AR223334A1 - Procedimiento para la preparacion de glicosidos de esteroides y espiro-cetalesteroides,y sus esteres,de actividad inhibitoria de las sintetasas de las prostaglandinas - Google Patents

Procedimiento para la preparacion de glicosidos de esteroides y espiro-cetalesteroides,y sus esteres,de actividad inhibitoria de las sintetasas de las prostaglandinas

Info

Publication number
AR223334A1
AR223334A1 AR274988A AR27498878A AR223334A1 AR 223334 A1 AR223334 A1 AR 223334A1 AR 274988 A AR274988 A AR 274988A AR 27498878 A AR27498878 A AR 27498878A AR 223334 A1 AR223334 A1 AR 223334A1
Authority
AR
Argentina
Prior art keywords
syntheases
prostaglandinas
cetalesteroides
glycosides
steroids
Prior art date
Application number
AR274988A
Other languages
English (en)
Spanish (es)
Original Assignee
Roecar Holdings Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Roecar Holdings Nv filed Critical Roecar Holdings Nv
Application granted granted Critical
Publication of AR223334A1 publication Critical patent/AR223334A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/70Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7028Compounds having saccharide radicals attached to non-saccharide compounds by glycosidic linkages
    • A61K31/7034Compounds having saccharide radicals attached to non-saccharide compounds by glycosidic linkages attached to a carbocyclic compound, e.g. phloridzin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/70Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7028Compounds having saccharide radicals attached to non-saccharide compounds by glycosidic linkages
    • A61K31/7034Compounds having saccharide radicals attached to non-saccharide compounds by glycosidic linkages attached to a carbocyclic compound, e.g. phloridzin
    • A61K31/704Compounds having saccharide radicals attached to non-saccharide compounds by glycosidic linkages attached to a carbocyclic compound, e.g. phloridzin attached to a condensed carbocyclic ring system, e.g. sennosides, thiocolchicosides, escin, daunorubicin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J17/00Normal steroids containing carbon, hydrogen, halogen or oxygen, having an oxygen-containing hetero ring not condensed with the cyclopenta(a)hydrophenanthrene skeleton
    • C07J17/005Glycosides
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J71/00Steroids in which the cyclopenta(a)hydrophenanthrene skeleton is condensed with a heterocyclic ring
    • C07J71/0005Oxygen-containing hetero ring

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Molecular Biology (AREA)
  • Epidemiology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
AR274988A 1977-12-31 1978-12-28 Procedimiento para la preparacion de glicosidos de esteroides y espiro-cetalesteroides,y sus esteres,de actividad inhibitoria de las sintetasas de las prostaglandinas AR223334A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19772759171 DE2759171A1 (de) 1977-12-31 1977-12-31 Arzneimittel mit wirkung als prostaglandinsynthetaseninhibitor

Publications (1)

Publication Number Publication Date
AR223334A1 true AR223334A1 (es) 1981-08-14

Family

ID=6027873

Family Applications (1)

Application Number Title Priority Date Filing Date
AR274988A AR223334A1 (es) 1977-12-31 1978-12-28 Procedimiento para la preparacion de glicosidos de esteroides y espiro-cetalesteroides,y sus esteres,de actividad inhibitoria de las sintetasas de las prostaglandinas

Country Status (19)

Country Link
JP (1) JPS54101436A (enrdf_load_stackoverflow)
AR (1) AR223334A1 (enrdf_load_stackoverflow)
AU (1) AU516933B2 (enrdf_load_stackoverflow)
BE (1) BE873222A (enrdf_load_stackoverflow)
CA (1) CA1113006A (enrdf_load_stackoverflow)
CH (1) CH637829A5 (enrdf_load_stackoverflow)
DE (1) DE2759171A1 (enrdf_load_stackoverflow)
DK (1) DK587778A (enrdf_load_stackoverflow)
ES (1) ES476443A1 (enrdf_load_stackoverflow)
FR (1) FR2425859A1 (enrdf_load_stackoverflow)
GB (1) GB2039217B (enrdf_load_stackoverflow)
IL (1) IL56345A (enrdf_load_stackoverflow)
IT (1) IT1109336B (enrdf_load_stackoverflow)
LU (1) LU80739A1 (enrdf_load_stackoverflow)
NL (1) NL7812656A (enrdf_load_stackoverflow)
NZ (1) NZ189297A (enrdf_load_stackoverflow)
PT (1) PT69012A (enrdf_load_stackoverflow)
SE (1) SE466683B (enrdf_load_stackoverflow)
ZA (1) ZA787399B (enrdf_load_stackoverflow)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2926463A1 (de) * 1978-07-05 1980-01-24 Roecar Holdings Nv Spiroketaline und ihre verwendung
JPS5874619A (ja) * 1981-10-29 1983-05-06 Nippon Shinyaku Co Ltd リポソ−ム及びその製法
IE54837B1 (en) 1982-04-19 1990-02-28 Roecar Holdings Nv Extract of plants of the family of hypoxidaceae for treatment of cancer
US4602003A (en) * 1982-05-17 1986-07-22 Medical Research Foundation Of Oregon Synthetic compounds to inhibit intestinal absorption of cholesterol in the treatment of hypercholesterolemia
US4602005A (en) * 1982-05-17 1986-07-22 Medical Research Foundation Of Oregon Tigogenin cellobioside for treating hypercholesterolemia and atherosclerosis
DE3401178A1 (de) * 1984-01-14 1985-07-18 Roecar Holdings (Netherlands Antilles) N.V., Willemstad, Curacao, Niederländische Antillen Verwendung von phytosterolglykosiden zur behandlung erhoehter 5(6)(alpha)-epoxicholesterolspiegel
DE3416112A1 (de) * 1984-04-30 1985-10-31 Roecar Holdings (Netherlands Antilles) N.V., Willemstad, Curacao, Niederländische Antillen Verwendung von sterolinen und spiroketalinen als lipoxygenaseregulatoren
DE3829641A1 (de) * 1988-09-01 1990-03-15 Roecar Holdings Nv Transdermal anwendbare pharmazeutische zubereitungen mit sterolinen und/oder spiroketalinen
DE3829640C1 (enrdf_load_stackoverflow) * 1988-09-01 1990-04-26 Roecar Holdings (Netherlands Antilles) N.V., Willemstad, Curacao, Niederlaendische Antillen, Nl
DE3829643A1 (de) * 1988-09-01 1990-03-15 Roecar Holdings Nv Phyto- und zoosterole und deren derivate mit verbesserter wasserloeslichkeit
US5166194A (en) * 1988-09-01 1992-11-24 Roecar Holdings Transdermally applicable pharmaceutical preparations having a pharmaceutically usable glycoside content
DE3838716A1 (de) * 1988-11-15 1990-05-17 Kanoldt Arzneimittel Gmbh Arzneimittelzubereitung aus esterderivaten des hecogenins und dessen verwendung zur behandlung von benigner prostatahyperplasie
US5502038A (en) * 1993-06-21 1996-03-26 Medical Research Foundation Of Oregon Cholesterol sequestrant glycosides that inhibit intestinal cholesterol absorption

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IE35018B1 (en) * 1970-03-18 1975-10-15 Liebenberg R W Therapeutic agent
US3966918A (en) * 1973-12-12 1976-06-29 Nippon Shinyaku Co., Ltd. Method of preparing aqueous solutions of sterol glycosides and their ester derivatives
JPS51118817A (en) * 1975-04-08 1976-10-19 Nippon Shinyaku Co Ltd A process for preparing absorbable steroid glycoside pharmaceutical

Also Published As

Publication number Publication date
AU516933B2 (en) 1981-07-02
ZA787399B (en) 1980-01-30
DK587778A (da) 1979-07-01
DE2759171A1 (de) 1979-07-12
GB2039217A (en) 1980-08-06
IL56345A0 (en) 1979-03-12
PT69012A (pt) 1979-01-01
JPS54101436A (en) 1979-08-10
SE7813443L (sv) 1979-07-01
FR2425859B1 (enrdf_load_stackoverflow) 1983-04-08
DE2759171C2 (enrdf_load_stackoverflow) 1990-10-25
IL56345A (en) 1984-11-30
AU4302478A (en) 1979-07-05
CA1113006A (en) 1981-11-24
SE466683B (sv) 1992-03-23
GB2039217B (en) 1982-08-04
ES476443A1 (es) 1979-10-16
IT1109336B (it) 1985-12-16
CH637829A5 (de) 1983-08-31
NZ189297A (en) 1984-10-19
NL7812656A (nl) 1979-07-03
BE873222A (fr) 1979-06-29
IT7852493A0 (it) 1978-12-29
FR2425859A1 (fr) 1979-12-14
LU80739A1 (de) 1980-01-22

Similar Documents

Publication Publication Date Title
AR220704A1 (es) Procedimiento para la preparacion de derivados de indanil y tetrahidronaftil octatrieno
MX5502E (es) Procedimiento para la preparacion de eteres y esteres de oximas
MX5950E (es) Procedimiento para la preparacion de derivados de la pirrolidin-2-ona
TR20779A (tr) Suebtitueye fenoksibenz loksi karbonil tuerevleri,bunlarin hazirlanisi icin usul ve bunlarin ensektisidler ve akarisidler olarak kullanilmalar
AR218948A1 (es) Procedimiento para la obtencion de preparaciones activas de enestesia local
MX5527E (es) Procedimiento para la preparacion de derivados de carboestirilo
MX5951E (es) Procedimiento para la preparacion de derivados de benzoimidazol
AR219734A1 (es) Procedimiento para la preparacion de derivados de (4-hidroxipirrolidin-2-on-1-il)-acilamida
AR223154A1 (es) Nuevos 3-hidroxidifenileteres desprovistos de actividad terapeutica,procedimiento para su obtencion y su aplicacion
MX4278E (es) Procedimiento para la preparacion de glicosidos de antraciclina
AR223334A1 (es) Procedimiento para la preparacion de glicosidos de esteroides y espiro-cetalesteroides,y sus esteres,de actividad inhibitoria de las sintetasas de las prostaglandinas
IT1097592B (it) Procedimento per la preparazione di isocianati da formammidi
MX6053E (es) Procedimiento microbiologico para la preparacion de derivados del sesquiterpeno
ES498607A0 (es) Procedimiento para la preparacion de nuevos esteres de azu- car y glicosidos
MX5479E (es) Procedimiento para la preparacion de derivados de 1-oxadetiacefalosporinas
IT7848752A0 (it) Tramezzo smontabile e procedimento per montarlo
MX5811E (es) Procedimiento para la preparacion de medios de cultivo micologicos
AR218296A1 (es) Procedimiento para la preparacion de nuevos derivados de 14-beta-amino-morfina
AR222815A1 (es) Procedimiento para la preparacion de acidos(alfa-trifluorometil-mercapto-propionil)-pirrolidinil-o tiazolidinil-carboxilicos
AR222844A1 (es) Procedimiento para la obtencion de nuevos derivados de n1-glucofuranosil-6-ilo-n3-nitroso-ureas
AR221215A1 (es) Procedimiento para la preparacion de cloroacetanilidas substituidas
MX5672E (es) Procedimiento para la preparacion de acidos 2-piridil y 2-pirimidil-aminobenzoicos
MX4884E (es) Procedimiento para la preparacion de derivados de la tienopiridina
MX5382E (es) Procedimiento para la preparacion de alcohol alfa-trifluoro-metil-3-fenoxibencilico
MX5530E (es) Procedimiento para la preparacion de dl-fenilglicinamida