DE69524696D1 - Verfahren zur Herstellung 17beta-carboxy Steroidderivate und neue Zwischenprodukte - Google Patents

Verfahren zur Herstellung 17beta-carboxy Steroidderivate und neue Zwischenprodukte

Info

Publication number
DE69524696D1
DE69524696D1 DE69524696T DE69524696T DE69524696D1 DE 69524696 D1 DE69524696 D1 DE 69524696D1 DE 69524696 T DE69524696 T DE 69524696T DE 69524696 T DE69524696 T DE 69524696T DE 69524696 D1 DE69524696 D1 DE 69524696D1
Authority
DE
Germany
Prior art keywords
formula
vii
epoxide
17beta
preparation
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
DE69524696T
Other languages
English (en)
Other versions
DE69524696T2 (de
Inventor
Patrick Roussel
Michel Vivat
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Aventis Pharma SA
Original Assignee
Aventis Pharma SA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Aventis Pharma SA filed Critical Aventis Pharma SA
Application granted granted Critical
Publication of DE69524696D1 publication Critical patent/DE69524696D1/de
Publication of DE69524696T2 publication Critical patent/DE69524696T2/de
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J3/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by one carbon atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J3/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by one carbon atom
    • C07J3/005—Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by one carbon atom the carbon atom being part of a carboxylic function
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
    • C07J41/0033—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005
    • C07J41/0094—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005 containing nitrile radicals, including thiocyanide radicals

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Toxicology (AREA)
  • Steroid Compounds (AREA)
DE69524696T 1994-09-06 1995-09-06 Verfahren zur Herstellung 17beta-carboxy Steroidderivate und neue Zwischenprodukte Expired - Fee Related DE69524696T2 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR9410661A FR2724174B1 (fr) 1994-09-06 1994-09-06 Procede de preparation d'un derive steroide 17beta-carboxy et nouveaux intermediaires

Publications (2)

Publication Number Publication Date
DE69524696D1 true DE69524696D1 (de) 2002-01-31
DE69524696T2 DE69524696T2 (de) 2002-08-22

Family

ID=9466727

Family Applications (1)

Application Number Title Priority Date Filing Date
DE69524696T Expired - Fee Related DE69524696T2 (de) 1994-09-06 1995-09-06 Verfahren zur Herstellung 17beta-carboxy Steroidderivate und neue Zwischenprodukte

Country Status (12)

Country Link
US (4) US5650526A (de)
EP (1) EP0702025B1 (de)
JP (1) JPH0881492A (de)
KR (1) KR100394203B1 (de)
AT (1) ATE211145T1 (de)
CA (1) CA2157550A1 (de)
DE (1) DE69524696T2 (de)
DK (1) DK0702025T3 (de)
ES (1) ES2169747T3 (de)
FR (1) FR2724174B1 (de)
HU (2) HU223949B1 (de)
PT (1) PT702025E (de)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU780751B2 (en) 1999-10-13 2005-04-14 Pharmacia & Upjohn Company Process to prepare androst-4-en-17-carboxylic acid cross-reference to related applications
CN111094364B (zh) 2017-09-12 2023-04-11 大金工业株式会社 聚二氟乙炔、聚二氟乙炔的制造方法、前体聚合物、成型体和粉末

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE42606C (de) * O. MILSTER in Remscheid, Cronenstr Ausrückvorrichtung des Schneckengetriebes von Lastwinden
GB929983A (en) 1960-11-07 1963-06-26 British Drug Houses Ltd 6-formyl steroids
US3118882A (en) * 1961-02-16 1964-01-21 American Home Prod Preparation of 17alpha-fluoroprogesterone and intermediates therein
US4179453A (en) * 1978-04-13 1979-12-18 Merck & Co., Inc. Process for preparing 17β-carboxy-5-androsten-3-ones
DE3024008C2 (de) * 1980-06-24 1982-04-15 Schering Ag, 1000 Berlin Und 4619 Bergkamen Verfahren zur Herstellung von 17α-Hydroxy-etiocarbonsäuren
FR2486947A1 (fr) * 1980-07-15 1982-01-22 Roussel Uclaf Nouveaux derives steroides 20-isonitriles 17(20) insatures, leur procede de preparation et leur application a la preparation des steroides 17a-hydroxy 20-ceto
US4389345A (en) * 1981-10-09 1983-06-21 G.D. Searle & Co. 3-Oxoestra-17-acetonitrile and unsaturated analogs
US4910226A (en) * 1987-04-29 1990-03-20 Smithkline Beckman Corporation Steroid 5-alpha-reductase inhibitors
IL105050A0 (en) 1992-03-27 1993-07-08 Lilly Co Eli Steroid derivatives
FR2700339B1 (fr) * 1993-01-14 1995-03-03 Roussel Uclaf Nouveaux dérivés 17,20-époxydes du pregnane, leur préparation, leur application à la préparation de dérivés cortisoniques et intermédiaires.

Also Published As

Publication number Publication date
FR2724174B1 (fr) 1997-01-17
HU9502601D0 (en) 1995-10-30
FR2724174A1 (fr) 1996-03-08
CA2157550A1 (fr) 1996-03-07
HUT71993A (en) 1996-03-28
KR960010680A (ko) 1996-04-20
PT702025E (pt) 2002-06-28
DE69524696T2 (de) 2002-08-22
ES2169747T3 (es) 2002-07-16
HU216343B (hu) 1999-06-28
EP0702025A1 (de) 1996-03-20
HU223949B1 (hu) 2005-03-29
US5650526A (en) 1997-07-22
DK0702025T3 (da) 2002-04-15
EP0702025B1 (de) 2001-12-19
US5919957A (en) 1999-07-06
ATE211145T1 (de) 2002-01-15
US5945530A (en) 1999-08-31
KR100394203B1 (ko) 2003-10-10
JPH0881492A (ja) 1996-03-26
US5770748A (en) 1998-06-23

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Legal Events

Date Code Title Description
8339 Ceased/non-payment of the annual fee