ATE487479T1 - Radioaktiv markierte neurokinin-1-rezeptor- antagonisten - Google Patents
Radioaktiv markierte neurokinin-1-rezeptor- antagonistenInfo
- Publication number
- ATE487479T1 ATE487479T1 AT03759348T AT03759348T ATE487479T1 AT E487479 T1 ATE487479 T1 AT E487479T1 AT 03759348 T AT03759348 T AT 03759348T AT 03759348 T AT03759348 T AT 03759348T AT E487479 T1 ATE487479 T1 AT E487479T1
- Authority
- AT
- Austria
- Prior art keywords
- neurokinin
- receptor antagonists
- radioactively labeled
- radioactively
- labeled
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
- Hydrogenated Pyridines (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Peptides Or Proteins (AREA)
- Preparation Of Compounds By Using Micro-Organisms (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US41322302P | 2002-09-24 | 2002-09-24 | |
PCT/US2003/029707 WO2004029024A2 (en) | 2002-09-24 | 2003-09-19 | Radiolabeled neurokinin-1 receptor antagonists |
Publications (1)
Publication Number | Publication Date |
---|---|
ATE487479T1 true ATE487479T1 (de) | 2010-11-15 |
Family
ID=32043220
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AT03759348T ATE487479T1 (de) | 2002-09-24 | 2003-09-19 | Radioaktiv markierte neurokinin-1-rezeptor- antagonisten |
Country Status (7)
Country | Link |
---|---|
US (1) | US7354935B2 (de) |
EP (1) | EP1545525B1 (de) |
AT (1) | ATE487479T1 (de) |
CA (1) | CA2499825C (de) |
DE (1) | DE60334922D1 (de) |
ES (1) | ES2354151T3 (de) |
WO (1) | WO2004029024A2 (de) |
Families Citing this family (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
ATE549921T1 (de) * | 2005-09-29 | 2012-04-15 | Merck Sharp & Dohme | Radioaktiv markierte glycintransporter-hemmer |
EP2336105B9 (de) * | 2008-09-19 | 2014-09-17 | Takeda Pharmaceutical Company Limited | Stickstoffhaltige heterozyklische verbindung und ihre verwendung |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US6020346A (en) | 1995-01-12 | 2000-02-01 | Glaxo Wellcome Inc. | Piperidine derivatives having tachykinin antagonist activity |
JP2002525325A (ja) * | 1998-09-29 | 2002-08-13 | メルク エンド カムパニー インコーポレーテッド | 放射標識化ニューロキニン−1受容体拮抗薬 |
GB0222426D0 (en) * | 2002-09-27 | 2002-11-06 | Imaging Res Solutions Ltd | Chemical process |
-
2003
- 2003-09-19 WO PCT/US2003/029707 patent/WO2004029024A2/en not_active Application Discontinuation
- 2003-09-19 DE DE60334922T patent/DE60334922D1/de not_active Expired - Lifetime
- 2003-09-19 AT AT03759348T patent/ATE487479T1/de not_active IP Right Cessation
- 2003-09-19 CA CA2499825A patent/CA2499825C/en not_active Expired - Fee Related
- 2003-09-19 EP EP03759348A patent/EP1545525B1/de not_active Expired - Lifetime
- 2003-09-19 US US10/528,888 patent/US7354935B2/en not_active Expired - Fee Related
- 2003-09-19 ES ES03759348T patent/ES2354151T3/es not_active Expired - Lifetime
Also Published As
Publication number | Publication date |
---|---|
EP1545525B1 (de) | 2010-11-10 |
CA2499825A1 (en) | 2004-04-08 |
EP1545525A4 (de) | 2009-07-01 |
WO2004029024A3 (en) | 2004-07-08 |
US20050214204A1 (en) | 2005-09-29 |
WO2004029024A2 (en) | 2004-04-08 |
CA2499825C (en) | 2011-11-01 |
US7354935B2 (en) | 2008-04-08 |
ES2354151T3 (es) | 2011-03-10 |
DE60334922D1 (de) | 2010-12-23 |
EP1545525A2 (de) | 2005-06-29 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
ATE439838T1 (de) | Radiomarkierte neurokinin-1 rezeptor antagonisten | |
EA200702619A1 (ru) | Антагонисты мускариновых ацетилхолиновых рецепторов | |
EA201100019A1 (ru) | Антагонисты мускариновых рецепторов ацетилхолина | |
DE60309481D1 (de) | Cyclische n-aroylamine als orexinrezeptorantagonisten | |
ATE421964T1 (de) | Radioaktiv markierte antagonisten des neuropeptid y y5-rezeptors | |
ATE430152T1 (de) | Aryl-substituierte diazabicycloalkane als nikotinische acetylcholinagonisten | |
CY1110243T1 (el) | Ανταγωνιστες npyy5 | |
DE60222396D1 (de) | N-(2-arylethyl) benzylamine als 5-ht6 rezeptor-antagoniste | |
DE60319714D1 (de) | Agonisten des cannabinoidrezeptors | |
ATE395915T1 (de) | Diaryläther als opioid-rezeptor antagonisten | |
DE60317677D1 (de) | Ox40 (=cd134) rezeptor agonisten und therapeutische verwendung | |
DK1316801T3 (da) | Sammensætninger og fremgangsmåder til detektion og behandling af sygdomme og tilstande, som er relateret til kemokinreceptorer | |
DK2064348T3 (da) | Profilering af receptorfamilie | |
DE602005022346D1 (de) | Radioaktiv markierte liganden auf chinolinbasis für die 5-ht6-rezeptorfunktionalität | |
BRPI0412537A (pt) | antagonista do receptor muscarìnico da acetilcolina | |
ATE477800T1 (de) | 2-aminocarbonlyl-chinolin-verbindungen als adenosin diphosphat plättchenrezeptor antagonisten | |
ATE356623T1 (de) | 5-ht3-rezeptorantagonisten und verwendungsverfahren | |
ATE549921T1 (de) | Radioaktiv markierte glycintransporter-hemmer | |
PE20010516A1 (es) | Peptidos ciclicos con afinidad mejorada por los receptores de somatostatina | |
DE60316411D1 (de) | Thiazolderivate als npy-rezeptorantagonisten | |
ITPD20050232A1 (it) | Apparato di fissazione esterna dell'anello pelvico | |
ATE487479T1 (de) | Radioaktiv markierte neurokinin-1-rezeptor- antagonisten | |
ATE325117T1 (de) | 3,4-dihydrochinolin-2(1h)-on verbindungen als nr2b rezeptor antagonisten | |
ATE495168T1 (de) | Heteroarylsubstituierte imidazolderivate als glutamatrezeptorantagonisten | |
DE69940923D1 (de) | Endogene, konstitutiv aktivierte g-protein gekoppelte waisenrezeptoren |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
RER | Ceased as to paragraph 5 lit. 3 law introducing patent treaties |