AT89201B - Process for the preparation of tropinone monocarboxylic acid esters. - Google Patents

Process for the preparation of tropinone monocarboxylic acid esters.

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Publication number
AT89201B
AT89201B AT89201DA AT89201B AT 89201 B AT89201 B AT 89201B AT 89201D A AT89201D A AT 89201DA AT 89201 B AT89201 B AT 89201B
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AT
Austria
Prior art keywords
acid esters
preparation
tropinone
monocarboxylic acid
tropinone monocarboxylic
Prior art date
Application number
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German (de)
Original Assignee
Merck Ag E
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
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Publication date
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Publication of AT89201B publication Critical patent/AT89201B/en

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Description

  

   <Desc/Clms Page number 1> 
 



  Verfahren zur Darstellung von Tropinonmonocarbonsäureestern. 



     Im #Journal of the Chemical Society" Band   111/112, (1917), S. 762 u.   ff.,   ist von Robert Robinson ein Verfahren zur   Darstemmg   von Tropinon beschrieben worden.   Es   besteht darin, dass man Succindialdehyd mit Salzen oder   Eltern der Aeetondicarbonsäure   und mit Methylamin kondensiert und die Reaktionsprodukte durch Abspaltung der Carboxyl-bzw. Estergruppen in Tropinon   überführt.   



   Der Übergang zu Tropinonmonocarbonsäureestern, welche bekanntlich erhebliche technische Bedeutung besitzen,   begegnet nach dem erwähnten   Verfahren Schwierigkeiten, insofern als die Reindarstellung von Monocarbonsäureester durch die Bildung von Tropinon als Nebenprodukt technisch schwer ausführbar ist. 



   Es wurde nun die neue und wichtige Beobachtung gemacht, dass man Tropinonmonocarbon-   säureester erhält, wenn   man von der Acetondicarbonestersäure ausgeht und deren Salze mit Succindialdehyd und Methylamin kondensiert. Das Kondensationsprodukt spaltet sehr leicht Kohlensäure ab und liefert   Tropinonmonoearbonsäureester   gemäss der Reaktionsgleichung : 
 EMI1.1 
 Beispiel : Man stellt   (nach Harries,   Ber. 34   1 [1901],   S. 1494) eine etwa   10% igue   Lösung von 
 EMI1.2 
 

**WARNUNG** Ende DESC Feld kannt Anfang CLMS uberlappen**.



   <Desc / Clms Page number 1>
 



  Process for the preparation of tropinone monocarboxylic acid esters.



     In the # Journal of the Chemical Society "Volume 111/112, (1917), p. 762 et seq., Robert Robinson has described a process for the preparation of tropinone. It consists in that succinic dialdehyde is mixed with salts or parents of the Aeetondicarboxylic acid and condensed with methylamine and the reaction products are converted into tropinone by splitting off the carboxyl or ester groups.



   The transition to tropinone monocarboxylic acid esters, which are known to be of considerable industrial importance, encounters difficulties after the process mentioned, insofar as the pure preparation of monocarboxylic acid esters through the formation of tropinone as a by-product is difficult to carry out industrially.



   The new and important observation has now been made that tropinone monocarboxylic acid esters are obtained when starting from acetone dicarboxylic acid and condensing its salts with succinic dialdehyde and methylamine. The condensation product splits off carbonic acid very easily and gives tropinone monoarboxylic acid ester according to the reaction equation:
 EMI1.1
 Example: According to Harries, Ber. 34 1 [1901], p. 1494, an approximately 10% solution of
 EMI1.2
 

** WARNING ** End of DESC field may overlap beginning of CLMS **.

 

Claims (1)

**WARNUNG** Ende CLMS Feld Kannt Anfang DESC uberlappen**. ** WARNING ** End of CLMS field may overlap beginning of DESC **.
AT89201D 1919-08-23 1920-10-20 Process for the preparation of tropinone monocarboxylic acid esters. AT89201B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE89201X 1919-08-23

Publications (1)

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AT89201B true AT89201B (en) 1922-08-25

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ID=5642648

Family Applications (1)

Application Number Title Priority Date Filing Date
AT89201D AT89201B (en) 1919-08-23 1920-10-20 Process for the preparation of tropinone monocarboxylic acid esters.

Country Status (1)

Country Link
AT (1) AT89201B (en)

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