ATE197453T1 - Imidazol-, triazol- und tetrazolderivate - Google Patents

Imidazol-, triazol- und tetrazolderivate

Info

Publication number
ATE197453T1
ATE197453T1 AT93907945T AT93907945T ATE197453T1 AT E197453 T1 ATE197453 T1 AT E197453T1 AT 93907945 T AT93907945 T AT 93907945T AT 93907945 T AT93907945 T AT 93907945T AT E197453 T1 ATE197453 T1 AT E197453T1
Authority
AT
Austria
Prior art keywords
pct
triazole
imidazole
tetrazole derivatives
receptors
Prior art date
Application number
AT93907945T
Other languages
English (en)
Inventor
Pineiro Jose Luis Castro
Victor Giulio Matassa
Original Assignee
Merck Sharp & Dohme
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck Sharp & Dohme filed Critical Merck Sharp & Dohme
Application granted granted Critical
Publication of ATE197453T1 publication Critical patent/ATE197453T1/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/06—Antimigraine agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Pain & Pain Management (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Epoxy Resins (AREA)
  • Paints Or Removers (AREA)
  • Lubricants (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Steroid Compounds (AREA)
AT93907945T 1992-04-03 1993-03-29 Imidazol-, triazol- und tetrazolderivate ATE197453T1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB929207396A GB9207396D0 (en) 1992-04-03 1992-04-03 Therapeutic agents
PCT/GB1993/000652 WO1993020066A1 (en) 1992-04-03 1993-03-29 Imidazole, triazole and tetrazole derivatives

Publications (1)

Publication Number Publication Date
ATE197453T1 true ATE197453T1 (de) 2000-11-11

Family

ID=10713456

Family Applications (1)

Application Number Title Priority Date Filing Date
AT93907945T ATE197453T1 (de) 1992-04-03 1993-03-29 Imidazol-, triazol- und tetrazolderivate

Country Status (10)

Country Link
US (1) US5607957A (de)
EP (1) EP0637307B1 (de)
JP (1) JP3285581B2 (de)
AT (1) ATE197453T1 (de)
AU (1) AU675641B2 (de)
CA (1) CA2133076A1 (de)
DE (1) DE69329645T2 (de)
ES (1) ES2152948T3 (de)
GB (1) GB9207396D0 (de)
WO (1) WO1993020066A1 (de)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9420529D0 (en) * 1994-10-12 1994-11-30 Pfizer Ltd Indoles
US5484763A (en) * 1995-02-10 1996-01-16 American Cyanamid Company Substituted benzisoxazole and benzisothiazole herbicidal agents
EP1223932A4 (de) 1999-10-01 2003-01-15 Smithkline Beecham Corp Verbindungen und verfahren
US20030176454A1 (en) * 2000-05-15 2003-09-18 Akira Yamada N-coating heterocyclic compounds
CA2508290C (en) 2002-12-20 2017-02-28 Ciba Specialty Chemicals Holding Inc. Synthesis of amines and intermediates for the synthesis thereof
AU2013348167A1 (en) 2012-11-20 2015-05-28 Vertex Pharmaceuticals Incorporated Compounds useful as inhibitors of indoleamine 2,3-dioxygenase
US11220492B2 (en) 2017-05-17 2022-01-11 Arcus Biosciences, Inc. Quinazoline-pyrazole derivatives for the treatment of cancer-related disorders
GB201801226D0 (en) 2018-01-25 2018-03-14 Redx Pharma Plc Modulators of Rho-associated protein kinase
AU2022309017A1 (en) * 2021-07-07 2024-01-25 Terran Biosciences Inc. N,n-dimethyltryptamine and related psychedlics and uses thereof

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4785016A (en) * 1984-12-04 1988-11-15 Glaxo Group Limited Indole derivatives
US4833153A (en) * 1985-11-08 1989-05-23 Glaxo Group Limited Indole derivatives
GB8724912D0 (en) * 1987-10-23 1987-11-25 Wellcome Found Indole derivatives
US5225431A (en) * 1987-10-23 1993-07-06 Burroughs Wellcome Co. Therapeutic substituted indole compounds and compositions thereof
NZ227841A (en) * 1988-02-12 1991-08-27 Merck Sharp & Dohme Heterocyclic compounds with at least two non-condensed five membered rings and pharmaceutical compositions
IL96891A0 (en) * 1990-01-17 1992-03-29 Merck Sharp & Dohme Indole-substituted five-membered heteroaromatic compounds,their preparation and pharmaceutical compositions containing them
AU646871B2 (en) * 1990-06-07 1994-03-10 Astrazeneca Uk Limited Therapeutic heterocyclic compounds
EP0494774A1 (de) * 1991-01-11 1992-07-15 MERCK SHARP & DOHME LTD. Indazol-substituierte 5-Kettenglieder heteroaromatische Verbindungen
SK278998B6 (sk) * 1991-02-01 1998-05-06 Merck Sharp & Dohme Limited Deriváty imidazolu, triazolu a tetrazolu, spôsob i
UA41297C2 (uk) * 1991-11-25 2001-09-17 Пфайзер, Інк. Похідні індолу, фармацевтична композиція і спосіб лікування

Also Published As

Publication number Publication date
US5607957A (en) 1997-03-04
WO1993020066A1 (en) 1993-10-14
ES2152948T3 (es) 2001-02-16
AU3895693A (en) 1993-11-08
EP0637307B1 (de) 2000-11-08
GB9207396D0 (en) 1992-05-13
EP0637307A1 (de) 1995-02-08
DE69329645D1 (de) 2000-12-14
DE69329645T2 (de) 2001-05-10
AU675641B2 (en) 1997-02-13
JP3285581B2 (ja) 2002-05-27
JPH07505382A (ja) 1995-06-15
CA2133076A1 (en) 1993-10-14

Similar Documents

Publication Publication Date Title
IL109337A0 (en) Indole derivatives for use in migraine
DE69324140D1 (de) Kondensierte imidazol- und triazolderivate als 5-hta rezeptoragonisten
DE69125731D1 (de) Indol-substituierte heteroaromatische Verbindungen
ES2083595T3 (es) Derivados de indol que inhiben la biosintesis de leucotrienos.
EP0860168A3 (de) Verwendung von Agonisten des zentralen Cannabinoid-Rezeptors CB1
ES2121193T3 (es) Derivados de bencimidazoles.
GR3015313T3 (en) Indole derivatives as antiallergy and antiinflammatory agents.
NZ290387A (en) Substituted 1,2,4-triazole derivatives
DE69329645D1 (de) Imidazol-, triazol- und tetrazolderivate
ES2127789T3 (es) Derivados de 1,2,4-triazol 4-sustituidos.
ES2116411T3 (es) La sal sulfato de un triazol sustituido, composiciones farmaceuticas de la misma y su uso en terapia
DE69301357D1 (de) Indol derivate als "5-ht1-like" agonisten
BR9507926A (pt) Endoparasiticidas
AU5614198A (en) Isoquinolinamine and phthalazinamine derivatives which interact with crf receptors
FI953002A0 (fi) Menetelmä kroonisen eturauhastulehduksen hoitamiseksi 17beta-N-monosubstituoiduilla karbamoyyli-4-atsa-5alfa-androst-1-en-3-oneilla
MY108739A (en) Imidazole, triazole and tetrazole derivatives
SE9404438D0 (sv) New process
DE69310721D1 (de) Zuckerderivate von makroliden
MY110795A (en) The sulphate salt of a substituted triazole, pharmaceutical compositions thereof, and their use in therapy
IS1783B (is) Aðferð við framleiðslu á 1,2,3,9-tetrahýdró-9-metýl-3-[(2-metýl-1H-imídazól-1-ýl)metýl]-4H-karbasól-4-ón
AU5269696A (en) Anellated beta-carbolines

Legal Events

Date Code Title Description
RER Ceased as to paragraph 5 lit. 3 law introducing patent treaties