AT254187B - Verfahren zur Herstellung von neuen bicyclischen Pyrazolverbindungen - Google Patents

Verfahren zur Herstellung von neuen bicyclischen Pyrazolverbindungen

Info

Publication number
AT254187B
AT254187B AT818165A AT818165A AT254187B AT 254187 B AT254187 B AT 254187B AT 818165 A AT818165 A AT 818165A AT 818165 A AT818165 A AT 818165A AT 254187 B AT254187 B AT 254187B
Authority
AT
Austria
Prior art keywords
preparation
pyrazole compounds
new bicyclic
bicyclic pyrazole
new
Prior art date
Application number
AT818165A
Other languages
English (en)
Original Assignee
Ciba Geigy
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US395016A external-priority patent/US3340269A/en
Application filed by Ciba Geigy filed Critical Ciba Geigy
Application granted granted Critical
Publication of AT254187B publication Critical patent/AT254187B/de

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
AT818165A 1964-09-08 1965-09-07 Verfahren zur Herstellung von neuen bicyclischen Pyrazolverbindungen AT254187B (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US395016A US3340269A (en) 1964-09-08 1964-09-08 1-substituted 4-acyl-2, 3-dioxo-piperidine
US432416A US3365459A (en) 1964-09-08 1965-02-12 Certain tetrahydro pyrazolo-pyridine and pyrazolo-piperidine derivatives

Publications (1)

Publication Number Publication Date
AT254187B true AT254187B (de) 1967-05-10

Family

ID=27014961

Family Applications (1)

Application Number Title Priority Date Filing Date
AT818165A AT254187B (de) 1964-09-08 1965-09-07 Verfahren zur Herstellung von neuen bicyclischen Pyrazolverbindungen

Country Status (6)

Country Link
US (1) US3365459A (de)
AT (1) AT254187B (de)
BE (1) BE669298A (de)
ES (1) ES317146A1 (de)
FR (2) FR5155M (de)
NL (1) NL6511645A (de)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR6121M (de) * 1966-01-12 1968-06-17
RU2131876C1 (ru) * 1993-07-06 1999-06-20 Пфайзер Инк. Бициклические тетрагидропиразолпиридины или их фармацевтически приемлемые соли, фармацевтическая композиция, способ ингибирования фосфодиэстеразы, способ лечения
US5508300A (en) * 1994-01-14 1996-04-16 Pfizer Inc. Dihydro pyrazolopyrroles, compositions and use
PL319758A1 (en) * 1994-10-20 1997-08-18 Pfizer Bicyclic tetrahydropyrasole pyridines and their application as medicines
DK1140941T3 (da) 1998-12-23 2005-02-14 Bristol Myers Squibb Pharma Co Nitrogenholdige heterobicykliske forbindelser som faktor Xa-inhibitorer
US6858616B2 (en) * 1998-12-23 2005-02-22 Bristol-Myers Squibb Pharma Company Nitrogen containing heterobicycles as factor Xa inhibitors
US6998408B2 (en) * 2001-03-23 2006-02-14 Bristol-Myers Squibb Pharma Company 6-5, 6-6, or 6-7 Heterobicycles as factor Xa inhibitors
US6960595B2 (en) * 2001-03-23 2005-11-01 Bristol-Myers Squibb Pharma Company 5-6 to 5-7 Heterobicycles as factor Xa inhibitors
WO2002085353A1 (en) 2001-04-18 2002-10-31 Bristol-Myers Squibb Company 1,4,5,6-tetrahydropyrazolo-[3,4-c]-pyridin-7-ones as factor xa inhibitors
WO2002085356A1 (en) 2001-04-18 2002-10-31 Bristol-Myers Squibb Company 1, 4, 5, 6-tetrahydropyrazolo-[3, 4-c]-pyrid in-7-ones as factor xa inhibitors
TWI331526B (en) * 2001-09-21 2010-10-11 Bristol Myers Squibb Pharma Co Lactam-containing compounds and derivatives thereof as factor xa inhibitors
CA2726702A1 (en) 2001-09-21 2003-04-03 Bristol-Myers Squibb Company Lactam-containing compounds and derivatives thereof as factor xa inhibitors
TW200302225A (en) * 2001-12-04 2003-08-01 Bristol Myers Squibb Co Substituted amino methyl factor Xa inhibitors
WO2003048081A2 (en) * 2001-12-04 2003-06-12 Bristol-Myers Squibb Company Glycinamides as factor xa inhibitors
AU2003273179A1 (en) * 2002-05-10 2003-12-12 Bristol-Myers Squibb Company 1,1-disubstituted cycloalkyl derivatives as factor xa inhibitors
US7122557B2 (en) * 2003-03-18 2006-10-17 Bristol-Myers Squibb Company Sulfonyl-amidino-containing and tetrahydropyrimidino-containing compounds as factor Xa inhibitors
US20040214856A1 (en) * 2003-04-23 2004-10-28 Pfizer Inc Cannabinoid receptor ligands and uses thereof
US7145012B2 (en) * 2003-04-23 2006-12-05 Pfizer Inc. Cannabinoid receptor ligands and uses thereof

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB964750A (en) * 1961-09-08 1964-07-22 Ciba Ltd New pyrazolo-pyridines
BE620332A (de) * 1961-09-08 1900-01-01

Also Published As

Publication number Publication date
US3365459A (en) 1968-01-23
FR5155M (de) 1967-06-12
NL6511645A (de) 1966-03-09
BE669298A (de) 1966-03-07
ES317146A1 (es) 1966-08-01
FR4903M (de) 1965-03-13

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