ATE486602T1 - Pyrrolo (3, 2, 1-ij) chinolin-4-on-derivate zur behandlung von tuberkulose - Google Patents

Pyrrolo (3, 2, 1-ij) chinolin-4-on-derivate zur behandlung von tuberkulose

Info

Publication number
ATE486602T1
ATE486602T1 AT08736082T AT08736082T ATE486602T1 AT E486602 T1 ATE486602 T1 AT E486602T1 AT 08736082 T AT08736082 T AT 08736082T AT 08736082 T AT08736082 T AT 08736082T AT E486602 T1 ATE486602 T1 AT E486602T1
Authority
AT
Austria
Prior art keywords
tuberculosis
treatment
derivatives
quinolin
pyrrolo
Prior art date
Application number
AT08736082T
Other languages
English (en)
Inventor
Lluis Ballell-Pages
David Barros-Aguirre
Julia Castro-Pichel
Modesto Jesus Remuinan-Blanco
Jose Maria Fiandor-Roman
Original Assignee
Glaxo Group Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Glaxo Group Ltd filed Critical Glaxo Group Ltd
Application granted granted Critical
Publication of ATE486602T1 publication Critical patent/ATE486602T1/de

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47—Quinolines; Isoquinolines
    • A61K31/4704—2-Quinolinones, e.g. carbostyril
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A61P31/06—Antibacterial agents for tuberculosis

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Pulmonology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
AT08736082T 2007-04-13 2008-04-10 Pyrrolo (3, 2, 1-ij) chinolin-4-on-derivate zur behandlung von tuberkulose ATE486602T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP07381033A EP1980251A1 (de) 2007-04-13 2007-04-13 Pyrrolo[3,2,1-ij]quinolin-4-on Derivate zur Behandlung der Tuberkulose
PCT/EP2008/054363 WO2008125594A1 (en) 2007-04-13 2008-04-10 Pyrrolo (3, 2, 1-ij) quinoline-4-one derivatives for treating tuberculosis

Publications (1)

Publication Number Publication Date
ATE486602T1 true ATE486602T1 (de) 2010-11-15

Family

ID=38456499

Family Applications (1)

Application Number Title Priority Date Filing Date
AT08736082T ATE486602T1 (de) 2007-04-13 2008-04-10 Pyrrolo (3, 2, 1-ij) chinolin-4-on-derivate zur behandlung von tuberkulose

Country Status (8)

Country Link
US (1) US20100048544A1 (de)
EP (2) EP1980251A1 (de)
JP (1) JP2010523622A (de)
CN (1) CN101678015A (de)
AT (1) ATE486602T1 (de)
DE (1) DE602008003322D1 (de)
ES (1) ES2353631T3 (de)
WO (1) WO2008125594A1 (de)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2006335042A1 (en) * 2005-10-21 2007-07-19 Glaxo Group Limited Compounds
GB0608263D0 (en) 2006-04-26 2006-06-07 Glaxo Group Ltd Compounds
PL2137196T3 (pl) * 2007-04-20 2011-03-31 Glaxo Group Ltd Tricykliczne związki zawierające azot jako środki przeciwbakteryjne
WO2009104147A2 (en) 2008-02-20 2009-08-27 Actelion Pharmaceuticals Ltd Azatricyclic antibiotic compounds
CN104151315B (zh) 2008-10-07 2017-01-11 埃科特莱茵药品有限公司 三环噁唑烷酮抗生素化合物
EP2417134B1 (de) 2009-04-08 2017-05-17 Idenix Pharmaceuticals LLC. Macrocyclische serinproteaseinhibitoren
CA2769652A1 (en) 2009-08-05 2011-02-10 Idenix Pharmaceuticals, Inc. Macrocyclic serine protease inhibitors useful against viral infections, particularly hcv
RU2608611C2 (ru) 2009-11-05 2017-01-23 Юниверсити Оф Нотр Дам Дю Лак СОЕДИНЕНИЯ ИМИДАЗО[1,2-а] ПИРИДИНА, ИХ СИНТЕЗ И СПОСОБЫ ПРИМЕНЕНИЯ
WO2012109398A1 (en) 2011-02-10 2012-08-16 Idenix Pharmaceuticals, Inc. Macrocyclic serine protease inhibitors, pharmaceutical compositions thereof, and their use for treating hcv infections
TW201313726A (zh) 2011-09-16 2013-04-01 Actelion Pharmaceuticals Ltd 製造合成之中間體之方法
EP2785721A1 (de) 2011-11-30 2014-10-08 Actelion Pharmaceuticals Ltd. 3,7-disubstituierte octahydro-2h-pyrido [4,3-e] [1,3] oxazin-2-on-antibiotika
EP3101012A1 (de) 2015-06-04 2016-12-07 Bayer Pharma Aktiengesellschaft Neue gadoliniumchelat-verbindung zur verwendung in der magnetresonanzbildgebung
BR112018005208B1 (pt) 2015-09-17 2023-12-12 Marvin J. Miller Compostos heterocíclicos que contêm benzilamina e composições úteis contra infecção micobacteriana
RU2755181C2 (ru) 2016-11-28 2021-09-14 Байер Фарма Акциенгезельшафт Новые хелатные соединения гадолиния с высокой релаксивностью для применения в магнитно-резонансной визуализации
SG11202104657RA (en) 2018-11-23 2021-06-29 Bayer Ag Formulation of contrast media and process of preparation thereof

Also Published As

Publication number Publication date
ES2353631T3 (es) 2011-03-03
DE602008003322D1 (de) 2010-12-16
US20100048544A1 (en) 2010-02-25
EP2136807B1 (de) 2010-11-03
CN101678015A (zh) 2010-03-24
JP2010523622A (ja) 2010-07-15
WO2008125594A1 (en) 2008-10-23
EP1980251A1 (de) 2008-10-15
EP2136807A1 (de) 2009-12-30

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