ATE227276T1 - Neue pyrimidinderivate - Google Patents
Neue pyrimidinderivateInfo
- Publication number
- ATE227276T1 ATE227276T1 AT98934105T AT98934105T ATE227276T1 AT E227276 T1 ATE227276 T1 AT E227276T1 AT 98934105 T AT98934105 T AT 98934105T AT 98934105 T AT98934105 T AT 98934105T AT E227276 T1 ATE227276 T1 AT E227276T1
- Authority
- AT
- Austria
- Prior art keywords
- pyrimidine derivatives
- new pyrimidine
- new
- purinoceptor
- transmembrane
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
- C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
- C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
- C07D239/56—One oxygen atom and one sulfur atom
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
- C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
- C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
- C07D239/52—Two oxygen atoms
- C07D239/54—Two oxygen atoms as doubly bound oxygen atoms or as unsubstituted hydroxy radicals
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Rheumatology (AREA)
- Pain & Pain Management (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Peptides Or Proteins (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
SE9702794A SE9702794D0 (sv) | 1997-07-24 | 1997-07-24 | New compounds |
PCT/SE1998/001391 WO1999005123A1 (en) | 1997-07-24 | 1998-07-15 | Novel pyrimidin derivatives |
Publications (1)
Publication Number | Publication Date |
---|---|
ATE227276T1 true ATE227276T1 (de) | 2002-11-15 |
Family
ID=20407823
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AT98934105T ATE227276T1 (de) | 1997-07-24 | 1998-07-15 | Neue pyrimidinderivate |
Country Status (8)
Country | Link |
---|---|
US (1) | US6200981B1 (de) |
EP (1) | EP1000038B1 (de) |
JP (1) | JP2001510833A (de) |
AT (1) | ATE227276T1 (de) |
AU (1) | AU8370498A (de) |
DE (1) | DE69809242D1 (de) |
SE (1) | SE9702794D0 (de) |
WO (1) | WO1999005123A1 (de) |
Families Citing this family (10)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
AU1356299A (en) * | 1997-11-21 | 1999-06-15 | Astra Pharmaceuticals Limited | New compounds which are p2-purinoceptor 7-transmembrane (tm) g-protein coupled receptor antagonists |
US7179481B2 (en) * | 2002-09-19 | 2007-02-20 | Kimberly-Clark Worldwide, Inc. | Vaginal health products |
US7098189B2 (en) * | 2002-12-16 | 2006-08-29 | Kimberly-Clark Worldwide, Inc. | Wound and skin care compositions |
US7056889B2 (en) | 2002-12-16 | 2006-06-06 | Kimberly-Clark, Worldwide, Inc. | Compounds that bind P2Y2 or P2Y1 receptors |
US7485666B2 (en) * | 2004-06-17 | 2009-02-03 | Kimberly-Clark Worldwide, Inc. | Vaginal health products |
MX2007014114A (es) | 2005-05-10 | 2008-03-14 | Intermune Inc | Derivados de piridona para modular el sistema de proteina cinasa activada por estres. |
RU2403250C2 (ru) | 2005-06-02 | 2010-11-10 | Ф.Хоффманн-Ля Рош Аг | Производные пиперидин-4-иламида и их применение в качестве антагонистов рецептора sst подтипа 5 |
CA3034994A1 (en) | 2008-06-03 | 2009-12-10 | Intermune, Inc. | Substituted aryl-2 pyridone compounds and use thereof for treating inflammatory and fibrotic disorders |
AR092742A1 (es) | 2012-10-02 | 2015-04-29 | Intermune Inc | Piridinonas antifibroticas |
CN106459042B (zh) | 2014-04-02 | 2019-06-28 | 英特穆恩公司 | 抗纤维化吡啶酮类 |
Family Cites Families (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
AU6930196A (en) * | 1995-09-12 | 1997-04-01 | Bayer Aktiengesellschaft | Uracil derivative |
-
1997
- 1997-07-24 SE SE9702794A patent/SE9702794D0/xx unknown
-
1998
- 1998-07-15 DE DE69809242T patent/DE69809242D1/de not_active Expired - Lifetime
- 1998-07-15 WO PCT/SE1998/001391 patent/WO1999005123A1/en active IP Right Grant
- 1998-07-15 AT AT98934105T patent/ATE227276T1/de not_active IP Right Cessation
- 1998-07-15 EP EP98934105A patent/EP1000038B1/de not_active Expired - Lifetime
- 1998-07-15 US US09/155,091 patent/US6200981B1/en not_active Expired - Fee Related
- 1998-07-15 JP JP2000504122A patent/JP2001510833A/ja active Pending
- 1998-07-15 AU AU83704/98A patent/AU8370498A/en not_active Abandoned
Also Published As
Publication number | Publication date |
---|---|
US6200981B1 (en) | 2001-03-13 |
SE9702794D0 (sv) | 1997-07-24 |
JP2001510833A (ja) | 2001-08-07 |
EP1000038B1 (de) | 2002-11-06 |
AU8370498A (en) | 1999-02-16 |
DE69809242D1 (de) | 2002-12-12 |
WO1999005123A1 (en) | 1999-02-04 |
EP1000038A1 (de) | 2000-05-17 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
RER | Ceased as to paragraph 5 lit. 3 law introducing patent treaties |