ATE211145T1 - Verfahren zur herstellung 17beta-carboxy steroidderivate und neue zwischenprodukte - Google Patents
Verfahren zur herstellung 17beta-carboxy steroidderivate und neue zwischenprodukteInfo
- Publication number
- ATE211145T1 ATE211145T1 AT95402013T AT95402013T ATE211145T1 AT E211145 T1 ATE211145 T1 AT E211145T1 AT 95402013 T AT95402013 T AT 95402013T AT 95402013 T AT95402013 T AT 95402013T AT E211145 T1 ATE211145 T1 AT E211145T1
- Authority
- AT
- Austria
- Prior art keywords
- formula
- vii
- 17beta
- producing
- epoxide
- Prior art date
Links
- 239000013067 intermediate product Substances 0.000 title 1
- 238000004519 manufacturing process Methods 0.000 title 1
- 150000002118 epoxides Chemical class 0.000 abstract 3
- -1 keto epoxide Chemical class 0.000 abstract 3
- 239000002253 acid Substances 0.000 abstract 2
- 150000002148 esters Chemical group 0.000 abstract 2
- 229930194542 Keto Natural products 0.000 abstract 1
- RTZKZFJDLAIYFH-UHFFFAOYSA-N ether Substances CCOCC RTZKZFJDLAIYFH-UHFFFAOYSA-N 0.000 abstract 1
- 125000001033 ether group Chemical group 0.000 abstract 1
- 125000001475 halogen functional group Chemical group 0.000 abstract 1
- 229910000039 hydrogen halide Inorganic materials 0.000 abstract 1
- 239000012433 hydrogen halide Substances 0.000 abstract 1
- 230000003301 hydrolyzing effect Effects 0.000 abstract 1
- 125000004356 hydroxy functional group Chemical group O* 0.000 abstract 1
- 150000002825 nitriles Chemical class 0.000 abstract 1
- 230000001681 protective effect Effects 0.000 abstract 1
- XLYOFNOQVPJJNP-UHFFFAOYSA-N water Chemical compound O XLYOFNOQVPJJNP-UHFFFAOYSA-N 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J3/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by one carbon atom
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J3/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by one carbon atom
- C07J3/005—Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by one carbon atom the carbon atom being part of a carboxylic function
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
- C07J41/0033—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005
- C07J41/0094—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005 containing nitrile radicals, including thiocyanide radicals
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Toxicology (AREA)
- Steroid Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR9410661A FR2724174B1 (fr) | 1994-09-06 | 1994-09-06 | Procede de preparation d'un derive steroide 17beta-carboxy et nouveaux intermediaires |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ATE211145T1 true ATE211145T1 (de) | 2002-01-15 |
Family
ID=9466727
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AT95402013T ATE211145T1 (de) | 1994-09-06 | 1995-09-06 | Verfahren zur herstellung 17beta-carboxy steroidderivate und neue zwischenprodukte |
Country Status (12)
| Country | Link |
|---|---|
| US (4) | US5650526A (de) |
| EP (1) | EP0702025B1 (de) |
| JP (1) | JPH0881492A (de) |
| KR (1) | KR100394203B1 (de) |
| AT (1) | ATE211145T1 (de) |
| CA (1) | CA2157550A1 (de) |
| DE (1) | DE69524696T2 (de) |
| DK (1) | DK0702025T3 (de) |
| ES (1) | ES2169747T3 (de) |
| FR (1) | FR2724174B1 (de) |
| HU (2) | HU216343B (de) |
| PT (1) | PT702025E (de) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6410760B1 (en) | 1999-10-13 | 2002-06-25 | Pharmacia & Upjohn Company | Process to prepare androst-4-en-17-carboxylic acid |
| WO2019054064A1 (ja) * | 2017-09-12 | 2019-03-21 | ダイキン工業株式会社 | ポリジフルオロアセチレン、ポリジフルオロアセチレンの製造方法、前駆体ポリマー、成形体及び粉末 |
Family Cites Families (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE42606C (de) * | O. MILSTER in Remscheid, Cronenstr | Ausrückvorrichtung des Schneckengetriebes von Lastwinden | ||
| GB929983A (en) | 1960-11-07 | 1963-06-26 | British Drug Houses Ltd | 6-formyl steroids |
| US3118882A (en) * | 1961-02-16 | 1964-01-21 | American Home Prod | Preparation of 17alpha-fluoroprogesterone and intermediates therein |
| US4179453A (en) * | 1978-04-13 | 1979-12-18 | Merck & Co., Inc. | Process for preparing 17β-carboxy-5-androsten-3-ones |
| DE3024008C2 (de) * | 1980-06-24 | 1982-04-15 | Schering Ag, 1000 Berlin Und 4619 Bergkamen | Verfahren zur Herstellung von 17α-Hydroxy-etiocarbonsäuren |
| FR2486947A1 (fr) * | 1980-07-15 | 1982-01-22 | Roussel Uclaf | Nouveaux derives steroides 20-isonitriles 17(20) insatures, leur procede de preparation et leur application a la preparation des steroides 17a-hydroxy 20-ceto |
| US4389345A (en) * | 1981-10-09 | 1983-06-21 | G.D. Searle & Co. | 3-Oxoestra-17-acetonitrile and unsaturated analogs |
| US4910226A (en) * | 1987-04-29 | 1990-03-20 | Smithkline Beckman Corporation | Steroid 5-alpha-reductase inhibitors |
| IL105050A0 (en) | 1992-03-27 | 1993-07-08 | Lilly Co Eli | Steroid derivatives |
| FR2700339B1 (fr) * | 1993-01-14 | 1995-03-03 | Roussel Uclaf | Nouveaux dérivés 17,20-époxydes du pregnane, leur préparation, leur application à la préparation de dérivés cortisoniques et intermédiaires. |
-
1994
- 1994-09-06 FR FR9410661A patent/FR2724174B1/fr not_active Expired - Fee Related
-
1995
- 1995-08-28 US US08/519,772 patent/US5650526A/en not_active Expired - Fee Related
- 1995-09-01 JP JP7246994A patent/JPH0881492A/ja not_active Abandoned
- 1995-09-05 KR KR1019950028946A patent/KR100394203B1/ko not_active Expired - Fee Related
- 1995-09-05 CA CA002157550A patent/CA2157550A1/fr not_active Abandoned
- 1995-09-05 HU HU9502601A patent/HU216343B/hu not_active IP Right Cessation
- 1995-09-05 HU HU9801519A patent/HU223949B1/hu not_active IP Right Cessation
- 1995-09-06 PT PT95402013T patent/PT702025E/pt unknown
- 1995-09-06 ES ES95402013T patent/ES2169747T3/es not_active Expired - Lifetime
- 1995-09-06 DK DK95402013T patent/DK0702025T3/da active
- 1995-09-06 DE DE69524696T patent/DE69524696T2/de not_active Expired - Fee Related
- 1995-09-06 AT AT95402013T patent/ATE211145T1/de not_active IP Right Cessation
- 1995-09-06 EP EP95402013A patent/EP0702025B1/de not_active Expired - Lifetime
-
1996
- 1996-12-02 US US08/758,951 patent/US5770748A/en not_active Expired - Fee Related
-
1997
- 1997-11-05 US US08/964,836 patent/US5945530A/en not_active Expired - Fee Related
-
1998
- 1998-08-04 US US09/130,531 patent/US5919957A/en not_active Expired - Fee Related
Also Published As
| Publication number | Publication date |
|---|---|
| US5770748A (en) | 1998-06-23 |
| PT702025E (pt) | 2002-06-28 |
| FR2724174A1 (fr) | 1996-03-08 |
| ES2169747T3 (es) | 2002-07-16 |
| HU9502601D0 (en) | 1995-10-30 |
| KR100394203B1 (ko) | 2003-10-10 |
| HU216343B (hu) | 1999-06-28 |
| JPH0881492A (ja) | 1996-03-26 |
| FR2724174B1 (fr) | 1997-01-17 |
| US5919957A (en) | 1999-07-06 |
| KR960010680A (ko) | 1996-04-20 |
| DK0702025T3 (da) | 2002-04-15 |
| DE69524696T2 (de) | 2002-08-22 |
| HUT71993A (en) | 1996-03-28 |
| CA2157550A1 (fr) | 1996-03-07 |
| EP0702025B1 (de) | 2001-12-19 |
| DE69524696D1 (de) | 2002-01-31 |
| US5945530A (en) | 1999-08-31 |
| HU223949B1 (hu) | 2005-03-29 |
| EP0702025A1 (de) | 1996-03-20 |
| US5650526A (en) | 1997-07-22 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| UEP | Publication of translation of european patent specification | ||
| REN | Ceased due to non-payment of the annual fee |