ATE411052T1 - Gonadotropin releasing hormone analoga konjugate mit steroid hormonen - Google Patents

Gonadotropin releasing hormone analoga konjugate mit steroid hormonen

Info

Publication number
ATE411052T1
ATE411052T1 AT04725716T AT04725716T ATE411052T1 AT E411052 T1 ATE411052 T1 AT E411052T1 AT 04725716 T AT04725716 T AT 04725716T AT 04725716 T AT04725716 T AT 04725716T AT E411052 T1 ATE411052 T1 AT E411052T1
Authority
AT
Austria
Prior art keywords
hormones
gonadotropin releasing
hormone
steroid
conjugates
Prior art date
Application number
AT04725716T
Other languages
English (en)
Inventor
R P Millar
Original Assignee
Medical Res Council
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Medical Res Council filed Critical Medical Res Council
Application granted granted Critical
Publication of ATE411052T1 publication Critical patent/ATE411052T1/de

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/50—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates
    • A61K47/51—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent
    • A61K47/62—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent the modifying agent being a protein, peptide or polyamino acid
    • A61K47/64—Drug-peptide, drug-protein or drug-polyamino acid conjugates, i.e. the modifying agent being a peptide, protein or polyamino acid which is covalently bonded or complexed to a therapeutically active agent
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/08—Drugs for disorders of the urinary system of the prostate
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/24—Drugs for disorders of the endocrine system of the sex hormones

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Molecular Biology (AREA)
  • Endocrinology (AREA)
  • Epidemiology (AREA)
  • Diabetes (AREA)
  • Urology & Nephrology (AREA)
  • Reproductive Health (AREA)
  • Dermatology (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
AT04725716T 2003-04-04 2004-04-05 Gonadotropin releasing hormone analoga konjugate mit steroid hormonen ATE411052T1 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GBGB0307777.3A GB0307777D0 (en) 2003-04-04 2003-04-04 Conjugate compounds

Publications (1)

Publication Number Publication Date
ATE411052T1 true ATE411052T1 (de) 2008-10-15

Family

ID=9956164

Family Applications (1)

Application Number Title Priority Date Filing Date
AT04725716T ATE411052T1 (de) 2003-04-04 2004-04-05 Gonadotropin releasing hormone analoga konjugate mit steroid hormonen

Country Status (8)

Country Link
US (1) US7700559B2 (de)
EP (1) EP1613357B1 (de)
JP (1) JP4614943B2 (de)
AT (1) ATE411052T1 (de)
DE (1) DE602004017151D1 (de)
ES (1) ES2318284T3 (de)
GB (1) GB0307777D0 (de)
WO (1) WO2004087215A1 (de)

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US9649382B2 (en) 2005-01-14 2017-05-16 Camurus Ab Topical bioadhesive formulations
CA2594710C (en) * 2005-01-14 2011-01-25 Camurus Ab Topical bioadhesive formulations
DE602005026998D1 (de) 2005-01-14 2011-04-28 Camurus Ab Somatostatin-analog-formulierungen
KR101245022B1 (ko) 2005-01-21 2013-03-19 카무러스 에이비 약제학적 지질 조성물
US8546326B2 (en) 2005-06-06 2013-10-01 Camurus Ab Glp-1 analogue formulations
EP2129402A2 (de) * 2007-02-16 2009-12-09 KTB Tumorforschungsgesellschaft mbH Prodrug mit rezeptor- und antigen-target
US20080261933A1 (en) * 2007-04-23 2008-10-23 Jens Hoffmann Combination of progesterone-receptor antagonist together with a lutein-hormone-releasing hormone agonist and antagonist for use in brca mediated diseases
GB0711656D0 (en) 2007-06-15 2007-07-25 Camurus Ab Formulations
GB0716385D0 (en) 2007-08-22 2007-10-03 Camurus Ab Formulations
ES2633453T3 (es) 2008-01-24 2017-09-21 Esperance Pharmaceuticals Constructos de fusión de dominios líticos y métodos de preparación y utilización de los mismos
GB0815435D0 (en) 2008-08-22 2008-10-01 Camurus Ab Formulations
US8828938B2 (en) * 2009-04-24 2014-09-09 Polypeptide Laboratories A/S Method for the manufacture of degarelix
US10093961B2 (en) 2009-12-22 2018-10-09 Esperance Pharmaceuticals Methods for diagnosis of and predicting treatment efficacy of hormone receptor expressing tumors, cancers and neoplasias
US20150272622A1 (en) 2011-12-22 2015-10-01 Previvo Genetics, Llc Recovery and processing of human embryos formed in vivo
US9216037B2 (en) 2013-06-21 2015-12-22 Previvo Genetics, Llc Uterine lavage for embryo retrieval
US11672843B2 (en) 2012-05-25 2023-06-13 Camurus Ab Somatostatin receptor agonist formulations
JP6559066B2 (ja) 2012-10-30 2019-08-14 エスペランス ファーマシューティカルズ， インコーポレイテッド 抗体／薬剤結合体及び使用方法
EP4223298A3 (de) 2013-03-15 2023-08-16 AbbVie Inc. Zusammensetzungen zur verwendung bei der behandlung von schweren menstruationsblutungen
EP3275888B1 (de) * 2016-07-28 2019-09-25 Council of Scientific & Industrial Research Hybrid aus progesteron und kationischem lipid als antikrebsmittel und verfahren zur synthese davon
JP7184775B2 (ja) 2016-12-14 2022-12-06 パーデュー・リサーチ・ファウンデイション 黄体化ホルモン放出ホルモン受容体（ｌｈｒｈ－ｒ）コンジュゲートおよびその使用
JP2021531236A (ja) 2018-04-19 2021-11-18 アッヴィ・インコーポレイテッド 重度の月経出血を治療する方法
CN113166086A (zh) * 2018-09-05 2021-07-23 组装生物科学股份有限公司 用于治疗hbv的环状磺酰胺化合物

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Also Published As

Publication number Publication date
US20060247177A1 (en) 2006-11-02
GB0307777D0 (en) 2003-05-07
WO2004087215A1 (en) 2004-10-14
JP4614943B2 (ja) 2011-01-19
DE602004017151D1 (en) 2008-11-27
ES2318284T3 (es) 2009-05-01
EP1613357A1 (de) 2006-01-11
JP2006522085A (ja) 2006-09-28
EP1613357B1 (de) 2008-10-15
US7700559B2 (en) 2010-04-20

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