ATE232528T1 - Pyrimidinylpyrazolderivate - Google Patents
PyrimidinylpyrazolderivateInfo
- Publication number
- ATE232528T1 ATE232528T1 AT95932229T AT95932229T ATE232528T1 AT E232528 T1 ATE232528 T1 AT E232528T1 AT 95932229 T AT95932229 T AT 95932229T AT 95932229 T AT95932229 T AT 95932229T AT E232528 T1 ATE232528 T1 AT E232528T1
- Authority
- AT
- Austria
- Prior art keywords
- group
- hydrogen atom
- chem
- formula
- pyrimidinylpyrazole
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Photoreceptors In Electrophotography (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Medicines Containing Material From Animals Or Micro-Organisms (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP22942294 | 1994-09-26 | ||
| JP13501095 | 1995-06-01 | ||
| PCT/JP1995/001934 WO1996010024A1 (fr) | 1994-09-26 | 1995-09-25 | Derive pyrimidinylpyrazole |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ATE232528T1 true ATE232528T1 (de) | 2003-02-15 |
Family
ID=26468965
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AT95932229T ATE232528T1 (de) | 1994-09-26 | 1995-09-25 | Pyrimidinylpyrazolderivate |
Country Status (13)
| Country | Link |
|---|---|
| US (1) | US5852019A (forum.php) |
| EP (1) | EP0784055B1 (forum.php) |
| KR (1) | KR100388568B1 (forum.php) |
| CN (1) | CN1071754C (forum.php) |
| AT (1) | ATE232528T1 (forum.php) |
| CA (1) | CA2201110A1 (forum.php) |
| DE (2) | DE69529619D1 (forum.php) |
| DK (1) | DK0784055T3 (forum.php) |
| ES (1) | ES2192584T3 (forum.php) |
| FI (1) | FI971227A7 (forum.php) |
| NO (1) | NO313196B1 (forum.php) |
| TW (1) | TW312694B (forum.php) |
| WO (1) | WO1996010024A1 (forum.php) |
Families Citing this family (16)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AU724394B2 (en) * | 1997-01-27 | 2000-09-21 | Daiichi Pharmaceutical Co., Ltd. | Pyrazole derivatives |
| US6169086B1 (en) | 1997-01-27 | 2001-01-02 | Daiichi Pharmaceutical Co., Ltd. | Pyrazole derivatives |
| WO2000005230A1 (fr) * | 1998-07-24 | 2000-02-03 | Daiichi Pharmaceutical Co., Ltd. | Derives de pyrazole et sels correspondants |
| JP4709388B2 (ja) * | 1999-01-25 | 2011-06-22 | 全薬工業株式会社 | 複素環式化合物及びそれを有効成分とする抗腫瘍剤 |
| DK1389617T3 (da) | 2001-04-27 | 2007-05-07 | Zenyaku Kogyo Kk | Heterocyclisk forbindelse og antitumormiddel indeholdende denne som den aktive bestanddel |
| US7109204B2 (en) * | 2001-08-01 | 2006-09-19 | Merck & Co., Inc. | Tyrosine kinase inhibitors |
| AU2004218260A1 (en) * | 2003-01-28 | 2004-09-16 | Aventis Pharma S.A. | N-aryl heteroaromatic products, compositions containing same and use thereof |
| US20050130989A1 (en) * | 2003-01-28 | 2005-06-16 | Aventis Pharma S. A. | N-arylheteroaromatic products compositions containing them and use thereof |
| FR2850379B1 (fr) * | 2003-01-28 | 2006-11-17 | Aventis Pharma Sa | Produits n-aryl-heteroaromatiques, compositions les contenant et utilisation |
| WO2005028467A1 (en) * | 2003-09-15 | 2005-03-31 | Anadys Pharmaceuticals, Inc. | Antibacterial 3,5-diaminopiperidine-substitute aromatic and heteroaromatic compounds |
| DK1741714T3 (da) * | 2004-03-31 | 2013-04-15 | Zenyaku Kogyo Kk | Heterocyklisk forbindelse og middel mod ondartet turmor, der indeholder denne som aktiv ingrediens |
| WO2006095906A1 (ja) | 2005-03-11 | 2006-09-14 | Zenyaku Kogyo Kabushikikaisha | 複素環式化合物を有効成分とする免疫抑制剤及び抗腫瘍剤 |
| US20070244110A1 (en) * | 2006-04-14 | 2007-10-18 | Zenyaku Kogyo Kabushiki Kaisha | Treatment of prostate cancer, melanoma or hepatic cancer |
| CL2007002904A1 (es) | 2006-10-10 | 2008-06-06 | Amgen Inc Soc Organizada Bajo | Compuestos derivados de pirazolopirimidina; composicion farmaceutica; y uso para tratar una enfermedad seleccionada de diabetes, obesidad, asma y artritis entre otras. |
| US10287269B2 (en) * | 2015-03-26 | 2019-05-14 | Merck Sharp & Dohme Corp. | Pyrazolyl pyrimidinone compounds as PDE2 inhibitors |
| CA3038280A1 (en) | 2015-09-30 | 2017-04-06 | Max-Planck-Gesellschaft Zur Forderung Der Wissenschaften E.V. - Generalverwaltung | Heteroaryl derivatives as sepiapterin reductase inhibitors |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3778433A (en) * | 1969-04-18 | 1973-12-11 | Sumitomo Chemical Co | Process for producing benzodiazepine derivatives |
| JPS4842072A (forum.php) * | 1971-09-29 | 1973-06-19 | ||
| JPS61129129A (ja) * | 1984-11-28 | 1986-06-17 | Kureha Chem Ind Co Ltd | 抗腫瘍剤 |
| US5102893A (en) * | 1986-07-07 | 1992-04-07 | Warner-Lambert Company | Trans-6-(2-(n-heteroaryl-3,5-disubstituted)pyrazol-4-yl)-ethyl- or ethenyl)tetrahydro-4-hydroxypyran-2-one inhibitors of cholesterol biosynthesis |
-
1995
- 1995-09-19 TW TW084109880A patent/TW312694B/zh active
- 1995-09-25 US US08/821,076 patent/US5852019A/en not_active Expired - Fee Related
- 1995-09-25 CN CN95196449A patent/CN1071754C/zh not_active Expired - Fee Related
- 1995-09-25 WO PCT/JP1995/001934 patent/WO1996010024A1/ja active IP Right Grant
- 1995-09-25 KR KR1019970701964A patent/KR100388568B1/ko not_active Expired - Fee Related
- 1995-09-25 AT AT95932229T patent/ATE232528T1/de not_active IP Right Cessation
- 1995-09-25 CA CA002201110A patent/CA2201110A1/en not_active Abandoned
- 1995-09-25 EP EP95932229A patent/EP0784055B1/en not_active Expired - Lifetime
- 1995-09-25 DK DK95932229T patent/DK0784055T3/da active
- 1995-09-25 ES ES95932229T patent/ES2192584T3/es not_active Expired - Lifetime
- 1995-09-25 DE DE69529619A patent/DE69529619D1/de not_active Expired - Fee Related
- 1995-09-25 DE DE69529619T patent/DE69529619T4/de not_active Expired - Lifetime
- 1995-09-25 FI FI971227A patent/FI971227A7/fi unknown
-
1997
- 1997-03-24 NO NO19971384A patent/NO313196B1/no not_active IP Right Cessation
Also Published As
| Publication number | Publication date |
|---|---|
| DE69529619T4 (de) | 2005-01-27 |
| CA2201110A1 (en) | 1996-04-04 |
| DK0784055T3 (da) | 2003-06-02 |
| DE69529619T2 (de) | 2003-12-18 |
| WO1996010024A1 (fr) | 1996-04-04 |
| ES2192584T3 (es) | 2003-10-16 |
| KR970706275A (ko) | 1997-11-03 |
| US5852019A (en) | 1998-12-22 |
| EP0784055A4 (en) | 1998-01-07 |
| NO971384D0 (no) | 1997-03-24 |
| DE69529619D1 (en) | 2003-03-20 |
| EP0784055B1 (en) | 2003-02-12 |
| HK1001396A1 (en) | 1998-06-19 |
| FI971227A0 (fi) | 1997-03-24 |
| CN1166833A (zh) | 1997-12-03 |
| TW312694B (forum.php) | 1997-08-11 |
| CN1071754C (zh) | 2001-09-26 |
| FI971227L (fi) | 1997-05-23 |
| KR100388568B1 (ko) | 2003-10-04 |
| NO313196B1 (no) | 2002-08-26 |
| NO971384L (no) | 1997-05-23 |
| EP0784055A1 (en) | 1997-07-16 |
| FI971227A7 (fi) | 1997-05-23 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| BE2018C008I2 (forum.php) | ||
| NO992549L (no) | Sukkerforbindelse, geleringsmiddel og fremgangsmåte for fremstilling derav | |
| ES2164241T3 (es) | Compuestos pentaciclicos. | |
| DK0784055T3 (da) | Pyrimidinylpyrazolderivater | |
| DK0918776T3 (da) | Totalsyntese af antitumor acylfulvener | |
| ATE248814T1 (de) | 16-ene-vitamin d derivate | |
| ATE210642T1 (de) | 2-substituierte vitamin-d3-derivate | |
| ATE245147T1 (de) | Substituierte aminochinazolinon (thion) derivate | |
| DK0963998T3 (da) | Azasteroidforbindelse til behandling eller prævention af prostatacancer | |
| DE69828087D1 (de) | Aminderivate | |
| ATE140919T1 (de) | Indolderivate | |
| ATE189813T1 (de) | Prostaglandin-i-analoga | |
| EP1466900A4 (en) | DERIVATIVES OF VITAMIN D-DOUBLE SUBSTITUTION | |
| ES2077697T3 (es) | Derivados de 1-fenoxicarbonil-2-pirrolidinona y agentes nootropicos. |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| UEP | Publication of translation of european patent specification |
Ref document number: 0784055 Country of ref document: EP |
|
| REN | Ceased due to non-payment of the annual fee |