ATE300545T1 - Substituierte indoline als 5-ht-rezeptor liganden - Google Patents
Substituierte indoline als 5-ht-rezeptor ligandenInfo
- Publication number
- ATE300545T1 ATE300545T1 AT02717304T AT02717304T ATE300545T1 AT E300545 T1 ATE300545 T1 AT E300545T1 AT 02717304 T AT02717304 T AT 02717304T AT 02717304 T AT02717304 T AT 02717304T AT E300545 T1 ATE300545 T1 AT E300545T1
- Authority
- AT
- Austria
- Prior art keywords
- receptor ligands
- substituted indolines
- indolines
- substituted
- ligands
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/06—Antimigraine agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
- A61P25/32—Alcohol-abuse
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
Landscapes
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Psychiatry (AREA)
- Addiction (AREA)
- Heart & Thoracic Surgery (AREA)
- Cardiology (AREA)
- Immunology (AREA)
- Pain & Pain Management (AREA)
- Psychology (AREA)
- Hospice & Palliative Care (AREA)
- Child & Adolescent Psychology (AREA)
- Diabetes (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Anesthesiology (AREA)
- Urology & Nephrology (AREA)
- Endocrinology (AREA)
- Reproductive Health (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US26036401P | 2001-01-08 | 2001-01-08 | |
US32650401P | 2001-10-02 | 2001-10-02 | |
PCT/US2002/000477 WO2002060903A1 (en) | 2001-01-08 | 2002-01-02 | Substituted indolines as 5-ht receptor ligands |
Publications (1)
Publication Number | Publication Date |
---|---|
ATE300545T1 true ATE300545T1 (de) | 2005-08-15 |
Family
ID=26947944
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AT02717304T ATE300545T1 (de) | 2001-01-08 | 2002-01-02 | Substituierte indoline als 5-ht-rezeptor liganden |
Country Status (10)
Country | Link |
---|---|
US (1) | US20020160999A1 (de) |
EP (1) | EP1351961B1 (de) |
JP (1) | JP2004521121A (de) |
AR (1) | AR034286A1 (de) |
AT (1) | ATE300545T1 (de) |
CA (1) | CA2429969A1 (de) |
DE (1) | DE60205213T2 (de) |
ES (1) | ES2246393T3 (de) |
PE (1) | PE20020794A1 (de) |
WO (1) | WO2002060903A1 (de) |
Families Citing this family (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US20040248880A1 (en) * | 2003-04-25 | 2004-12-09 | Jacobsen Eric Jon | 1,2,3,4,5,6-Hexahydroazepino[4,5-B]indoles containing arylsulfones at the 9-position |
EP2464227A4 (de) * | 2009-08-10 | 2013-02-20 | Galenea Corp | Verbindungen und anwendungsverfahren dafür |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2663935A1 (fr) * | 1990-06-27 | 1992-01-03 | Adir | Nouveaux 1,2,3,4,5,6-hexahydroazepino [4,5-b] indoles et 1,2,3,4-tetrahydrobethacarbolines, leurs procedes de preparation et les compositions pharmaceutiques qui les contiennent. |
AR023574A1 (es) * | 1999-04-23 | 2002-09-04 | Pharmacia & Upjohn Co Llc | Compuestos de azepinindol tetraciclico,composiciones farmaceuticas y el uso de dichos compuestos para preparar un medicamento, e intermediarios |
MY122278A (en) * | 1999-07-19 | 2006-04-29 | Upjohn Co | 1,2,3,4,5,6-hexahydroazepino[4,5-b]indoles containing arylsulfones at the 9-position |
-
2001
- 2001-12-28 US US10/033,241 patent/US20020160999A1/en not_active Abandoned
-
2002
- 2002-01-02 DE DE60205213T patent/DE60205213T2/de not_active Expired - Fee Related
- 2002-01-02 JP JP2002561471A patent/JP2004521121A/ja active Pending
- 2002-01-02 ES ES02717304T patent/ES2246393T3/es not_active Expired - Lifetime
- 2002-01-02 EP EP02717304A patent/EP1351961B1/de not_active Expired - Lifetime
- 2002-01-02 CA CA002429969A patent/CA2429969A1/en not_active Abandoned
- 2002-01-02 AT AT02717304T patent/ATE300545T1/de not_active IP Right Cessation
- 2002-01-02 WO PCT/US2002/000477 patent/WO2002060903A1/en active IP Right Grant
- 2002-01-07 PE PE2002000005A patent/PE20020794A1/es not_active Application Discontinuation
- 2002-01-08 AR ARP020100044A patent/AR034286A1/es unknown
Also Published As
Publication number | Publication date |
---|---|
AR034286A1 (es) | 2004-02-18 |
WO2002060903A1 (en) | 2002-08-08 |
EP1351961B1 (de) | 2005-07-27 |
US20020160999A1 (en) | 2002-10-31 |
EP1351961A1 (de) | 2003-10-15 |
DE60205213T2 (de) | 2006-06-01 |
DE60205213D1 (de) | 2005-09-01 |
PE20020794A1 (es) | 2002-09-13 |
JP2004521121A (ja) | 2004-07-15 |
ES2246393T3 (es) | 2006-02-16 |
CA2429969A1 (en) | 2002-08-08 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
ATE501118T1 (de) | Substituierte indole | |
ATE340792T1 (de) | Substituierte indole als alpha-1 agonisten | |
ATE392206T1 (de) | Indolderivate als beta-2 agonisten | |
NO20035359D0 (no) | Nye indolderivater med 5-HT6-reseptoraffinitet | |
DK1173440T3 (da) | Tetracycliske azepinoindolforbindelser som 5-HT receptorligander | |
ATE253067T1 (de) | Diazabicyloderivate als nikotin-acetylcholin- rezeptorliganden | |
DE602004018629D1 (de) | 3-(1-naphthyl)-2-cyanopropansäurederivate als östrogen rezeptor liganden | |
DE60331444D1 (de) | 1h-1,2,4- triazol-3- carboxamid derivate als cannabinoid-cb1 receptor liganden | |
ATE384053T1 (de) | Triazolderivate als tachykininrezeptor- antagonisten | |
DE60023167D1 (de) | Pyrazol-derivate als cannabinoidrezeptor-antagonisten | |
ATE344030T1 (de) | 4-piperazinylbenzolsulfonyl-indole mit 5-ht6 rezeptor-affinität | |
ATE197300T1 (de) | Indolderivate als 5-ht rezeptorantagoniste | |
ATE316527T1 (de) | Substituierte indolinone als tyrosinkinase inhibitoren | |
DE50014679D1 (de) | Substituierte indol-mannichbasen | |
DE602005006567D1 (de) | Indolderivate als histaminrezeptorantagonisten | |
ATE308519T1 (de) | 2,3-substituierte indolverbindungen als cox-2 inhibitoren | |
ATE292115T1 (de) | Indolderivate als cox-ii-inhibitoren | |
DE602004014772D1 (de) | Pyrrol-2,5-dithionderivate als modulatoren des liver-x-rezeptors | |
NO20015737L (no) | Indol derivater | |
ATE325123T1 (de) | Imidazoquinoline derivate als adenosine a3 rezeptor liganden | |
DE602005004515D1 (de) | (indol-3-yl)-heterozyklus-derivate als agonisten des cannabinoid-cb1-rezeptors | |
ATE196766T1 (de) | Indolin-derivate verwendbar als 5-ht-2c rezeptor- antagonisten | |
ATE433956T1 (de) | Cannabinoid-rezeptorliganden | |
PT1228041E (pt) | Derivados de indol | |
NO20052012L (no) | Indoler nyttige for behadling av androgen-reseptor relaterte sykdommer |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
RER | Ceased as to paragraph 5 lit. 3 law introducing patent treaties |