ATE488514T1 - Piperidinverbindungen und anwendungen davon - Google Patents

Piperidinverbindungen und anwendungen davon

Info

Publication number
ATE488514T1
ATE488514T1 AT08762541T AT08762541T ATE488514T1 AT E488514 T1 ATE488514 T1 AT E488514T1 AT 08762541 T AT08762541 T AT 08762541T AT 08762541 T AT08762541 T AT 08762541T AT E488514 T1 ATE488514 T1 AT E488514T1
Authority
AT
Austria
Prior art keywords
piperidine compounds
piperidine
compounds
Prior art date
Application number
AT08762541T
Other languages
English (en)
Inventor
Gregory Basarab
Pamela Hill
Fei Zhou
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Application granted granted Critical
Publication of ATE488514T1 publication Critical patent/ATE488514T1/de

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Virology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
AT08762541T 2007-06-12 2008-06-11 Piperidinverbindungen und anwendungen davon ATE488514T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US94344007P 2007-06-12 2007-06-12
PCT/GB2008/050431 WO2008152418A1 (en) 2007-06-12 2008-06-11 Piperidine compounds and uses thereof

Publications (1)

Publication Number Publication Date
ATE488514T1 true ATE488514T1 (de) 2010-12-15

Family

ID=39673349

Family Applications (1)

Application Number Title Priority Date Filing Date
AT08762541T ATE488514T1 (de) 2007-06-12 2008-06-11 Piperidinverbindungen und anwendungen davon

Country Status (30)

Country Link
US (1) US20080312255A1 (de)
EP (1) EP2158199B1 (de)
JP (1) JP2010529184A (de)
KR (1) KR20100038095A (de)
CN (1) CN102648199A (de)
AR (1) AR066977A1 (de)
AT (1) ATE488514T1 (de)
AU (1) AU2008263580A1 (de)
BR (1) BRPI0812473A2 (de)
CA (1) CA2689076A1 (de)
CL (1) CL2008001740A1 (de)
CO (1) CO6311102A2 (de)
CY (1) CY1111442T1 (de)
DE (1) DE602008003575D1 (de)
DK (1) DK2158199T3 (de)
ES (1) ES2354647T3 (de)
HK (1) HK1140198A1 (de)
HR (1) HRP20110048T1 (de)
IL (1) IL202367A0 (de)
MX (1) MX2009013501A (de)
NZ (1) NZ582516A (de)
PE (1) PE20090555A1 (de)
PL (1) PL2158199T3 (de)
PT (1) PT2158199E (de)
RU (1) RU2010100352A (de)
SA (1) SA08290357B1 (de)
SI (1) SI2158199T1 (de)
TW (1) TW200906412A (de)
UY (1) UY31141A1 (de)
WO (1) WO2008152418A1 (de)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US8399489B2 (en) * 2005-02-18 2013-03-19 Astrazeneca Ab Antibacterial piperdine derivatives
US8071605B2 (en) * 2008-12-12 2011-12-06 Astrazeneca Ab Piperidine compounds for use in the treatment of bacterial infections
TW201026694A (en) * 2008-12-12 2010-07-16 Astrazeneca Ab Compound 468
WO2011024004A1 (en) 2009-08-26 2011-03-03 Astrazeneca Ab Heterocyclic urea derivatives useful for treatment of bacterial infection
WO2014164195A1 (en) * 2013-03-13 2014-10-09 Avon Products, Inc Tyrosinase inhibitors
WO2014164200A1 (en) 2013-03-13 2014-10-09 Avon Products, Inc Tyrosinase inhibitors
MX2018003562A (es) 2015-09-30 2018-06-19 Daiichi Sankyo Co Ltd Derivados de hidroxialquil tiadiazol.
CA3056571C (en) 2017-03-14 2021-11-23 Daiichi Sankyo Company, Limited N-phosphonoxymethyl prodrugs of hydroxyalkyl thiadiazole derivatives
AU2018239711A1 (en) 2017-03-24 2019-11-07 Taisho Pharmaceutical Co., Ltd. 2(1h)-quinolinone derivative
EP3847172A1 (de) 2018-09-03 2021-07-14 Univerza v Ljubljani Neue klasse von dna-gyrase- und/oder topoisomerase-iv-inhibitoren mit aktivität gegen grampositive und gramnegative bakterien
CN110172435B (zh) * 2019-06-06 2020-12-29 江南大学 一种催化合成2,5-二甲基吡嗪的重组菌
EP4263503A1 (de) 2020-12-17 2023-10-25 Univerza V Ljubljani Neue n-phenylpyrrolamid-inhibitoren der dna-gyrase und topoisomerase iv mit antibakterieller wirkung
CN115466246B (zh) * 2021-06-11 2024-02-06 中国医学科学院药物研究所 吡咯酰哌啶胺类化合物及其用途

Family Cites Families (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4046775A (en) * 1973-04-11 1977-09-06 Sterling Drug Inc. 4,5-Dihalopyrrole-2-carboxamides
US3963480A (en) * 1973-04-11 1976-06-15 Sterling Drug Inc. Herbicidal pyrrole-2-carboxamides
US4791112A (en) * 1987-02-02 1988-12-13 The Boc Group, Inc. N-heterocyclic-N-(4-piperidyl)amides and pharmaceutical compositions and methods employing such compounds
US4912109A (en) * 1987-02-02 1990-03-27 Boc, Inc. N-heterocyclic-N-(4-piperidinyl) amides and pharmaceutical compositions and methods employing such compounds
US5739135A (en) * 1993-09-03 1998-04-14 Bristol-Myers Squibb Company Inhibitors of microsomal triglyceride transfer protein and method
ES2222336T3 (es) * 2000-01-18 2005-02-01 Vertex Pharma Inhibidores de girasas y sus usos.
DE60309701T2 (de) * 2002-06-13 2007-09-06 Vertex Pharmaceuticals Inc., Cambridge 2-ureido-6-heteroaryl-3h-benzoimidazol-4-carbonsäurederivate und verwandte verbindungen als gyrase und/oder topoisomerase iv inhibitoren zur behandlung von bakteriellen infektionen
TW200526626A (en) * 2003-09-13 2005-08-16 Astrazeneca Ab Chemical compounds
GB0321509D0 (en) * 2003-09-13 2003-10-15 Astrazeneca Ab Chemical compounds
US20050197336A1 (en) * 2004-03-08 2005-09-08 Miikana Therapeutics Corporation Inhibitors of histone deacetylase
US7345043B2 (en) * 2004-04-01 2008-03-18 Miikana Therapeutics Inhibitors of histone deacetylase
US8399489B2 (en) * 2005-02-18 2013-03-19 Astrazeneca Ab Antibacterial piperdine derivatives
TW200819437A (en) * 2006-08-17 2008-05-01 Astrazeneca Ab Chemical compounds

Also Published As

Publication number Publication date
DE602008003575D1 (de) 2010-12-30
MX2009013501A (es) 2010-01-18
WO2008152418A1 (en) 2008-12-18
CN102648199A (zh) 2012-08-22
US20080312255A1 (en) 2008-12-18
PL2158199T3 (pl) 2011-04-29
UY31141A1 (es) 2009-01-30
PT2158199E (pt) 2011-01-19
KR20100038095A (ko) 2010-04-12
CA2689076A1 (en) 2008-12-18
JP2010529184A (ja) 2010-08-26
SA08290357B1 (ar) 2011-06-22
CO6311102A2 (es) 2011-08-22
CL2008001740A1 (es) 2009-07-17
DK2158199T3 (da) 2011-02-07
BRPI0812473A2 (pt) 2014-12-02
IL202367A0 (en) 2010-06-30
HK1140198A1 (en) 2010-10-08
TW200906412A (en) 2009-02-16
ES2354647T3 (es) 2011-03-16
NZ582516A (en) 2012-03-30
AR066977A1 (es) 2009-09-23
CY1111442T1 (el) 2015-08-05
EP2158199A1 (de) 2010-03-03
RU2010100352A (ru) 2011-07-20
EP2158199B1 (de) 2010-11-17
AU2008263580A1 (en) 2008-12-18
PE20090555A1 (es) 2009-06-04
HRP20110048T1 (hr) 2011-03-31
SI2158199T1 (sl) 2011-02-28

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