AR219948A1 - Procedimiento para obtener nuevos 7-azabenzimidazoles con cadenas laterales basicas y sus sales - Google Patents
Procedimiento para obtener nuevos 7-azabenzimidazoles con cadenas laterales basicas y sus salesInfo
- Publication number
- AR219948A1 AR219948A1 AR273835A AR27383578A AR219948A1 AR 219948 A1 AR219948 A1 AR 219948A1 AR 273835 A AR273835 A AR 273835A AR 27383578 A AR27383578 A AR 27383578A AR 219948 A1 AR219948 A1 AR 219948A1
- Authority
- AR
- Argentina
- Prior art keywords
- azabenzimidazoles
- salts
- procedure
- side chains
- obtain new
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/72—Nitrogen atoms
- C07D213/74—Amino or imino radicals substituted by hydrocarbon or substituted hydrocarbon radicals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/72—Nitrogen atoms
- C07D213/75—Amino or imino radicals, acylated by carboxylic or carbonic acids, or by sulfur or nitrogen analogues thereof, e.g. carbamates
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB3991977 | 1977-09-26 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AR219948A1 true AR219948A1 (es) | 1980-09-30 |
Family
ID=10412196
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AR273835A AR219948A1 (es) | 1977-09-26 | 1978-09-25 | Procedimiento para obtener nuevos 7-azabenzimidazoles con cadenas laterales basicas y sus sales |
Country Status (20)
| Country | Link |
|---|---|
| US (1) | US4247556A (no) |
| JP (1) | JPS5455595A (no) |
| AR (1) | AR219948A1 (no) |
| AT (1) | AT365188B (no) |
| BE (1) | BE870709A (no) |
| CA (1) | CA1103673A (no) |
| DD (1) | DD139579A5 (no) |
| DE (1) | DE2841209A1 (no) |
| DK (1) | DK424678A (no) |
| EG (1) | EG13604A (no) |
| ES (1) | ES473201A1 (no) |
| FI (1) | FI782909A (no) |
| FR (1) | FR2404009A1 (no) |
| IT (1) | IT7851230A0 (no) |
| NL (1) | NL7809713A (no) |
| NO (1) | NO783239L (no) |
| PT (1) | PT68584A (no) |
| SE (1) | SE7810050L (no) |
| SU (1) | SU795478A3 (no) |
| ZA (1) | ZA785430B (no) |
Families Citing this family (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| KR950001015B1 (ko) * | 1986-01-10 | 1995-02-07 | 닛뽕 케미화 가부시끼가이샤 | 술폭시드 유도체의 제조방법 |
| US4772600A (en) * | 1986-06-09 | 1988-09-20 | A. H. Robins Company, Inc. | Fused imidazoheterocyclic compounds and pharmaceutical compositions |
| UA72448C2 (en) | 1997-09-26 | 2005-03-15 | Zentaris Gmbh | Azabenzimidazole-based compounds, methods for their synthesis and pharmaceutical composition, method for modulating function of serine/threonine protein kinases with azabenzimidazole-based compounds, method for identifying compounds modulating functioning of serine/threonine protein kinase, method for preventing and treating serine/threonine protein kinase-related abnormal conditions with azabenzimidazole-based compounds |
| FR2832148B1 (fr) * | 2001-11-14 | 2004-05-21 | Oreal | Nouvelles bases d'oxydation 2,5-diaminopyridine utiles pour la teinture des fibres keratiniques |
| US20090281075A1 (en) * | 2006-02-17 | 2009-11-12 | Pharmacopeia, Inc. | Isomeric purinones and 1h-imidazopyridinones as pkc-theta inhibitors |
| US7989459B2 (en) | 2006-02-17 | 2011-08-02 | Pharmacopeia, Llc | Purinones and 1H-imidazopyridinones as PKC-theta inhibitors |
| US7902187B2 (en) | 2006-10-04 | 2011-03-08 | Wyeth Llc | 6-substituted 2-(benzimidazolyl)purine and purinone derivatives for immunosuppression |
| CL2007002867A1 (es) | 2006-10-04 | 2008-06-27 | Pharmacopeia Inc | Compuestos derivados de 2-(bencimidazolil)purina, inhibidores de janus quinasa 3; composicion farmaceutica que los contiene; y su uso para tratar enfermedades autoinmune, inflamatorias, cardiovasculares, rechazo de implante, entre otras. |
| CL2007002866A1 (es) | 2006-10-04 | 2008-07-04 | Pharmacopeia Inc | Compuestos derivados de 6-sustituidos-2-(bencimidazolil) purina y purinona; composicion farmaceutica que comprende a dicho compuesto; y uso del compuesto en el tratamiento de enfermedades autoinmunes, enfermedad inflamatoria, enfermedad mediada por m |
| ES2885424T3 (es) | 2013-03-15 | 2021-12-13 | Knopp Biosciences Llc | Imidazo(4,5-B)piridin-2-il amidas como activadores del canal Kv7 |
| LT3572405T (lt) | 2014-09-12 | 2023-10-25 | Biohaven Therapeutics Ltd. | Benzoimidazol-1,2-ilo amidai, kaip kv7 kanalų aktyvatoriai |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3004978A (en) * | 1961-10-17 | Certain i-tert-amino lower alkyl | ||
| US2987518A (en) * | 1958-12-10 | 1961-06-06 | Ciba Pharmacentical Products I | Certain 1h [4, 5-c]-imidazopyridines |
| CH386438A (de) * | 1959-03-18 | 1965-01-15 | Ciba Geigy | Verfahren zur Herstellung neuer 7-Aza-benzimidazole |
| US3719683A (en) * | 1970-11-20 | 1973-03-06 | Ciba Geigy Corp | Imidazo(4,5-b)pyridines |
| US4002623A (en) * | 1974-08-07 | 1977-01-11 | Pfizer Inc. | Anti-inflammatory 1-[3-(dialkylamino)propyl]-2-acylaminobenzimidazoles and 2-acylamino-3-[3-(dialkylamino)-propyl]imidazo[4,5-b]pyridines |
| US4059584A (en) * | 1974-08-07 | 1977-11-22 | Pfizer | 2-Acylamino-3-[3-(dialkylamino)propyl]imidazo[4,5-b]pyridines |
| SE422799B (sv) * | 1975-05-28 | 1982-03-29 | Merck & Co Inc | Analogiforfarande for framstellning av 1,3-dihydroimidazo (4,5-b)pyridin-2-oner |
-
1978
- 1978-09-08 ES ES473201A patent/ES473201A1/es not_active Expired
- 1978-09-13 FR FR7826249A patent/FR2404009A1/fr active Granted
- 1978-09-19 SU SU782664732A patent/SU795478A3/ru active
- 1978-09-20 DD DD78207957A patent/DD139579A5/de unknown
- 1978-09-22 PT PT68584A patent/PT68584A/pt unknown
- 1978-09-22 DE DE19782841209 patent/DE2841209A1/de not_active Withdrawn
- 1978-09-22 BE BE6046611A patent/BE870709A/xx unknown
- 1978-09-25 NO NO783239A patent/NO783239L/no unknown
- 1978-09-25 AR AR273835A patent/AR219948A1/es active
- 1978-09-25 AT AT0690278A patent/AT365188B/de not_active IP Right Cessation
- 1978-09-25 CA CA312,055A patent/CA1103673A/en not_active Expired
- 1978-09-25 NL NL7809713A patent/NL7809713A/xx not_active Application Discontinuation
- 1978-09-25 FI FI782909A patent/FI782909A/fi unknown
- 1978-09-25 SE SE7810050A patent/SE7810050L/xx unknown
- 1978-09-25 ZA ZA00785430A patent/ZA785430B/xx unknown
- 1978-09-25 IT IT7851230A patent/IT7851230A0/it unknown
- 1978-09-25 DK DK424678A patent/DK424678A/da unknown
- 1978-09-26 EG EG576/78A patent/EG13604A/xx active
- 1978-09-26 JP JP11753778A patent/JPS5455595A/ja active Pending
-
1979
- 1979-01-15 US US06/003,385 patent/US4247556A/en not_active Expired - Lifetime
Also Published As
| Publication number | Publication date |
|---|---|
| AT365188B (de) | 1981-12-28 |
| JPS5455595A (en) | 1979-05-02 |
| ZA785430B (en) | 1979-09-26 |
| ES473201A1 (es) | 1979-03-16 |
| SU795478A3 (ru) | 1981-01-07 |
| CA1103673A (en) | 1981-06-23 |
| DD139579A5 (de) | 1980-01-09 |
| ATA690278A (de) | 1981-05-15 |
| DK424678A (da) | 1979-03-27 |
| US4247556A (en) | 1981-01-27 |
| FR2404009B1 (no) | 1981-09-18 |
| BE870709A (fr) | 1979-03-22 |
| DE2841209A1 (de) | 1979-04-05 |
| IT7851230A0 (it) | 1978-09-25 |
| FR2404009A1 (fr) | 1979-04-20 |
| FI782909A (fi) | 1979-03-27 |
| SE7810050L (sv) | 1979-03-27 |
| PT68584A (de) | 1978-10-01 |
| EG13604A (en) | 1982-03-31 |
| NO783239L (no) | 1979-03-27 |
| NL7809713A (nl) | 1979-03-28 |
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