/en not_active Expired - Fee Related
- 2000-02-09 KR KR1020017009984A patent/KR20010101819A/ko not_active Application Discontinuation
-
2002
- 2002-01-07 HK HK02100099.8A patent/HK1040083A1/zh unknown
Also Published As
Publication number | Publication date |
---|---|
WO2000047597A1 (fr) | 2000-08-17 |
CA2362253A1 (en) | 2000-08-17 |
AU769612B2 (en) | 2004-01-29 |
KR20010101819A (ko) | 2001-11-14 |
MXPA01007963A (es) | 2004-01-29 |
ES2387384T3 (es) | 2012-09-21 |
EP1160252A1 (de) | 2001-12-05 |
BR0009861A (pt) | 2002-01-15 |
CA2362253C (en) | 2008-09-23 |
EP1160252B1 (de) | 2012-05-02 |
NZ514026A (en) | 2001-09-28 |
CN1202116C (zh) | 2005-05-18 |
CN1637011A (zh) | 2005-07-13 |
AU2459000A (en) | 2000-08-29 |
EP2332949A1 (de) | 2011-06-15 |
HK1040083A1 (zh) | 2002-05-24 |
US6605595B1 (en) | 2003-08-12 |
JP4832645B2 (ja) | 2011-12-07 |
EP1160252A4 (de) | 2002-07-17 |
CN1346362A (zh) | 2002-04-24 |
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