ATE525359T1 - Modulatoren der aktivität des glucokortikoidrezeptors von ap-1 und/oder von nf- kb und anwendung davon - Google Patents

Modulatoren der aktivität des glucokortikoidrezeptors von ap-1 und/oder von nf- kb und anwendung davon

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Publication number
ATE525359T1
ATE525359T1 AT06773159T AT06773159T ATE525359T1 AT E525359 T1 ATE525359 T1 AT E525359T1 AT 06773159 T AT06773159 T AT 06773159T AT 06773159 T AT06773159 T AT 06773159T AT E525359 T1 ATE525359 T1 AT E525359T1
Authority
AT
Austria
Prior art keywords
glucocorticoid receptor
modulators
application
receptor activity
diseases
Prior art date
Application number
AT06773159T
Other languages
English (en)
Inventor
Jingwu Duan
Zhonghui Lu
David Weinstein
Bin Jiang
Original Assignee
Bristol Myers Squibb Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bristol Myers Squibb Co filed Critical Bristol Myers Squibb Co
Application granted granted Critical
Publication of ATE525359T1 publication Critical patent/ATE525359T1/de

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    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
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AT06773159T 2005-06-14 2006-06-14 Modulatoren der aktivität des glucokortikoidrezeptors von ap-1 und/oder von nf- kb und anwendung davon ATE525359T1 (de)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US69035505P 2005-06-14 2005-06-14
US78263606P 2006-03-15 2006-03-15
US11/451,660 US7888381B2 (en) 2005-06-14 2006-06-13 Modulators of glucocorticoid receptor, AP-1, and/or NF-κB activity, and use thereof
PCT/US2006/023164 WO2006138373A2 (en) 2005-06-14 2006-06-14 MODULATORS OF GLUCOCORTICOID RECEPTOR, AP-1, AND/OR NF-kB ACTIVITY AND USE THEREOF

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ATE525359T1 true ATE525359T1 (de) 2011-10-15

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AT06773159T ATE525359T1 (de) 2005-06-14 2006-06-14 Modulatoren der aktivität des glucokortikoidrezeptors von ap-1 und/oder von nf- kb und anwendung davon

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Country Link
US (1) US7888381B2 (de)
EP (1) EP1896424B1 (de)
JP (1) JP2008546702A (de)
AT (1) ATE525359T1 (de)
WO (1) WO2006138373A2 (de)

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