ATE541835T1 - Neue inhibitoren von glutaminylcyclase - Google Patents
Neue inhibitoren von glutaminylcyclaseInfo
- Publication number
- ATE541835T1 ATE541835T1 AT05707206T AT05707206T ATE541835T1 AT E541835 T1 ATE541835 T1 AT E541835T1 AT 05707206 T AT05707206 T AT 05707206T AT 05707206 T AT05707206 T AT 05707206T AT E541835 T1 ATE541835 T1 AT E541835T1
- Authority
- AT
- Austria
- Prior art keywords
- impaired
- glutaminyl cyclase
- sleep
- regulation
- disease
- Prior art date
Links
- 102000003642 glutaminyl-peptide cyclotransferase Human genes 0.000 title abstract 2
- 108010081484 glutaminyl-peptide cyclotransferase Proteins 0.000 title abstract 2
- 239000003112 inhibitor Substances 0.000 title abstract 2
- 230000001771 impaired effect Effects 0.000 abstract 5
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 abstract 2
- 208000035475 disorder Diseases 0.000 abstract 2
- 208000007848 Alcoholism Diseases 0.000 abstract 1
- 208000024827 Alzheimer disease Diseases 0.000 abstract 1
- 208000019901 Anxiety disease Diseases 0.000 abstract 1
- 206010010904 Convulsion Diseases 0.000 abstract 1
- 206010012289 Dementia Diseases 0.000 abstract 1
- 201000010374 Down Syndrome Diseases 0.000 abstract 1
- 208000023105 Huntington disease Diseases 0.000 abstract 1
- 206010020772 Hypertension Diseases 0.000 abstract 1
- 208000018737 Parkinson disease Diseases 0.000 abstract 1
- 206010062519 Poor quality sleep Diseases 0.000 abstract 1
- 208000028017 Psychotic disease Diseases 0.000 abstract 1
- 206010037660 Pyrexia Diseases 0.000 abstract 1
- 208000007271 Substance Withdrawal Syndrome Diseases 0.000 abstract 1
- 201000007930 alcohol dependence Diseases 0.000 abstract 1
- 208000022531 anorexia Diseases 0.000 abstract 1
- 230000036506 anxiety Effects 0.000 abstract 1
- 230000037424 autonomic function Effects 0.000 abstract 1
- 210000001124 body fluid Anatomy 0.000 abstract 1
- 239000010839 body fluid Substances 0.000 abstract 1
- 208000010877 cognitive disease Diseases 0.000 abstract 1
- 206010061428 decreased appetite Diseases 0.000 abstract 1
- 230000008482 dysregulation Effects 0.000 abstract 1
- 230000037149 energy metabolism Effects 0.000 abstract 1
- 206010015037 epilepsy Diseases 0.000 abstract 1
- 230000037406 food intake Effects 0.000 abstract 1
- 235000012631 food intake Nutrition 0.000 abstract 1
- 230000003284 homeostatic effect Effects 0.000 abstract 1
- 230000003054 hormonal effect Effects 0.000 abstract 1
- 230000001537 neural effect Effects 0.000 abstract 1
- 208000015122 neurodegenerative disease Diseases 0.000 abstract 1
- 230000001717 pathogenic effect Effects 0.000 abstract 1
- 201000000980 schizophrenia Diseases 0.000 abstract 1
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (4)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US54213304P | 2004-02-05 | 2004-02-05 | |
| US10/838,993 US7371871B2 (en) | 2003-05-05 | 2004-05-05 | Inhibitors of glutaminyl cyclase |
| US63436404P | 2004-12-08 | 2004-12-08 | |
| PCT/EP2005/001153 WO2005075436A2 (en) | 2004-02-05 | 2005-02-04 | Novel inhibitors of glutaminyl cyclase |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ATE541835T1 true ATE541835T1 (de) | 2012-02-15 |
Family
ID=42121404
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AT05707206T ATE541835T1 (de) | 2004-02-05 | 2005-02-04 | Neue inhibitoren von glutaminylcyclase |
Country Status (4)
| Country | Link |
|---|---|
| AT (1) | ATE541835T1 (de) |
| DK (1) | DK1713780T3 (de) |
| EA (1) | EA013790B1 (de) |
| IL (1) | IL176765A (de) |
Family Cites Families (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS605593B2 (ja) * | 1981-03-20 | 1985-02-12 | 北興化学工業株式会社 | イミダゾ−ル誘導体および農園芸用殺菌剤 |
| AU2764797A (en) * | 1996-05-14 | 1997-12-05 | Novo Nordisk A/S | Somatostatin agonists and antagonists |
| ES2297897T3 (es) * | 1997-10-21 | 2008-05-01 | Wyeth | Compuestos farmaceuticamente activos y metodos de uso. |
| HUP0302962A2 (hu) * | 1998-06-12 | 2003-12-29 | Societe De Conseils De Recherches Et D'applications Scientifiques S.A.S. | Béta-karbolinszármazékok, ezeket a vegyületeket tartalmazó gyógyászati készítmények és a vegyületek alkalmazása |
| KR100564902B1 (ko) * | 2000-08-21 | 2006-03-30 | 주식회사 태평양 | 신규 티오우레아 유도체 및 이를 함유하는 약제학적 조성물 |
| SE0100566D0 (sv) * | 2001-02-20 | 2001-02-20 | Astrazeneca Ab | Compounds |
| ATE462432T1 (de) * | 2003-05-05 | 2010-04-15 | Probiodrug Ag | Glutaminylcyclase-hemmer |
| NZ543146A (en) * | 2003-05-05 | 2008-09-26 | Probiodrug Ag | Use of effectors of glutaminyl cyclase (QC) activity in combination with inhibitors of DP IV or DP IV-like enzymes for the treatment of conditions that can be treated by modulation of QC-and/or DPIV-activity |
-
2005
- 2005-02-04 AT AT05707206T patent/ATE541835T1/de active
- 2005-02-04 EA EA200601411A patent/EA013790B1/ru not_active IP Right Cessation
- 2005-02-04 DK DK05707206.8T patent/DK1713780T3/da active
-
2006
- 2006-07-10 IL IL176765A patent/IL176765A/en active IP Right Grant
Also Published As
| Publication number | Publication date |
|---|---|
| EA013790B1 (ru) | 2010-06-30 |
| HK1100943A1 (en) | 2007-10-05 |
| EA200601411A1 (ru) | 2007-02-27 |
| DK1713780T3 (da) | 2012-05-07 |
| IL176765A0 (en) | 2006-10-31 |
| IL176765A (en) | 2011-08-31 |
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